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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-methyl-5-[[(2R)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C16H27N3O3
6-methyl-5-[[(2R)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(2R)-1-pyridin-4-ylpropan-2-yl]pyrimidin-2-amine —— C19H21N5
4-(2,6-dimethylpyridin-3-yl)-N-[(2R)-1-pyridin-4-ylpropan-2-yl]pyrimidin-2-amine
—— 2-methyl-5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]pyrazine —— C13H16N4O
2-methyl-5-[[2-[(3R)-oxolan-3-yl]imidazol-1-yl]methyl]pyrazine
—— 2-methyl-5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]pyrazine —— C13H16N4O
2-methyl-5-[[2-[(3S)-oxolan-3-yl]imidazol-1-yl]methyl]pyrazine
—— 5-[[(2S)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C15H25N3O3
5-[[(2S)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione
—— N-[(3S)-oxolan-3-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C11H14F3N3O
N-[(3S)-oxolan-3-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 7-[(2R)-2-methyloxolane-2-carbonyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H20N4O3
7-[(2R)-2-methyloxolane-2-carbonyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-[(3R)-oxolan-3-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C11H14F3N3O
N-[(3R)-oxolan-3-yl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 7-[(2R)-2-pyrazol-1-ylbutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2R)-2-pyrazol-1-ylbutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (3R)-N,N-diethyl-1-(2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide —— C22H30N6O
(3R)-N,N-diethyl-1-(2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide
—— 7-[(2S)-2-pyrazol-1-ylbutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2S)-2-pyrazol-1-ylbutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 3-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]-5-[2-[(2R)-piperidin-2-yl]ethyl]phenol —— C22H31N5O
3-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]-5-[2-[(2R)-piperidin-2-yl]ethyl]phenol
—— morpholin-4-yl-[(3S)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone —— C20H29N5O3
morpholin-4-yl-[(3S)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone
—— 3-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]-5-[2-[(2S)-piperidin-2-yl]ethyl]phenol —— C22H31N5O
3-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]-5-[2-[(2S)-piperidin-2-yl]ethyl]phenol
—— 4-cyclobutyl-N-[(3R)-1-ethylpiperidin-3-yl]-6-methylpyrimidin-2-amine —— C16H26N4
4-cyclobutyl-N-[(3R)-1-ethylpiperidin-3-yl]-6-methylpyrimidin-2-amine
—— 4-cyclobutyl-N-[(3S)-1-ethylpiperidin-3-yl]-6-methylpyrimidin-2-amine —— C16H26N4
4-cyclobutyl-N-[(3S)-1-ethylpiperidin-3-yl]-6-methylpyrimidin-2-amine
—— 1-[4-[[(3R)-1-methylpiperidin-3-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H26N6O
1-[4-[[(3R)-1-methylpiperidin-3-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— (3S)-N,N-diethyl-1-(2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide —— C22H30N6O
(3S)-N,N-diethyl-1-(2-pyridin-4-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidin-4-yl)piperidine-3-carboxamide
—— 1-[4-[[(3S)-1-methylpiperidin-3-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H26N6O
1-[4-[[(3S)-1-methylpiperidin-3-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 2-methyl-5-[(3S)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C20H25N3O2
2-methyl-5-[(3S)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— 7-[(2S)-2-methyloxolane-2-carbonyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H20N4O3
7-[(2S)-2-methyloxolane-2-carbonyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2S)-2-methyloxolane-2-carbonyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H20N4O3
7-[(2S)-2-methyloxolane-2-carbonyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2R)-2-methyloxolane-2-carbonyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H20N4O3
7-[(2R)-2-methyloxolane-2-carbonyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— morpholin-4-yl-[(3R)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone —— C20H29N5O3
morpholin-4-yl-[(3R)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone
—— 7-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2R)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 2-methyl-5-[(3R)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one —— C20H25N3O2
2-methyl-5-[(3R)-3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidin-6-one
—— [(2S)-2-(4-methylpentyl)morpholin-4-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone —— C20H26N4O2
[(2S)-2-(4-methylpentyl)morpholin-4-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone
—— 7-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2S)-2-methyl-3-pyrazol-1-ylpropanoyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— [(2R)-2-(4-methylpentyl)morpholin-4-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone —— C20H26N4O2
[(2R)-2-(4-methylpentyl)morpholin-4-yl]-(2-pyridin-3-ylpyrimidin-5-yl)methanone
—— 4-[(1R)-1-[4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl]ethyl]morpholine —— C23H26N4O
4-[(1R)-1-[4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl]ethyl]morpholine
—— [(3R)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone —— C21H31N5O3
[(3R)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone
—— 1-[(3R)-1-[[2-(propylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]pyrrolidin-2-one —— C17H27N5O
1-[(3R)-1-[[2-(propylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]pyrrolidin-2-one
—— 6-(2-methoxyphenyl)-N-[[(2S)-oxan-2-yl]methyl]pyridazin-3-amine —— C17H21N3O2
6-(2-methoxyphenyl)-N-[[(2S)-oxan-2-yl]methyl]pyridazin-3-amine
—— 4-[(1S)-1-[4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl]ethyl]morpholine —— C23H26N4O
4-[(1S)-1-[4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl]ethyl]morpholine
—— [(3R)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone —— C22H30N4O
[(3R)-3-[2-(2-methylphenyl)ethyl]piperidin-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrimidin-2-amine —— C20H19N7O
4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)ethyl]pyrimidin-2-amine
—— 6-(2-methoxyphenyl)-N-[[(2R)-oxan-2-yl]methyl]pyridazin-3-amine —— C17H21N3O2
6-(2-methoxyphenyl)-N-[[(2R)-oxan-2-yl]methyl]pyridazin-3-amine
—— [(3S)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone —— C21H31N5O3
[(3S)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone
—— 1-[(3S)-1-[[2-(propylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]pyrrolidin-2-one —— C17H27N5O
1-[(3S)-1-[[2-(propylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]pyrrolidin-2-one
—— 4-cyclopentyl-N-[(1S)-1-pyridin-2-ylpropyl]pyrimidin-2-amine —— C17H22N4
4-cyclopentyl-N-[(1S)-1-pyridin-2-ylpropyl]pyrimidin-2-amine
—— 4-cyclobutyl-N-[[(3S)-1-ethylpiperidin-3-yl]methyl]-6-methylpyrimidin-2-amine —— C17H28N4
4-cyclobutyl-N-[[(3S)-1-ethylpiperidin-3-yl]methyl]-6-methylpyrimidin-2-amine
—— 5-[1-[(1S)-1-pyridin-4-ylpropyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C19H17N5S
5-[1-[(1S)-1-pyridin-4-ylpropyl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— 4-cyclopentyl-N-[(1R)-1-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine —— C17H22N4
4-cyclopentyl-N-[(1R)-1-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
—— 4-cyclopentyl-N-[(1R)-1-pyridin-2-ylpropyl]pyrimidin-2-amine —— C17H22N4
4-cyclopentyl-N-[(1R)-1-pyridin-2-ylpropyl]pyrimidin-2-amine
—— 7-[(2S)-2-pyrazol-1-ylbutanoyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2S)-2-pyrazol-1-ylbutanoyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine —— C16H19N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
—— 1-[(3S)-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]piperidin-3-yl]pyrrolidin-2-one —— C19H27N5O2
1-[(3S)-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]piperidin-3-yl]pyrrolidin-2-one
—— (2S)-2-N-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-N,1-N-dimethylpropane-1,2-diamine —— C14H24N4
(2S)-2-N-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-N,1-N-dimethylpropane-1,2-diamine
—— 7-[(5R)-3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H17N5O3
7-[(5R)-3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2S)-N-(benzylsulfamoyl)-1-pyrazin-2-ylpropan-2-amine —— C14H18N4O2S
(2S)-N-(benzylsulfamoyl)-1-pyrazin-2-ylpropan-2-amine