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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-(3-fluorophenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C19H21FN6O2S
5-(3-fluorophenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 4-[2-amino-4-[(2R)-1-(2-cyclopentylacetyl)piperidin-2-yl]pyrimidin-5-yl]benzamide —— C23H29N5O2
4-[2-amino-4-[(2R)-1-(2-cyclopentylacetyl)piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5-phenylpyrimidin-2-amine —— C19H22N6O2S
4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]-5-phenylpyrimidin-2-amine
—— 1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-3-phenoxypropan-1-one —— C24H26N4O2
1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-3-phenoxypropan-1-one
—— 5-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24F2N4O
1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H22ClFN4O2
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H22F2N4O2
1-[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— [(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C21H24N6O2
[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24F2N4O
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— N-[2-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]methanesulfonamide —— C18H22ClN5O3S
N-[2-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]methanesulfonamide
—— 5-(3-methoxyphenyl)-4-[(2S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine —— C23H28N6O
5-(3-methoxyphenyl)-4-[(2S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-2-yl]pyrimidin-2-amine
—— 5-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22FN5O2
5-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 5-(4-fluorophenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C19H21FN6O2S
5-(4-fluorophenyl)-4-[(2S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone —— C22H24ClN5O2
1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone
—— 1-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H23FN4O2
1-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 4-[2-amino-4-[(2R)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]pyrimidin-5-yl]benzamide —— C25H26FN5O2
4-[2-amino-4-[(2R)-1-[3-(4-fluorophenyl)propanoyl]piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 4-[2-amino-4-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide —— C20H26N6O2
4-[2-amino-4-[(2S)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H22ClFN4O2
1-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 5-(4-chlorophenyl)-4-[(2S)-1-(1H-pyrazol-4-ylsulfonyl)piperidin-2-yl]pyrimidin-2-amine —— C18H19ClN6O2S
5-(4-chlorophenyl)-4-[(2S)-1-(1H-pyrazol-4-ylsulfonyl)piperidin-2-yl]pyrimidin-2-amine
—— 5-(4-chlorophenyl)-4-[(2R)-1-(1H-pyrazol-4-ylsulfonyl)piperidin-2-yl]pyrimidin-2-amine —— C18H19ClN6O2S
5-(4-chlorophenyl)-4-[(2R)-1-(1H-pyrazol-4-ylsulfonyl)piperidin-2-yl]pyrimidin-2-amine
—— [(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20ClN5OS
[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C21H23N5O2S
[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 5-(4-chlorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine —— C19H21ClN6O2S
5-(4-chlorophenyl)-4-[(2R)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone —— C23H28F3N5O
[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone
—— 5-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22ClN5O2
5-[(2S)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— [(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C20H21FN6O
[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C24H25FN4O3
1-[(2S)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 5-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C23H25N5O3
5-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24ClFN4O
1-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— [(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone —— C22H28FN5O
[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone
—— [(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C20H21FN6O
[(2R)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 5-(4-chlorophenyl)-4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine —— C20H22ClN5O3S
5-(4-chlorophenyl)-4-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]pyrimidin-2-amine
—— 1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24F2N4O
1-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— [(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C21H21F3N6O
[(2R)-2-[2-amino-5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 5-(4-chlorophenyl)-4-[(2S)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-2-yl]pyrimidin-2-amine —— C22H25ClN6
5-(4-chlorophenyl)-4-[(2S)-1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-2-yl]pyrimidin-2-amine
—— 5-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H23N5O2
5-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenoxypropan-1-one —— C25H28N4O3
1-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-phenoxypropan-1-one
—— 4-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine —— C20H22FN5O3S
4-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone —— C22H24ClN5O2
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone
—— 6-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24ClFN4O
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C23H23FN4O2
1-[(2S)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 1-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone —— C22H24ClN5O2
1-[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(3,5-dimethyl-1,2-oxazol-4-yl)ethanone
—— 4-[2-amino-4-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide —— C20H26N6O2
4-[2-amino-4-[(2R)-1-[2-(dimethylamino)acetyl]piperidin-2-yl]pyrimidin-5-yl]benzamide
—— [(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20ClN5OS
[(2R)-2-[2-amino-5-(3-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C20H21FN6O
[(2S)-2-[2-amino-5-(2-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 6-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one —— C21H21FN6O2
6-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-2-methylpyridazin-3-one
—— [(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19FN6O
[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— 5-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H23N5O2
5-[(2R)-2-(2-amino-5-phenylpyrimidin-4-yl)piperidine-1-carbonyl]-1-methylpyridin-2-one