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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— methyl (6R)-6-[5-(3-chloro-4-methylphenyl)furan-2-yl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C19H19ClN2O4
methyl (6R)-6-[5-(3-chloro-4-methylphenyl)furan-2-yl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— methyl (6S)-6-[5-(3-chloro-4-methylphenyl)furan-2-yl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C19H19ClN2O4
methyl (6S)-6-[5-(3-chloro-4-methylphenyl)furan-2-yl]-3,4-dimethyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— N-[(2R)-butan-2-yl]-2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C14H19Cl2N3O4S
N-[(2R)-butan-2-yl]-2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— 5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C20H32N4O2
5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 3-[2-[(2R)-piperidin-2-yl]ethyl]-5-thieno[2,3-d]pyrimidin-4-ylphenol —— C19H21N3OS
3-[2-[(2R)-piperidin-2-yl]ethyl]-5-thieno[2,3-d]pyrimidin-4-ylphenol
—— N-[(2S)-butan-2-yl]-2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C14H19Cl2N3O4S
N-[(2S)-butan-2-yl]-2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— (9aR)-2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-6,9-dione —— C18H20N6O2
(9aR)-2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-6,9-dione
—— (2-amino-4-phenylpyrimidin-5-yl)-[(2R)-2-(cyclohexylmethyl)morpholin-4-yl]methanone —— C22H28N4O2
(2-amino-4-phenylpyrimidin-5-yl)-[(2R)-2-(cyclohexylmethyl)morpholin-4-yl]methanone
—— (2S)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one —— C18H23N5O2
(2S)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one
—— [(2R)-2-(3-phenylpropyl)morpholin-4-yl]-(2-pyridin-4-ylpyrimidin-5-yl)methanone —— C23H24N4O2
[(2R)-2-(3-phenylpropyl)morpholin-4-yl]-(2-pyridin-4-ylpyrimidin-5-yl)methanone
—— (2-amino-4-phenylpyrimidin-5-yl)-[(2R)-2-(trifluoromethyl)morpholin-4-yl]methanone —— C16H15F3N4O2
(2-amino-4-phenylpyrimidin-5-yl)-[(2R)-2-(trifluoromethyl)morpholin-4-yl]methanone
—— (2-amino-4-phenylpyrimidin-5-yl)-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methanone —— C24H25FN4O
(2-amino-4-phenylpyrimidin-5-yl)-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methanone
—— 5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C17H26N4O2
5-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— 6-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H26N4O3
6-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-(2-methoxyphenyl)-N-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]pyridazin-3-amine —— C17H19N5O
6-(2-methoxyphenyl)-N-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]pyridazin-3-amine
—— 6-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H26N4O3
6-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (2S)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one —— C19H25N5OS
(2S)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one
—— ethyl (4S)-4-ethyl-6-[(4-ethyl-5-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24N2O5S
ethyl (4S)-4-ethyl-6-[(4-ethyl-5-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (9aS)-2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-6,9-dione —— C18H20N6O2
(9aS)-2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1,3,4,7,8,9a-hexahydropyrazino[1,2-a]pyrazine-6,9-dione
—— (2-amino-4-phenylpyrimidin-5-yl)-[(2S)-2-(trifluoromethyl)morpholin-4-yl]methanone —— C16H15F3N4O2
(2-amino-4-phenylpyrimidin-5-yl)-[(2S)-2-(trifluoromethyl)morpholin-4-yl]methanone
—— 6-[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione —— C19H22N4O4
6-[(3R)-4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (2R)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one —— C18H23N5O2
(2R)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one
—— (2-amino-4-phenylpyrimidin-5-yl)-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methanone —— C24H25FN4O
(2-amino-4-phenylpyrimidin-5-yl)-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methanone
—— N-[(1R)-1-(cyclohexen-1-yl)ethyl]-2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetamide —— C15H21N3O2
N-[(1R)-1-(cyclohexen-1-yl)ethyl]-2-(2-methyl-6-oxo-1H-pyrimidin-5-yl)acetamide
—— [6-[(2S)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C21H26N4O3
[6-[(2S)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— 6-[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione —— C19H22N4O4
6-[(3S)-4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one —— C17H26N4O2
5-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepane-1-carbonyl]-1H-pyrazin-2-one
—— [6-[(2R)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C21H26N4O3
[6-[(2R)-2-[(3-methoxyphenyl)methyl]morpholin-4-yl]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— [(3R)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone —— C21H31N5O2
[(3R)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone
—— 6-(2-methoxyphenyl)-N-[(1R)-1-(1-methylpyrazol-4-yl)ethyl]pyridazin-3-amine —— C17H19N5O
6-(2-methoxyphenyl)-N-[(1R)-1-(1-methylpyrazol-4-yl)ethyl]pyridazin-3-amine
—— [(3S)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone —— C21H31N5O2
[(3S)-1-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone
—— (2-amino-4-phenylpyrimidin-5-yl)-[(2S)-2-(cyclohexylmethyl)morpholin-4-yl]methanone —— C22H28N4O2
(2-amino-4-phenylpyrimidin-5-yl)-[(2S)-2-(cyclohexylmethyl)morpholin-4-yl]methanone
—— (2R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one —— C19H25N5OS
(2R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one
—— 4-cyclobutyl-6-methyl-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-2-amine —— C17H28N4O2S
4-cyclobutyl-6-methyl-N-[2-[(2S)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-2-amine
—— ethyl (4R)-4-ethyl-6-[(4-ethyl-5-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24N2O5S
ethyl (4R)-4-ethyl-6-[(4-ethyl-5-methylthiophene-2-carbonyl)oxymethyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone —— C21H26F2N4O
[(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]-[2-(propan-2-ylamino)pyrimidin-5-yl]methanone
—— 4-cyclobutyl-6-methyl-N-[2-[(2R)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-2-amine —— C17H28N4O2S
4-cyclobutyl-6-methyl-N-[2-[(2R)-1-methylsulfonylpiperidin-2-yl]ethyl]pyrimidin-2-amine
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine —— C18H23N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
—— N-[[(2S)-1-ethylpiperidin-2-yl]methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C15H23F3N4
N-[[(2S)-1-ethylpiperidin-2-yl]methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine —— C18H23N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
—— (3R)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]piperidin-2-one —— C16H19N5O
(3R)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]piperidin-2-one
—— N-[[(2R)-1-ethylpiperidin-2-yl]methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C15H23F3N4
N-[[(2R)-1-ethylpiperidin-2-yl]methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— (3S)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]piperidin-2-one —— C16H19N5O
(3S)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]piperidin-2-one
—— N-[(2S)-2-(N-methylanilino)propyl]-6-oxo-1H-pyrimidine-5-carboxamide —— C15H18N4O2
N-[(2S)-2-(N-methylanilino)propyl]-6-oxo-1H-pyrimidine-5-carboxamide
—— N-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine —— C19H24N6
N-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
—— 4-cyclopentyl-N-[(R)-cyclopropyl-(4-methylpyridin-2-yl)methyl]pyrimidin-2-amine —— C19H24N4
4-cyclopentyl-N-[(R)-cyclopropyl-(4-methylpyridin-2-yl)methyl]pyrimidin-2-amine
—— 3-[(1R)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-hydroxyethyl]phenol —— C17H21N3O2
3-[(1R)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-hydroxyethyl]phenol
—— 3-ethyl-5-[(1R)-1-[2-[2-(furan-2-yl)pyrimidin-5-yl]imidazol-1-yl]ethyl]-1,2,4-oxadiazole —— C17H16N6O2
3-ethyl-5-[(1R)-1-[2-[2-(furan-2-yl)pyrimidin-5-yl]imidazol-1-yl]ethyl]-1,2,4-oxadiazole
—— 4-cyclopentyl-N-[(S)-cyclopropyl-(4-methylpyridin-2-yl)methyl]pyrimidin-2-amine —— C19H24N4
4-cyclopentyl-N-[(S)-cyclopropyl-(4-methylpyridin-2-yl)methyl]pyrimidin-2-amine
—— N-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine —— C19H24N6
N-[(2R)-2-(3,5-dimethylpyrazol-1-yl)propyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine