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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (6S)-3-ethyl-6-(3-methoxyphenyl)-4-[(4-methylphenoxy)methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H28N2O5
ethyl (6S)-3-ethyl-6-(3-methoxyphenyl)-4-[(4-methylphenoxy)methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2-chlorophenyl)-4-[(2-fluorophenoxy)methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C21H20ClFN2O4
ethyl (6R)-6-(2-chlorophenyl)-4-[(2-fluorophenoxy)methyl]-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— methyl (6R)-3-butyl-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C22H31N3O4
methyl (6R)-3-butyl-6-[4-(2,2-dimethylpropanoylamino)phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 1-[4-[2-[4-[(1S,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one —— C18H25N5O3S
1-[4-[2-[4-[(1S,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one
—— (7S)-4-(azocan-1-yl)-7-methyl-2-pyridin-3-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine —— C23H28N4S
(7S)-4-(azocan-1-yl)-7-methyl-2-pyridin-3-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine
—— (7R)-4-(azocan-1-yl)-7-methyl-2-pyridin-3-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine —— C23H28N4S
(7R)-4-(azocan-1-yl)-7-methyl-2-pyridin-3-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine
—— ethyl (6R)-3-butyl-6-[4-(hexanoylamino)phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H35N3O4
ethyl (6R)-3-butyl-6-[4-(hexanoylamino)phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-ethyl-4-[(4-fluorophenoxy)methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C20H21FN2O4S
ethyl (6R)-3-ethyl-4-[(4-fluorophenoxy)methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— [(3S)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]-(2-methylpyrimidin-4-yl)methanone —— C16H20N4OS
[(3S)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]-(2-methylpyrimidin-4-yl)methanone
—— ethyl (6S)-3-butyl-6-[4-(hexanoylamino)phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H35N3O4
ethyl (6S)-3-butyl-6-[4-(hexanoylamino)phenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— 1-[4-[2-[4-[(1R,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one —— C18H25N5O3S
1-[4-[2-[4-[(1R,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one
—— 1-[4-[2-[4-[(1R,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one —— C18H25N5O3S
1-[4-[2-[4-[(1R,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one
—— ethyl (6S)-3-ethyl-4-[(4-fluorophenoxy)methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C20H21FN2O4S
ethyl (6S)-3-ethyl-4-[(4-fluorophenoxy)methyl]-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— 1-[4-[2-[4-[(1S,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one —— C18H25N5O3S
1-[4-[2-[4-[(1S,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-2-oxoethyl]-1,3-thiazol-2-yl]-1,3-diazinan-2-one
—— ethyl (6R)-3-methyl-4-[(4-methylphenoxy)methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H26N2O4
ethyl (6R)-3-methyl-4-[(4-methylphenoxy)methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— [(3R)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]-(2-methylpyrimidin-4-yl)methanone —— C16H20N4OS
[(3R)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]-(2-methylpyrimidin-4-yl)methanone
—— ethyl (6S)-4-[(2-fluorophenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate —— C19H19FN2O4S
ethyl (6S)-4-[(2-fluorophenoxy)methyl]-3-methyl-2-oxo-6-thiophen-3-yl-1,6-dihydropyrimidine-5-carboxylate
—— (2-cyclopropylpyrimidin-4-yl)-[(3R)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C18H22N4OS
(2-cyclopropylpyrimidin-4-yl)-[(3R)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— (2-cyclopropylpyrimidin-4-yl)-[(3S)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C18H22N4OS
(2-cyclopropylpyrimidin-4-yl)-[(3S)-3-(4,5-dimethyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C14H15ClN4OS
(5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C14H15ClN4OS
(5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C14H16ClN5O
(5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidin-1-yl]methanone —— C15H19ClN6O
(5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidin-1-yl]methanone
—— ethyl (6S)-3-methyl-4-[(4-methylphenoxy)methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H26N2O4
ethyl (6S)-3-methyl-4-[(4-methylphenoxy)methyl]-6-(3-methylphenyl)-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidin-1-yl]methanone —— C15H19ClN6O
(5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)piperidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C14H16ClN5O
(5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— N-[(2R)-1-(2-methoxyethoxy)propan-2-yl]-2-[2-(2-oxo-1,3-diazinan-1-yl)-1,3-thiazol-4-yl]acetamide —— C15H24N4O4S
N-[(2R)-1-(2-methoxyethoxy)propan-2-yl]-2-[2-(2-oxo-1,3-diazinan-1-yl)-1,3-thiazol-4-yl]acetamide
—— N-[(R)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-1-methyl-6-oxo-4,5-dihydropyridazine-3-carboxamide —— C14H18N4O2S
N-[(R)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-1-methyl-6-oxo-4,5-dihydropyridazine-3-carboxamide
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone —— C15H17ClN4OS
(5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]methanone
—— N-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-1-methyl-6-oxo-4,5-dihydropyridazine-3-carboxamide —— C14H18N4O2S
N-[(S)-cyclopropyl-(5-methyl-1,3-thiazol-2-yl)methyl]-1-methyl-6-oxo-4,5-dihydropyridazine-3-carboxamide
—— N-[(2S)-1-(2-methoxyethoxy)propan-2-yl]-2-[2-(2-oxo-1,3-diazinan-1-yl)-1,3-thiazol-4-yl]acetamide —— C15H24N4O4S
N-[(2S)-1-(2-methoxyethoxy)propan-2-yl]-2-[2-(2-oxo-1,3-diazinan-1-yl)-1,3-thiazol-4-yl]acetamide
—— N-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-5-methylpyrazine-2-carboxamide —— C14H16N4OS
N-[(S)-cyclopropyl-(4-methyl-1,3-thiazol-2-yl)methyl]-5-methylpyrazine-2-carboxamide
—— 2-(2-chlorophenyl)-7-phenyl-N-propylpyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H19ClN4O
2-(2-chlorophenyl)-7-phenyl-N-propylpyrazolo[1,5-a]pyrimidine-6-carboxamide
—— N-[4-(dimethylamino)-6-(3-methylphenyl)pyrimidin-5-yl]cyclobutanecarboxamide —— C18H22N4O
N-[4-(dimethylamino)-6-(3-methylphenyl)pyrimidin-5-yl]cyclobutanecarboxamide
—— N-[4-(dimethylamino)-6-(3-methylphenyl)pyrimidin-5-yl]-4-methylbenzamide —— C21H22N4O
N-[4-(dimethylamino)-6-(3-methylphenyl)pyrimidin-5-yl]-4-methylbenzamide
—— N-[4-(dimethylamino)-6-phenylpyrimidin-5-yl]-3-methylbutanamide —— C17H22N4O
N-[4-(dimethylamino)-6-phenylpyrimidin-5-yl]-3-methylbutanamide
—— N-[4-(dimethylamino)-6-phenylpyrimidin-5-yl]-4-methylbenzamide —— C20H20N4O
N-[4-(dimethylamino)-6-phenylpyrimidin-5-yl]-4-methylbenzamide
—— ethyl (6S)-6-(3-methoxyphenyl)-3-methyl-4-[(3-methylphenoxy)methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H26N2O5
ethyl (6S)-6-(3-methoxyphenyl)-3-methyl-4-[(3-methylphenoxy)methyl]-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (1R,2R)-2-(2,5-difluorophenyl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]cyclopropane-1-carboxamide —— C17H18F2N4O
(1R,2R)-2-(2,5-difluorophenyl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]cyclopropane-1-carboxamide
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C16H20ClN5O2
(5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(5-propan-2-yl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C14H16ClN5O2
(5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-6-(2-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H25FN2O4
ethyl (6R)-4-[(3,4-dimethylphenoxy)methyl]-6-(2-fluorophenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— N-[(1S,3R)-3-ethoxyspiro[3.5]nonan-1-yl]tetrazolo[1,5-b]pyridazin-6-amine —— C15H22N6O
N-[(1S,3R)-3-ethoxyspiro[3.5]nonan-1-yl]tetrazolo[1,5-b]pyridazin-6-amine
—— N-[1-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]pyrazol-4-yl]pyrazine-2-carboxamide —— C16H20N6O3
N-[1-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]pyrazol-4-yl]pyrazine-2-carboxamide
—— N-[1-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]pyrazol-4-yl]pyrazine-2-carboxamide —— C16H20N6O3
N-[1-[2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]pyrazol-4-yl]pyrazine-2-carboxamide
—— methyl (6R)-6-[3-(cyclopropanecarbonylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate —— C20H25N3O4
methyl (6R)-6-[3-(cyclopropanecarbonylamino)phenyl]-4-methyl-2-oxo-3-propyl-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-4-[(3,4-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C24H28N2O5
ethyl (6S)-4-[(3,4-dimethylphenoxy)methyl]-6-(3-methoxyphenyl)-3-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (1S,2S)-2-(2,5-difluorophenyl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]cyclopropane-1-carboxamide —— C17H18F2N4O
(1S,2S)-2-(2,5-difluorophenyl)-N-[2-[(6-methylpyridazin-3-yl)amino]ethyl]cyclopropane-1-carboxamide
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone —— C14H16ClN5O2
(5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methanone
—— N-[1-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]pyrazol-4-yl]pyrazine-2-carboxamide —— C16H20N6O3
N-[1-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]pyrazol-4-yl]pyrazine-2-carboxamide