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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[1-(Cyclobutanecarbonyl)piperidin-4-yl]-6-(3-fluoro-4-methoxyphenyl)pyridazin-3-one —— C21H24FN3O3
2-[1-(Cyclobutanecarbonyl)piperidin-4-yl]-6-(3-fluoro-4-methoxyphenyl)pyridazin-3-one
—— 4-[3-(3-fluoro-4-methoxyphenyl)-6-oxopyridazin-1-yl]-N,N-dimethylpiperidine-1-sulfonamide —— C18H23FN4O4S
4-[3-(3-fluoro-4-methoxyphenyl)-6-oxopyridazin-1-yl]-N,N-dimethylpiperidine-1-sulfonamide
—— (1S,3R)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide —— C18H23N3O4
(1S,3R)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide
—— (2S)-N-[2-(6-oxo-3-thiophen-2-ylpyridazin-1-yl)ethyl]oxolane-2-carboxamide —— C15H17N3O3S
(2S)-N-[2-(6-oxo-3-thiophen-2-ylpyridazin-1-yl)ethyl]oxolane-2-carboxamide
—— (1R,3R)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide —— C18H23N3O4
(1R,3R)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide
—— (2R)-N-[2-(6-oxo-3-thiophen-2-ylpyridazin-1-yl)ethyl]oxolane-2-carboxamide —— C15H17N3O3S
(2R)-N-[2-(6-oxo-3-thiophen-2-ylpyridazin-1-yl)ethyl]oxolane-2-carboxamide
—— (1S,3S)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide —— C18H23N3O4
(1S,3S)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide
—— (1R,3S)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide —— C18H23N3O4
(1R,3S)-N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-3-methoxycyclohexane-1-carboxamide
—— 1-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone —— C19H24ClN5O
1-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
—— 1-[(3R)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C25H27FN4O2
1-[(3R)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[4-[(3R)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]piperidin-1-yl]ethanone —— C22H28FN5O
1-[4-[(3R)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]piperidin-1-yl]ethanone
—— N,N-diethyl-2-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide —— C18H30N4O2
N,N-diethyl-2-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-4-methylpyrimidine-5-carboxamide
—— 5-(4-methoxyphenyl)-4-[(3S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-2-amine —— C20H24N6O3S
5-(4-methoxyphenyl)-4-[(3S)-1-(1-methylimidazol-4-yl)sulfonylpiperidin-3-yl]pyrimidin-2-amine
—— N-[1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidin-4-yl]-5-methylpyrazine-2-carboxamide —— C20H20FN5OS
N-[1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidin-4-yl]-5-methylpyrazine-2-carboxamide
—— 2-[(2S)-1-(cyclobutanecarbonyl)piperidin-2-yl]-N,N-diethyl-4-methylpyrimidine-5-carboxamide —— C20H30N4O2
2-[(2S)-1-(cyclobutanecarbonyl)piperidin-2-yl]-N,N-diethyl-4-methylpyrimidine-5-carboxamide
—— N-benzyl-4-methyl-2-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide —— C24H25N5O2
N-benzyl-4-methyl-2-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide
—— N,N-diethyl-4-methyl-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C21H27N5O2
N,N-diethyl-4-methyl-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide
—— [(3R)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone —— C23H28F3N5O
[(3R)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpiperidin-4-yl)methanone
—— [(3S)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C21H21F3N6O
[(3S)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 4-[(3R)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-5-(4-methoxyphenyl)pyrimidin-2-amine —— C25H27N5O
4-[(3R)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-5-(4-methoxyphenyl)pyrimidin-2-amine
—— 4-[(3S)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-5-(4-methoxyphenyl)pyrimidin-2-amine —— C25H27N5O
4-[(3S)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-5-(4-methoxyphenyl)pyrimidin-2-amine
—— [(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H20ClN5OS
[(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— 1-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one —— C24H24F2N4O
1-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(4-fluorophenyl)propan-1-one
—— 1-[4-[(3S)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]piperidin-1-yl]ethanone —— C22H28FN5O
1-[4-[(3S)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]piperidin-1-yl]ethanone
—— 2-[(2R)-1-(cyclobutanecarbonyl)piperidin-2-yl]-N,N-diethyl-4-methylpyrimidine-5-carboxamide —— C20H30N4O2
2-[(2R)-1-(cyclobutanecarbonyl)piperidin-2-yl]-N,N-diethyl-4-methylpyrimidine-5-carboxamide
—— 3-[2-amino-4-[(3S)-1-(4-phenylbutanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide —— C26H29N5O2
3-[2-amino-4-[(3S)-1-(4-phenylbutanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide
—— 3-[2-amino-4-[(3R)-1-(4-phenylbutanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide —— C26H29N5O2
3-[2-amino-4-[(3R)-1-(4-phenylbutanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide
—— 1-[(3R)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C24H25FN4O3
1-[(3R)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— 1-[(3R)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-pyrrolidin-1-ylethanone —— C22H26F3N5O
1-[(3R)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-2-pyrrolidin-1-ylethanone
—— 1-[(3S)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone —— C22H29N5O3
1-[(3S)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone
—— N-[2-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]methanesulfonamide —— C18H22FN5O3S
N-[2-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-oxoethyl]methanesulfonamide
—— 4-[2-amino-4-[(3S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-3-yl]pyrimidin-5-yl]benzamide —— C25H26FN5O2
4-[2-amino-4-[(3S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-3-yl]pyrimidin-5-yl]benzamide
—— 5-[(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22ClN5O2
5-[(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— N-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyridin-3-ylmethyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C24H26FN5O
N-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(pyridin-3-ylmethyl)piperidin-2-yl]pyrimidine-5-carboxamide
—— 1-[4-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]piperidin-1-yl]ethanone —— C22H28ClN5O
1-[4-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]piperidin-1-yl]ethanone
—— N-[1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidin-4-yl]pyrazine-2-carboxamide —— C19H18FN5OS
N-[1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidin-4-yl]pyrazine-2-carboxamide
—— 1-[(3S)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-4-phenylbutan-1-one —— C26H30N4O2
1-[(3S)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-4-phenylbutan-1-one
—— 1-[(3R)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone —— C19H24FN5O
1-[(3R)-3-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
—— 5-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one —— C22H22ClN5O2
5-[(3R)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl]-1-methylpyridin-2-one
—— 1-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone —— C21H26FN5O2
1-[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-morpholin-4-ylethanone
—— [(3R)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C20H19F3N6O
[(3R)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— 3-[(3S)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidine-1-carbonyl]-1H-pyridazin-6-one —— C21H19F3N6O2
3-[(3S)-3-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]piperidine-1-carbonyl]-1H-pyridazin-6-one
—— N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-pyrazin-2-ylpiperidin-3-yl]pyrimidine-5-carboxamide —— C23H26N6O2
N-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-pyrazin-2-ylpiperidin-3-yl]pyrimidine-5-carboxamide
—— 4-[2-amino-4-[(3R)-1-(4-phenylbutanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide —— C26H29N5O2
4-[2-amino-4-[(3R)-1-(4-phenylbutanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide
—— 5-(4-chlorophenyl)-4-[(3S)-1-(oxan-4-yl)piperidin-3-yl]pyrimidin-2-amine —— C20H25ClN4O
5-(4-chlorophenyl)-4-[(3S)-1-(oxan-4-yl)piperidin-3-yl]pyrimidin-2-amine
—— 1-[(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone —— C19H24ClN5O
1-[(3S)-3-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(dimethylamino)ethanone
—— 1-[(3S)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C24H25FN4O3
1-[(3S)-3-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-2-(4-fluorophenoxy)ethanone
—— [(3S)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone —— C21H25FN4O
[(3S)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-cyclopentylmethanone
—— [(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone —— C19H19FN6O
[(3R)-3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(1H-pyrazol-5-yl)methanone
—— N,N-diethyl-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide —— C21H27N5O2
N,N-diethyl-4-methyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]pyrimidine-5-carboxamide