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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[3-[4-[(4,6-Dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]azetidin-1-yl]-2-methoxyethanone —— C17H22N6O2
1-[3-[4-[(4,6-Dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]azetidin-1-yl]-2-methoxyethanone
—— 5-[[(6S)-4-[(3-methylimidazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6S)-4-[(3-methylimidazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 2-methyl-6-[(3S)-1-propan-2-ylpyrrolidin-3-yl]-N-pyrimidin-2-ylpyrimidin-4-amine —— C16H22N6
2-methyl-6-[(3S)-1-propan-2-ylpyrrolidin-3-yl]-N-pyrimidin-2-ylpyrimidin-4-amine
—— 5-[[(6S)-4-(2-methylpyrazole-3-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H20N6O3
5-[[(6S)-4-(2-methylpyrazole-3-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 6-[1-(1H-imidazol-2-ylmethyl)azetidin-3-yl]-2-methyl-N-pyrimidin-2-ylpyrimidin-4-amine —— C16H18N8
6-[1-(1H-imidazol-2-ylmethyl)azetidin-3-yl]-2-methyl-N-pyrimidin-2-ylpyrimidin-4-amine
—— 2-[(2R)-2-[2-methyl-6-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol —— C16H22N6O
2-[(2R)-2-[2-methyl-6-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol
—— 2-methyl-6-[(2S)-1-propan-2-ylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine —— C16H22N6
2-methyl-6-[(2S)-1-propan-2-ylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine
—— 1-[3-[2-Methyl-6-[(5-methyl-1,3-thiazol-2-yl)amino]pyrimidin-4-yl]azetidin-1-yl]ethanone —— C14H17N5OS
1-[3-[2-Methyl-6-[(5-methyl-1,3-thiazol-2-yl)amino]pyrimidin-4-yl]azetidin-1-yl]ethanone
—— 5-[[(6R)-4-(cyclopentanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C17H24N4O3
5-[[(6R)-4-(cyclopentanecarbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— N-methyl-5-[[(6S)-4-(1H-pyrazole-5-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H20N6O3
N-methyl-5-[[(6S)-4-(1H-pyrazole-5-carbonyl)-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 2-methyl-6-[(2R)-1-methylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine —— C14H18N6
2-methyl-6-[(2R)-1-methylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine
—— N-[6-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-2-methylpyrimidin-4-yl]-1,3-thiazol-2-amine —— C16H23N5OS
N-[6-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-2-methylpyrimidin-4-yl]-1,3-thiazol-2-amine
—— 2-[(2S)-2-[2-methyl-6-(1,3-thiazol-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol —— C15H21N5OS
2-[(2S)-2-[2-methyl-6-(1,3-thiazol-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol
—— 6-[(2R)-1-(2-methoxyethyl)pyrrolidin-2-yl]-2-methyl-N-pyrimidin-2-ylpyrimidin-4-amine —— C16H22N6O
6-[(2R)-1-(2-methoxyethyl)pyrrolidin-2-yl]-2-methyl-N-pyrimidin-2-ylpyrimidin-4-amine
—— 2-methyl-N-(3-methylpyridin-2-yl)-6-[(3R)-1-methylpyrrolidin-3-yl]pyrimidin-4-amine —— C16H21N5
2-methyl-N-(3-methylpyridin-2-yl)-6-[(3R)-1-methylpyrrolidin-3-yl]pyrimidin-4-amine
—— [3-[2-Methyl-6-(pyrimidin-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]-pyrazin-2-ylmethanone —— C17H16N8O
[3-[2-Methyl-6-(pyrimidin-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]-pyrazin-2-ylmethanone
—— 2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-(6-methylpyridin-2-yl)pyrimidin-4-amine —— C19H23N7
2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-(6-methylpyridin-2-yl)pyrimidin-4-amine
—— 2-methyl-N-(3-methylpyridin-2-yl)-6-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-amine —— C18H25N5
2-methyl-N-(3-methylpyridin-2-yl)-6-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-amine
—— N-[2-methyl-6-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C14H19N5S
N-[2-methyl-6-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 2-[(2R)-2-[2-methyl-6-[(6-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]ethanol —— C18H25N5O
2-[(2R)-2-[2-methyl-6-[(6-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]ethanol
—— 5-ethyl-N-[6-methyl-2-[(3R)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C18H26N6OS
5-ethyl-N-[6-methyl-2-[(3R)-1-(oxan-4-yl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 5-methyl-N-[2-methyl-6-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C15H21N5S
5-methyl-N-[2-methyl-6-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 5-methyl-N-[2-methyl-6-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C16H24N6S
5-methyl-N-[2-methyl-6-[(2R)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-pyrimidin-2-ylpyrimidin-4-amine —— C17H20N8
2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-pyrimidin-2-ylpyrimidin-4-amine
—— 2-methyl-6-[(3R)-1-pyrazin-2-ylpyrrolidin-3-yl]-N-pyrimidin-2-ylpyrimidin-4-amine —— C17H18N8
2-methyl-6-[(3R)-1-pyrazin-2-ylpyrrolidin-3-yl]-N-pyrimidin-2-ylpyrimidin-4-amine
—— N-[2-methyl-6-[(3R)-1-methylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C12H16N6S
N-[2-methyl-6-[(3R)-1-methylpyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,2-oxazol-3-amine —— C17H21N7O
N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,2-oxazol-3-amine
—— 2-[(3R)-3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol —— C15H20N6O
2-[(3R)-3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol
—— 2-methyl-N-(3-methylpyridin-2-yl)-6-[(2R)-1-methylpyrrolidin-2-yl]pyrimidin-4-amine —— C16H21N5
2-methyl-N-(3-methylpyridin-2-yl)-6-[(2R)-1-methylpyrrolidin-2-yl]pyrimidin-4-amine
—— 5-methyl-N-[2-methyl-6-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C16H24N6S
5-methyl-N-[2-methyl-6-[(2S)-1-propan-2-ylpiperidin-2-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 4,6-dimethyl-N-[2-methyl-6-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C16H22N6O2S
4,6-dimethyl-N-[2-methyl-6-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-(6-methylpyridin-2-yl)pyrimidin-4-amine —— C19H23N7
2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-(6-methylpyridin-2-yl)pyrimidin-4-amine
—— 5-[[(6S)-4-[(2-methylpyrazol-3-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6S)-4-[(2-methylpyrazol-3-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 2-[(2S)-2-[2-methyl-6-[(6-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]ethanol —— C18H25N5O
2-[(2S)-2-[2-methyl-6-[(6-methylpyridin-2-yl)amino]pyrimidin-4-yl]piperidin-1-yl]ethanol
—— 2-methyl-N-(3-methylpyridin-2-yl)-6-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-amine —— C16H21N5O2S
2-methyl-N-(3-methylpyridin-2-yl)-6-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-amine
—— (3S)-3-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C17H25N7O2S
(3S)-3-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— 2-methyl-6-[(3S)-1-methylpyrrolidin-3-yl]-N-pyridin-2-ylpyrimidin-4-amine —— C15H19N5
2-methyl-6-[(3S)-1-methylpyrrolidin-3-yl]-N-pyridin-2-ylpyrimidin-4-amine
—— 2-methyl-6-[(2S)-1-(6-methylpyrimidin-4-yl)pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine —— C18H20N8
2-methyl-6-[(2S)-1-(6-methylpyrimidin-4-yl)pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine
—— 6-[(2S)-1-(2-methoxyethyl)pyrrolidin-2-yl]-2-methyl-N-pyrimidin-2-ylpyrimidin-4-amine —— C16H22N6O
6-[(2S)-1-(2-methoxyethyl)pyrrolidin-2-yl]-2-methyl-N-pyrimidin-2-ylpyrimidin-4-amine
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-oxolane-2-carboxylate —— C12H12N2O4S
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (2R)-oxolane-2-carboxylate
—— N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-4,6-dimethylpyrimidin-2-amine —— C19H24N8
N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-4,6-dimethylpyrimidin-2-amine
—— 4,6-dimethyl-N-[2-methyl-6-[(3R)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C16H22N6O2S
4,6-dimethyl-N-[2-methyl-6-[(3R)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 2-[(3S)-3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol —— C15H20N6O
2-[(3S)-3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol
—— 1-[3-[2-Methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]ethanone —— C14H16N6O
1-[3-[2-Methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]ethanone
—— 4,6-dimethyl-N-[6-methyl-2-[1-(oxan-4-yl)azetidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C19H26N6O
4,6-dimethyl-N-[6-methyl-2-[1-(oxan-4-yl)azetidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 5-ethyl-N-[2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H22N8S
5-ethyl-N-[2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 6-methyl-2-[(3R)-1-(oxan-4-yl)pyrrolidin-3-yl]-N-pyrazin-2-ylpyrimidin-4-amine —— C18H24N6O
6-methyl-2-[(3R)-1-(oxan-4-yl)pyrrolidin-3-yl]-N-pyrazin-2-ylpyrimidin-4-amine
—— 5-[[(6S)-4-[(1-methylpyrazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide —— C16H22N6O2
5-[[(6S)-4-[(1-methylpyrazol-4-yl)methyl]-1,4-oxazepan-6-yl]methyl]pyrazine-2-carboxamide
—— 2-methyl-N-(3-methylpyridin-2-yl)-6-[(3S)-1-methylpyrrolidin-3-yl]pyrimidin-4-amine —— C16H21N5
2-methyl-N-(3-methylpyridin-2-yl)-6-[(3S)-1-methylpyrrolidin-3-yl]pyrimidin-4-amine
—— 2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-pyrazin-2-ylpyrimidin-4-amine —— C17H20N8
2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-pyrazin-2-ylpyrimidin-4-amine