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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[1-[[1-(2-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(3-methyl-6-oxopyridazin-1-yl)acetamide —— C24H31FN4O2
N-[1-[[1-(2-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(3-methyl-6-oxopyridazin-1-yl)acetamide
—— 2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)-N-[1-[[1-(4-methylphenyl)cyclopentyl]methyl]piperidin-4-yl]acetamide —— C25H34N4O3
2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)-N-[1-[[1-(4-methylphenyl)cyclopentyl]methyl]piperidin-4-yl]acetamide
—— 4-[(3R)-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C20H22N6O
4-[(3R)-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)-N-[1-[(1-phenylcyclopentyl)methyl]piperidin-4-yl]acetamide —— C24H32N4O3
2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)-N-[1-[(1-phenylcyclopentyl)methyl]piperidin-4-yl]acetamide
—— 2-(2,4-dioxopyrimidin-1-yl)-N-[1-[[1-(4-methylphenyl)cyclohexyl]methyl]piperidin-4-yl]acetamide —— C25H34N4O3
2-(2,4-dioxopyrimidin-1-yl)-N-[1-[[1-(4-methylphenyl)cyclohexyl]methyl]piperidin-4-yl]acetamide
—— N-[1-[[1-(2-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide —— C23H29FN4O2
N-[1-[[1-(2-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide
—— 2-(3-methyl-6-oxopyridazin-1-yl)-N-[1-[(1-phenylcyclopentyl)methyl]piperidin-4-yl]acetamide —— C24H32N4O2
2-(3-methyl-6-oxopyridazin-1-yl)-N-[1-[(1-phenylcyclopentyl)methyl]piperidin-4-yl]acetamide
—— 6-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C21H24N6O
6-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— N-[1-[[1-(3-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide —— C23H29FN4O2
N-[1-[[1-(3-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide
—— N-[1-[[1-(3-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide —— C24H31FN4O3
N-[1-[[1-(3-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide
—— N-[1-[[1-(4-methylphenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide —— C24H32N4O2
N-[1-[[1-(4-methylphenyl)cyclopentyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide
—— 2-(2,4-dioxopyrimidin-1-yl)-N-[1-[(1-phenylcyclopentyl)methyl]piperidin-4-yl]acetamide —— C23H30N4O3
2-(2,4-dioxopyrimidin-1-yl)-N-[1-[(1-phenylcyclopentyl)methyl]piperidin-4-yl]acetamide
—— 2-(2,4-dioxopyrimidin-1-yl)-N-[1-[[1-(2-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]acetamide —— C23H29FN4O3
2-(2,4-dioxopyrimidin-1-yl)-N-[1-[[1-(2-fluorophenyl)cyclopentyl]methyl]piperidin-4-yl]acetamide
—— N-[1-[[1-(4-chlorophenyl)cyclobutyl]methyl]piperidin-4-yl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide —— C23H29ClN4O3
N-[1-[[1-(4-chlorophenyl)cyclobutyl]methyl]piperidin-4-yl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide
—— N-[1-[[1-(4-chlorophenyl)cyclobutyl]methyl]piperidin-4-yl]-2-(3-methyl-6-oxopyridazin-1-yl)acetamide —— C23H29ClN4O2
N-[1-[[1-(4-chlorophenyl)cyclobutyl]methyl]piperidin-4-yl]-2-(3-methyl-6-oxopyridazin-1-yl)acetamide
—— 4-[(3S)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C23H24N4O3
4-[(3S)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 6-[(3R)-1-[(2-ethylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H24N6OS
6-[(3R)-1-[(2-ethylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 4-[(3R)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C23H24N4O3
4-[(3R)-1-[(6-methyl-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 6-[(3S)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H30N8O
6-[(3S)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C21H22N6OS
6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 2-pyridin-2-yl-4-[(3R)-1-(thiophen-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C19H20N4OS
2-pyridin-2-yl-4-[(3R)-1-(thiophen-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— N-[1-[[1-(4-chlorophenyl)cyclobutyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide —— C22H27ClN4O2
N-[1-[[1-(4-chlorophenyl)cyclobutyl]methyl]piperidin-4-yl]-2-(2-oxopyrimidin-1-yl)acetamide
—— 6-[(3R)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H26N6O
6-[(3R)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 2-pyridin-2-yl-4-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
2-pyridin-2-yl-4-[(3R)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 6-[(3S)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C22H26N6O
6-[(3S)-1-[(2-propylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C21H24N6O
6-[(3S)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 4-[(3S)-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C20H22N6O
4-[(3S)-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 4-[(3S)-1-[(4-oxochromen-3-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C24H22N4O3
4-[(3S)-1-[(4-oxochromen-3-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 2-pyridin-2-yl-4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
2-pyridin-2-yl-4-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C20H22N6O2
6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C20H23N7O
6-[(3S)-1-[[2-(methylamino)pyrimidin-5-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C24H30N8O
6-[(3R)-1-[[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C20H22N6OS
6-[(3S)-1-[(2-methylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C23H24N4O4
6-[(3R)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 2-pyridin-3-yl-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
2-pyridin-3-yl-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 6-[(3R)-1-[(2-propylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-4-one —— C22H26N6OS
6-[(3R)-1-[(2-propylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-4-yl-1H-pyrimidin-4-one
—— 6-[(3R)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C20H22N6O2
6-[(3R)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C23H24N4O4
6-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C22H26N6O
6-[(3S)-1-[(2-propan-2-ylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C20H22N6O2
6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H22N6OS
6-[(3S)-1-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 2-pyridin-2-yl-4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C20H21N5O
2-pyridin-2-yl-4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 2-pyridin-2-yl-4-[(3S)-1-(thiophen-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C19H20N4OS
2-pyridin-2-yl-4-[(3S)-1-(thiophen-3-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 6-[(3R)-1-[(6-ethoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C24H26N4O4
6-[(3R)-1-[(6-ethoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— 2-pyridin-2-yl-4-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one —— C19H20N4OS
2-pyridin-2-yl-4-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrimidin-6-one
—— 4-[(3S)-1-[(2-piperidin-1-ylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C24H29N7O
4-[(3S)-1-[(2-piperidin-1-ylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— 6-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one —— C23H24N4O4
6-[(3S)-1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]-2-pyridin-2-yl-1H-pyrimidin-4-one
—— 2-pyridin-3-yl-6-[(3R)-1-(quinolin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-4-one —— C24H23N5O
2-pyridin-3-yl-6-[(3R)-1-(quinolin-4-ylmethyl)piperidin-3-yl]-1H-pyrimidin-4-one
—— 4-[(3R)-1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C20H22N4OS
4-[(3R)-1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— 6-[(3S)-1-[(2-ethylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C21H24N6OS
6-[(3S)-1-[(2-ethylsulfanylpyrimidin-5-yl)methyl]piperidin-3-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one