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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H28F2N4
5-[[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— (3R)-4-[(4-fluorophenyl)methyl]-1-(6-oxo-1H-pyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one —— C20H23FN4O3
(3R)-4-[(4-fluorophenyl)methyl]-1-(6-oxo-1H-pyrimidine-5-carbonyl)-3-propan-2-yl-1,4-diazepan-5-one
—— ethyl (4S)-6-[[5-(3,4-dimethylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H24N4O4S
ethyl (4S)-6-[[5-(3,4-dimethylphenyl)-1,3,4-oxadiazol-2-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methylpyrimidin-5-yl)methanone —— C21H27FN4O
[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methylpyrimidin-5-yl)methanone
—— [(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methylpyrimidin-5-yl)methanone —— C21H27FN4O
[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-(2-methylpyrimidin-5-yl)methanone
—— 2-[2-[2-[(4R)-2,2-dimethyloxan-4-yl]imidazol-1-yl]ethylamino]-6-methyl-1H-pyrimidin-4-one —— C17H25N5O2
2-[2-[2-[(4R)-2,2-dimethyloxan-4-yl]imidazol-1-yl]ethylamino]-6-methyl-1H-pyrimidin-4-one
—— (3S)-4-benzyl-3-ethyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one —— C19H22N4O2
(3S)-4-benzyl-3-ethyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one —— C19H22N4O2
(3R)-4-benzyl-3-ethyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
—— 7-[(2S)-2-phenoxybutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H22N4O3
7-[(2S)-2-phenoxybutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylbutan-1-one —— C19H25N5O
(2R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylbutan-1-one
—— [(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone —— C20H32N4O
[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone
—— [(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone —— C20H32N4O
[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]-(2-propan-2-ylpyrimidin-4-yl)methanone
—— 1-[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]pyrrolidin-2-one —— C14H20N4O2
1-[(3S)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]pyrrolidin-2-one
—— 7-[(2R)-2-phenoxybutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H22N4O3
7-[(2R)-2-phenoxybutanoyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 6-(2-methoxyphenyl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine —— C18H19N5O
6-(2-methoxyphenyl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine
—— (2-amino-6-methylpyrimidin-4-yl)-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C18H29N5O
(2-amino-6-methylpyrimidin-4-yl)-[(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— 1-[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]pyrrolidin-2-one —— C14H20N4O2
1-[(3R)-1-(3-methoxypyrazin-2-yl)piperidin-3-yl]pyrrolidin-2-one
—— [(3S)-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone —— C21H31N5O2
[(3S)-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone
—— (2-amino-6-methylpyrimidin-4-yl)-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C18H29N5O
(2-amino-6-methylpyrimidin-4-yl)-[(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— 6-(2-methoxyphenyl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine —— C18H19N5O
6-(2-methoxyphenyl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyridazin-3-amine
—— N-[(1S)-1-cyclopropylethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C12H16F3N3
N-[(1S)-1-cyclopropylethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 7-[(2R)-2-pyrazol-1-ylbutanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2R)-2-pyrazol-1-ylbutanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— N-[(1R)-1-cyclopropylethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C12H16F3N3
N-[(1R)-1-cyclopropylethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 4-cyclopentyl-N-[(3S)-oxolan-3-yl]pyrimidin-2-amine —— C13H19N3O
4-cyclopentyl-N-[(3S)-oxolan-3-yl]pyrimidin-2-amine
—— 4-cyclopentyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine —— C16H21N5
4-cyclopentyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine
—— 4-cyclopentyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine —— C16H21N5
4-cyclopentyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine
—— (5S)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one —— C20H24N6O2
(5S)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one
—— (5R)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one —— C20H24N6O2
(5R)-5-[2-[4-(dimethylamino)-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl]pyrrolidin-2-one
—— N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-6-(2-methoxyphenyl)pyridazin-3-amine —— C18H21N5O
N-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-6-(2-methoxyphenyl)pyridazin-3-amine
—— 7-[(2S)-2-pyrazol-1-ylbutanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N6O2
7-[(2S)-2-pyrazol-1-ylbutanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 4-cyclopentyl-N-[(3R)-oxolan-3-yl]pyrimidin-2-amine —— C13H19N3O
4-cyclopentyl-N-[(3R)-oxolan-3-yl]pyrimidin-2-amine
—— N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-6-(2-methoxyphenyl)pyridazin-3-amine —— C18H21N5O
N-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-6-(2-methoxyphenyl)pyridazin-3-amine
—— 6-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H20FN3O3
6-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H20FN3O3
6-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (2-amino-4-methylpyrimidin-5-yl)-[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methanone —— C19H22F2N4O
(2-amino-4-methylpyrimidin-5-yl)-[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methanone
—— (2-amino-4-methylpyrimidin-5-yl)-[(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methanone —— C19H22F2N4O
(2-amino-4-methylpyrimidin-5-yl)-[(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methanone
—— 6-[4-[(3S)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C20H29N5O4
6-[4-[(3S)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— [(3R)-3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl]-(4-propylpyrimidin-5-yl)methanone —— C22H29N3O2
[(3R)-3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl]-(4-propylpyrimidin-5-yl)methanone
—— N-[(S)-cyclopropyl-(4-methylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine —— C21H23N5
N-[(S)-cyclopropyl-(4-methylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
—— 1-[2-[(2S)-2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C17H25N3O4
1-[2-[(2S)-2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— N-[(1R)-2-imidazol-1-yl-1-phenylethyl]-6-(1-methylimidazol-2-yl)pyridazin-3-amine —— C19H19N7
N-[(1R)-2-imidazol-1-yl-1-phenylethyl]-6-(1-methylimidazol-2-yl)pyridazin-3-amine
—— (2R)-4-(6-phenylpyridazin-3-yl)-2-(trifluoromethyl)morpholine —— C15H14F3N3O
(2R)-4-(6-phenylpyridazin-3-yl)-2-(trifluoromethyl)morpholine
—— (2S)-4-(6-phenylpyridazin-3-yl)-2-(trifluoromethyl)morpholine —— C15H14F3N3O
(2S)-4-(6-phenylpyridazin-3-yl)-2-(trifluoromethyl)morpholine
—— 5-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C19H22FN3O2
5-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— 5-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C19H22FN3O2
5-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— N-[(R)-cyclopropyl-(4-methylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine —— C21H23N5
N-[(R)-cyclopropyl-(4-methylpyridin-2-yl)methyl]-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
—— N-[(1S)-2-imidazol-1-yl-1-phenylethyl]-6-(1-methylimidazol-2-yl)pyridazin-3-amine —— C19H19N7
N-[(1S)-2-imidazol-1-yl-1-phenylethyl]-6-(1-methylimidazol-2-yl)pyridazin-3-amine
—— 1-[2-[(2R)-2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C17H25N3O4
1-[2-[(2R)-2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— 6-[4-[(3R)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C20H29N5O4
6-[4-[(3R)-3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (2R)-1-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]butan-2-ol —— C15H20N4O
(2R)-1-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]butan-2-ol