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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H28N6O
1-[4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 1-[4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H28N6O
1-[4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 1-[4-[[(3S)-1-methylpiperidin-3-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H26N6O
1-[4-[[(3S)-1-methylpiperidin-3-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— (3S)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylpentane-1,2-dione —— C20H25N5O2
(3S)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylpentane-1,2-dione
—— (3R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylpentane-1,2-dione —— C20H25N5O2
(3R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylpentane-1,2-dione
—— 2-ethoxy-5-[2-[[(1R)-1-phenylethyl]amino]pyrimidin-4-yl]benzoic acid —— C21H21N3O3
2-ethoxy-5-[2-[[(1R)-1-phenylethyl]amino]pyrimidin-4-yl]benzoic acid
—— 2-ethoxy-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]benzoic acid —— C21H21N3O3
2-ethoxy-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]benzoic acid
—— N-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C13H16F3N5
N-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 1-[4-[[(3R)-1-methylpiperidin-3-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H26N6O
1-[4-[[(3R)-1-methylpiperidin-3-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 1-[4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H28N6O
1-[4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 5-[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3S)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3R)-3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— (2S)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-4-methylpentan-1-one —— C20H27N5O2
(2S)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-4-methylpentan-1-one
—— 7-[(2R)-2-hydroxypropanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C15H16N4O3
7-[(2R)-2-hydroxypropanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 1-[4-[[(1R)-2,3-dihydro-1H-inden-1-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C23H23N5O
1-[4-[[(1R)-2,3-dihydro-1H-inden-1-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 4-cyclobutyl-6-methyl-N-[(2R)-1-(6-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine —— C18H24N4
4-cyclobutyl-6-methyl-N-[(2R)-1-(6-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
—— 1-[4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H28N6O
1-[4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethylamino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidin-2-amine —— C18H22N6
4-(2,6-dimethylpyridin-3-yl)-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidin-2-amine
—— 4-cyclobutyl-6-methyl-N-[(2S)-1-(6-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine —— C18H24N4
4-cyclobutyl-6-methyl-N-[(2S)-1-(6-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
—— 1-[4-[[(1S)-2,3-dihydro-1H-inden-1-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C23H23N5O
1-[4-[[(1S)-2,3-dihydro-1H-inden-1-yl]amino]-2-pyridin-2-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 7-[(2S)-2-hydroxypropanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C15H16N4O3
7-[(2S)-2-hydroxypropanoyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 6-(2-methoxyphenyl)-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]pyridazin-3-amine —— C18H24N4O
6-(2-methoxyphenyl)-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]pyridazin-3-amine
—— (5R)-3-methyl-N-[2-(6-oxo-3-phenyl-4,5-dihydropyridazin-1-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C17H20N4O3
(5R)-3-methyl-N-[2-(6-oxo-3-phenyl-4,5-dihydropyridazin-1-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (3S)-1-(2-ethylpyrimidine-5-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C22H27FN4O2
(3S)-1-(2-ethylpyrimidine-5-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— (3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-diazepan-5-one —— C21H31N5O2
(3S)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-diazepan-5-one
—— 5-[1-[(2R)-1-pyridin-3-ylpropan-2-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C19H17N5S
5-[1-[(2R)-1-pyridin-3-ylpropan-2-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— 5-[1-[(2S)-1-pyridin-3-ylpropan-2-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine —— C19H17N5S
5-[1-[(2S)-1-pyridin-3-ylpropan-2-yl]imidazol-2-yl]-2-thiophen-2-ylpyrimidine
—— (2R)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-4-methylpentan-1-one —— C20H27N5O2
(2R)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-4-methylpentan-1-one
—— 6-(2-methoxyphenyl)-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]pyridazin-3-amine —— C18H24N4O
6-(2-methoxyphenyl)-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]pyridazin-3-amine
—— (3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-diazepan-5-one —— C21H31N5O2
(3R)-4-(cyclopropylmethyl)-3-propan-2-yl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-diazepan-5-one
—— 4-cyclopentyl-N-[(1S)-1-pyridin-4-ylpropyl]pyrimidin-2-amine —— C17H22N4
4-cyclopentyl-N-[(1S)-1-pyridin-4-ylpropyl]pyrimidin-2-amine
—— 1-[4-[[(2R)-butan-2-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H23N5O
1-[4-[[(2R)-butan-2-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 1-[4-[[(2S)-butan-2-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C18H23N5O
1-[4-[[(2S)-butan-2-yl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 5-[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— [(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone —— C21H28FN5O
[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone
—— (3R)-1-(2-ethylpyrimidine-5-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one —— C22H27FN4O2
(3R)-1-(2-ethylpyrimidine-5-carbonyl)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-5-one
—— [(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone —— C21H28FN5O
[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]-[2-(methylamino)pyrimidin-5-yl]methanone
—— (2-amino-4-methylpyrimidin-5-yl)-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C21H28FN5O
(2-amino-4-methylpyrimidin-5-yl)-[(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— 5-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H26FN3O2
5-[(3R)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine —— C20H26F2N4
5-[[(3S)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine
—— 5-[[(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine —— C20H26F2N4
5-[[(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-ethylpyrimidin-2-amine
—— (2-amino-4-methylpyrimidin-5-yl)-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone —— C21H28FN5O
(2-amino-4-methylpyrimidin-5-yl)-[(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1,4-diazepan-1-yl]methanone
—— 5-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H26FN3O2
5-[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— 5-[(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one —— C21H25F2N3O2
5-[(3R)-3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl]-2-propan-2-yl-1H-pyrimidin-6-one
—— (5R)-5-[[(7-acetyl-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)amino]methyl]-1-methylpyrrolidin-2-one —— C20H24N6O2
(5R)-5-[[(7-acetyl-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)amino]methyl]-1-methylpyrrolidin-2-one
—— (5S)-5-[[(7-acetyl-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)amino]methyl]-1-methylpyrrolidin-2-one —— C20H24N6O2
(5S)-5-[[(7-acetyl-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)amino]methyl]-1-methylpyrrolidin-2-one
—— (2S)-2-(3-methyl-6-oxopyridazin-1-yl)hexanehydrazide —— C11H18N4O2
(2S)-2-(3-methyl-6-oxopyridazin-1-yl)hexanehydrazide
—— 2-[(2R,3S)-3-hydroxybutan-2-yl]-6-methylpyridazin-3-one —— C9H14N2O2
2-[(2R,3S)-3-hydroxybutan-2-yl]-6-methylpyridazin-3-one
—— 1,3-Dimethyl-4-amino-5-methansulfonylamino-uracil 89852-69-7 C7H12N4O4S
1,3-Dimethyl-4-amino-5-methansulfonylamino-uracil
—— 6-methyl-2-[(3S)-2-oxooctan-3-yl]pyridazin-3-one —— C13H20N2O2
6-methyl-2-[(3S)-2-oxooctan-3-yl]pyridazin-3-one