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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylcyclopentanecarboxamide —— C24H31N5O2
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylcyclopentanecarboxamide
—— N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylethanesulfonamide —— C20H27N5O3S
N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylethanesulfonamide
—— N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N,2,2-trimethylpropanamide —— C23H31N5O2
N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N,2,2-trimethylpropanamide
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylpropanamide —— C21H27N5O2
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylpropanamide
—— (4S)-1-benzyl-4-[2-[[dimethylsulfamoyl(methyl)amino]methyl]-6-(methylamino)pyrimidin-4-yl]pyrrolidin-2-one —— C20H28N6O3S
(4S)-1-benzyl-4-[2-[[dimethylsulfamoyl(methyl)amino]methyl]-6-(methylamino)pyrimidin-4-yl]pyrrolidin-2-one
—— N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-methoxy-N-methylacetamide —— C21H27N5O3
N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-methoxy-N-methylacetamide
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-methoxy-N-methylacetamide —— C21H27N5O3
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-methoxy-N-methylacetamide
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylcyclohexanecarboxamide —— C25H33N5O2
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylcyclohexanecarboxamide
—— N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide —— C20H25N5O2
N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide
—— N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylpropanamide —— C21H27N5O2
N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylpropanamide
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-(1-ethylpyrazol-3-yl)-2-methylpyrimidin-4-amine —— C16H20N6O
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-(1-ethylpyrazol-3-yl)-2-methylpyrimidin-4-amine
—— 2-[(3S)-5,5-dimethyl-2-oxooxolan-3-yl]-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]acetamide —— C21H20F3N5O3
2-[(3S)-5,5-dimethyl-2-oxooxolan-3-yl]-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]acetamide
—— N-[(4-methoxyphenyl)methyl]-4-(4-methyl-1,3-thiazol-5-yl)-5-phenylpyrimidin-2-amine —— C22H20N4OS
N-[(4-methoxyphenyl)methyl]-4-(4-methyl-1,3-thiazol-5-yl)-5-phenylpyrimidin-2-amine
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylethanesulfonamide —— C20H27N5O3S
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylethanesulfonamide
—— 5-(3-chlorophenyl)-N-methyl-4-(1-methylimidazol-2-yl)-N-(2-pyridin-2-ylethyl)pyrimidin-2-amine —— C22H21ClN6
5-(3-chlorophenyl)-N-methyl-4-(1-methylimidazol-2-yl)-N-(2-pyridin-2-ylethyl)pyrimidin-2-amine
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-hydroxy-N,2-dimethylpropanamide —— C22H29N5O3
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-hydroxy-N,2-dimethylpropanamide
—— (4R)-1-benzyl-4-[2-[[dimethylsulfamoyl(methyl)amino]methyl]-6-(methylamino)pyrimidin-4-yl]pyrrolidin-2-one —— C20H28N6O3S
(4R)-1-benzyl-4-[2-[[dimethylsulfamoyl(methyl)amino]methyl]-6-(methylamino)pyrimidin-4-yl]pyrrolidin-2-one
—— N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-cyclopentyl-N-methylacetamide —— C25H33N5O2
N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-cyclopentyl-N-methylacetamide
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-cyclopentyl-N-methylacetamide —— C25H33N5O2
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-2-cyclopentyl-N-methylacetamide
—— N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylcyclohexanecarboxamide —— C25H33N5O2
N-[[4-[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylcyclohexanecarboxamide
—— N-[(2-methoxyphenyl)methyl]-4-(4-methyl-1,3-thiazol-5-yl)-5-phenylpyrimidin-2-amine —— C22H20N4OS
N-[(2-methoxyphenyl)methyl]-4-(4-methyl-1,3-thiazol-5-yl)-5-phenylpyrimidin-2-amine
—— N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide —— C20H25N5O2
N-[[4-[(3S)-1-benzyl-5-oxopyrrolidin-3-yl]-6-(methylamino)pyrimidin-2-yl]methyl]-N-methylacetamide
—— 5-(3-chlorophenyl)-N-(3-methoxypropyl)-4-(1-methylimidazol-2-yl)pyrimidin-2-amine —— C18H20ClN5O
5-(3-chlorophenyl)-N-(3-methoxypropyl)-4-(1-methylimidazol-2-yl)pyrimidin-2-amine
—— 4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-[[(1R)-1-pyridin-4-ylethyl]amino]-1H-pyrimidin-6-one —— C18H19F3N6O
4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-[[(1R)-1-pyridin-4-ylethyl]amino]-1H-pyrimidin-6-one
—— 1-[4-[4-(3-Fluoroanilino)-6-pyridin-3-ylpyrimidin-2-yl]piperidin-1-yl]-3-methoxypropan-1-one —— C24H26FN5O2
1-[4-[4-(3-Fluoroanilino)-6-pyridin-3-ylpyrimidin-2-yl]piperidin-1-yl]-3-methoxypropan-1-one
—— 2-(2-methoxyethylamino)-4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-1H-pyrimidin-6-one —— C14H18F3N5O2
2-(2-methoxyethylamino)-4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-1H-pyrimidin-6-one
—— 2-(3-methoxyphenyl)-N-[[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]acetamide —— C20H21N5O2
2-(3-methoxyphenyl)-N-[[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]methyl]acetamide
—— 5-(3-chlorophenyl)-N-(2-methoxyethyl)-4-(1-methylimidazol-2-yl)pyrimidin-2-amine —— C17H18ClN5O
5-(3-chlorophenyl)-N-(2-methoxyethyl)-4-(1-methylimidazol-2-yl)pyrimidin-2-amine
—— (4R)-1-ethyl-4-[(3R)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidine-1-carbonyl]pyrrolidin-2-one —— C22H28N6O2
(4R)-1-ethyl-4-[(3R)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidine-1-carbonyl]pyrrolidin-2-one
—— 2-[(3R)-5,5-dimethyl-2-oxooxolan-3-yl]-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]acetamide —— C21H20F3N5O3
2-[(3R)-5,5-dimethyl-2-oxooxolan-3-yl]-N-[[4-[2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenyl]methyl]acetamide
—— (5R)-5-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]pyrrolidin-2-one —— C24H24N6O2
(5R)-5-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]pyrrolidin-2-one
—— 2-(methoxymethyl)-3-(4-methoxyphenyl)-5-(6-methylpyridin-3-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H20N4O3
2-(methoxymethyl)-3-(4-methoxyphenyl)-5-(6-methylpyridin-3-yl)-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (4R)-4-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one —— C25H26N6O2
(4R)-4-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one
—— 4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-[[(1R)-1-pyridin-2-ylethyl]amino]-1H-pyrimidin-6-one —— C18H19F3N6O
4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-[[(1R)-1-pyridin-2-ylethyl]amino]-1H-pyrimidin-6-one
—— 1-[(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-methylpropan-1-one —— C24H27N5O
1-[(2R)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-methylpropan-1-one
—— (4R)-4-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one —— C25H26N6O2
(4R)-4-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one
—— 1-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methylphenyl)ethanone —— C24H27N5O
1-[(3R)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methylphenyl)ethanone
—— 4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-[[(1S)-1-pyridin-4-ylethyl]amino]-1H-pyrimidin-6-one —— C18H19F3N6O
4-[2-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]ethyl]-2-[[(1S)-1-pyridin-4-ylethyl]amino]-1H-pyrimidin-6-one
—— (4R)-1-ethyl-4-[(3S)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidine-1-carbonyl]pyrrolidin-2-one —— C22H28N6O2
(4R)-1-ethyl-4-[(3S)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidine-1-carbonyl]pyrrolidin-2-one
—— N-phenyl-6-pyridin-3-yl-2-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-4-amine —— C26H26N6
N-phenyl-6-pyridin-3-yl-2-[(3S)-1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-4-amine
—— 5-(3-fluorophenyl)-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C17H11FN4O
5-(3-fluorophenyl)-2-pyridin-2-yl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (4S)-4-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one —— C25H26N6O2
(4S)-4-[(3S)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one
—— 2-(3-ethoxypropylamino)-4-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrimidin-6-one —— C14H22N4O3
2-(3-ethoxypropylamino)-4-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrimidin-6-one
—— 1-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methylphenyl)ethanone —— C24H27N5O
1-[(3S)-3-[6-(methylamino)-2-pyridin-3-ylpyrimidin-4-yl]piperidin-1-yl]-2-(3-methylphenyl)ethanone
—— (4-oxo-6,7,8,9-tetrahydropyrimido[2,1-b][1,3]benzothiazol-2-yl)methyl (3R)-3-phenylbutanoate —— C21H22N2O3S
(4-oxo-6,7,8,9-tetrahydropyrimido[2,1-b][1,3]benzothiazol-2-yl)methyl (3R)-3-phenylbutanoate
—— 2-(3-ethoxypropylamino)-4-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrimidin-6-one —— C14H22N4O3
2-(3-ethoxypropylamino)-4-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrimidin-6-one
—— 4-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-2-(thiophen-2-ylmethylamino)-1H-pyrimidin-6-one —— C14H16N4O2S
4-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-2-(thiophen-2-ylmethylamino)-1H-pyrimidin-6-one
—— 1-[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-methylpropan-1-one —— C24H27N5O
1-[(2S)-2-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)piperidin-1-yl]-2-methylpropan-1-one
—— (4S)-1-ethyl-4-[(3S)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidine-1-carbonyl]pyrrolidin-2-one —— C22H28N6O2
(4S)-1-ethyl-4-[(3S)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidine-1-carbonyl]pyrrolidin-2-one
—— (4S)-4-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one —— C25H26N6O2
(4S)-4-[(3R)-3-(4-anilino-6-pyridin-3-ylpyrimidin-2-yl)pyrrolidine-1-carbonyl]-1-methylpyrrolidin-2-one