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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C17H18N6S
N-[4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— N-(3-methylpyridin-2-yl)-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H24N6
N-(3-methylpyridin-2-yl)-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— N-(5-methylpyridin-2-yl)-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H24N6
N-(5-methylpyridin-2-yl)-4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 4-[(2S)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C19H20N6O3S
4-[(2S)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— N-pyridin-2-yl-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C20H22N6
N-pyridin-2-yl-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 4-[(2R)-1-methylsulfonylpiperidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine —— C15H19N5O2S
4-[(2R)-1-methylsulfonylpiperidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine
—— 4-[(2R)-1-(2-phenylethyl)pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C20H22N6
4-[(2R)-1-(2-phenylethyl)pyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— N-[4-[(2S)-1-(pyridin-4-ylmethyl)piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C18H20N6S
N-[4-[(2S)-1-(pyridin-4-ylmethyl)piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— N-[4-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C18H20N6S
N-[4-[(2S)-1-(pyridin-3-ylmethyl)piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— 6-N-methyl-4-N-[4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C20H24N8
6-N-methyl-4-N-[4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— N-[4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C17H18N6S
N-[4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— 4-[(2S)-1-methylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C14H18N6
4-[(2S)-1-methylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— 4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-N-[3-(trifluoromethyl)pyridin-2-yl]pyrimidin-2-amine —— C21H21F3N6
4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-N-[3-(trifluoromethyl)pyridin-2-yl]pyrimidin-2-amine
—— cyclohexyl-[(3S)-3-[2-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C20H26N6O
cyclohexyl-[(3S)-3-[2-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N,N-bis(3-methylbutyl)acetamide —— C19H30N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N,N-bis(3-methylbutyl)acetamide
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-(2,2,2-trifluoroethyl)acetamide —— C11H11F3N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
—— 2-[(4-Fluorophenyl)methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile —— C14H12FN3O
2-[(4-Fluorophenyl)methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile
—— 4-[(2S)-1-methylsulfonylpiperidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine —— C15H19N5O2S
4-[(2S)-1-methylsulfonylpiperidin-2-yl]-N-pyridin-2-ylpyrimidin-2-amine
—— N-pyrazin-2-yl-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C18H19N7
N-pyrazin-2-yl-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 2-[(2-Fluorophenyl)methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile —— C14H12FN3O
2-[(2-Fluorophenyl)methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile
—— N-pyridin-2-yl-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C19H20N6
N-pyridin-2-yl-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 2-[[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile —— C16H12ClN5O2
2-[[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile
—— 4-[(2S)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C19H19FN6O2S
4-[(2S)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— 4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-N-[3-(trifluoromethyl)pyridin-2-yl]pyrimidin-2-amine —— C21H21F3N6
4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-N-[3-(trifluoromethyl)pyridin-2-yl]pyrimidin-2-amine
—— 4-[(2S)-1-(2-phenylethyl)piperidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C21H24N6
4-[(2S)-1-(2-phenylethyl)piperidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— [(2S)-2-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]pyrrolidin-1-yl]-pyrazin-2-ylmethanone —— C19H19N7O
[(2S)-2-[2-[(5-methylpyridin-2-yl)amino]pyrimidin-4-yl]pyrrolidin-1-yl]-pyrazin-2-ylmethanone
—— N-[4-[(2R)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C17H18N6S
N-[4-[(2R)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— N-[4-[(2R)-1-(pyridin-4-ylmethyl)piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C18H20N6S
N-[4-[(2R)-1-(pyridin-4-ylmethyl)piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— 4-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C19H19FN6O2S
4-[(2R)-1-(4-fluorophenyl)sulfonylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— 4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C18H17FN6O2S
4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(1R)-1-(4-ethylphenyl)ethyl]acetamide —— C19H22N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(1R)-1-(4-ethylphenyl)ethyl]acetamide
—— cyclohexyl-[(3R)-3-[2-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C20H26N6O
cyclohexyl-[(3R)-3-[2-(pyrimidin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 6-N-methyl-4-N-[4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C20H24N8
6-N-methyl-4-N-[4-[(3S)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— 4-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C13H16N6O2S
4-[(2R)-1-methylsulfonylpyrrolidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(1S)-1-(4-ethylphenyl)ethyl]acetamide —— C19H22N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-[(1S)-1-(4-ethylphenyl)ethyl]acetamide
—— 2-[(3S)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol —— C15H20N6O
2-[(3S)-3-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]ethanol
—— N-pyrazin-2-yl-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C19H21N7
N-pyrazin-2-yl-4-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
—— 4-[(2S)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C18H17FN6O2S
4-[(2S)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— 4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C18H17FN6O2S
4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— N-pyridin-2-yl-4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C19H20N6
N-pyridin-2-yl-4-[(2S)-1-(pyridin-4-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 4-[(2R)-1-(2-phenylethyl)piperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine —— C21H24N6
4-[(2R)-1-(2-phenylethyl)piperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-2-amine
—— 2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-cyclopentylacetamide —— C14H18N4O2
2-(5-cyano-3,4-dimethyl-6-oxopyridazin-1-yl)-N-cyclopentylacetamide
—— pyrazin-2-yl-[(2S)-2-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C18H18N8O
pyrazin-2-yl-[(2S)-2-[2-(pyrazin-2-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— 6-N-methyl-4-N-[4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C20H24N8
6-N-methyl-4-N-[4-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— N-(5-methylpyridin-2-yl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H22N6
N-(5-methylpyridin-2-yl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— N-(3-methylpyridin-2-yl)-4-[(3S)-1-methylsulfonylpiperidin-3-yl]pyrimidin-2-amine —— C16H21N5O2S
N-(3-methylpyridin-2-yl)-4-[(3S)-1-methylsulfonylpiperidin-3-yl]pyrimidin-2-amine
—— cyclohexyl-[(2S)-2-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone —— C20H26N6O
cyclohexyl-[(2S)-2-[2-(pyrimidin-5-ylamino)pyrimidin-4-yl]piperidin-1-yl]methanone
—— N-(5-methylpyridin-2-yl)-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H22N6
N-(5-methylpyridin-2-yl)-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 4-[(3S)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-pyrimidin-5-ylpyrimidin-2-amine —— C20H22N6O3S
4-[(3S)-1-(4-methoxyphenyl)sulfonylpiperidin-3-yl]-N-pyrimidin-5-ylpyrimidin-2-amine
—— N-(5-methylpyridin-2-yl)-4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-amine —— C21H24N6
N-(5-methylpyridin-2-yl)-4-[(3R)-1-(pyridin-4-ylmethyl)piperidin-3-yl]pyrimidin-2-amine