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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[2-amino-4-[(2R)-1-(4-fluorobenzoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C22H20FN5O2
3-[2-amino-4-[(2R)-1-(4-fluorobenzoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— [(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-phenylmethanone —— C22H19F3N4O
[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-phenylmethanone
—— 2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-1-pyrrolidin-1-ylethanone —— C20H24FN5O
2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-1-pyrrolidin-1-ylethanone
—— 1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanone —— C17H20N4O2
1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanone
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone —— C22H21FN4O2
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone
—— 5-(4-chlorophenyl)-4-[(2S)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine —— C20H18ClFN4O2S
5-(4-chlorophenyl)-4-[(2S)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone —— C22H23N5O2
1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-pyridin-2-ylethanone
—— 5-(4-chlorophenyl)-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H20ClN5
5-(4-chlorophenyl)-4-[(2R)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— (2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C16H20ClN5O2S
(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— [(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone —— C20H18FN5O
[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone
—— 5-(3-fluorophenyl)-4-[(2R)-1-(2-methoxyethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C17H21FN4O
5-(3-fluorophenyl)-4-[(2R)-1-(2-methoxyethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 2-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-pyridin-2-ylacetamide —— C21H21ClN6O
2-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-pyridin-2-ylacetamide
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone —— C22H21FN4O
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone
—— 3-[2-amino-4-[(2S)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C24H25N5O2
3-[2-amino-4-[(2S)-1-(3-phenylpropanoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— [(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C20H18FN5O
[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— 4-[(2S)-1-benzylsulfonylpyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine —— C21H21FN4O2S
4-[(2S)-1-benzylsulfonylpyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine
—— [(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone —— C22H21FN4O2
[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone
—— 2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-methoxyphenyl)acetamide —— C23H24FN5O2
2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-methoxyphenyl)acetamide
—— 2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-fluorophenyl)acetamide —— C22H21F2N5O
2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-fluorophenyl)acetamide
—— 2-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-dimethylacetamide —— C18H22FN5O
2-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N,N-dimethylacetamide
—— 1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C24H25ClN4O2
1-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— 1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one —— C24H26N4O2
1-[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one
—— [(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone —— C21H21N5O2
[(2R)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone
—— 2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-1-pyrrolidin-1-ylethanone —— C20H24FN5O
2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-1-pyrrolidin-1-ylethanone
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C24H25FN4O2
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— 4-[(2S)-1-benzylpyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine —— C21H21FN4
4-[(2S)-1-benzylpyrrolidin-2-yl]-5-(4-fluorophenyl)pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone —— C17H19ClN4O2
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone
—— [(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone —— C20H18ClN5O
[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-4-ylmethanone
—— 3-[2-amino-4-[(2S)-1-(4-chlorobenzoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C22H20ClN5O2
3-[2-amino-4-[(2S)-1-(4-chlorobenzoyl)pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— 1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone —— C23H24N4O2
1-[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone
—— 2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-pyridin-2-ylacetamide —— C21H21ClN6O
2-[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-pyridin-2-ylacetamide
—— 4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-5-(4-methoxyphenyl)pyrimidin-2-amine —— C21H21FN4O3S
4-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-5-(4-methoxyphenyl)pyrimidin-2-amine
—— 3-[2-amino-4-[(2R)-1-[(4-chlorophenyl)methyl]pyrrolidin-2-yl]pyrimidin-5-yl]benzamide —— C22H22ClN5O
3-[2-amino-4-[(2R)-1-[(4-chlorophenyl)methyl]pyrrolidin-2-yl]pyrimidin-5-yl]benzamide
—— (2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C17H23N5O3S
(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— [(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone —— C21H18F2N4O
[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-fluorophenyl)methanone
—— 1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone —— C17H19FN4O2
1-[(2R)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone
—— 1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone —— C18H21FN4O2
1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-2-methoxyethanone
—— [(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C21H21N5O2
[(2S)-2-[2-amino-5-(4-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— 5-(4-fluorophenyl)-4-[(2S)-1-(2-methoxyethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C17H21FN4O
5-(4-fluorophenyl)-4-[(2S)-1-(2-methoxyethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone —— C23H21F3N4O2
1-[(2R)-2-[2-amino-5-[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone
—— 1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone —— C22H21FN4O
1-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenylethanone
—— 2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-fluorophenyl)acetamide —— C22H21F2N5O
2-[(2R)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(4-fluorophenyl)acetamide
—— 1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C24H25FN4O2
1-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— [(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C20H18FN5O
[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— [(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone —— C20H18ClN5O
[(2S)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-pyridin-3-ylmethanone
—— 2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)acetamide —— C19H19FN6OS
2-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)acetamide
—— 5-(4-chlorophenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine —— C20H20ClN5
5-(4-chlorophenyl)-4-[(2S)-1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]pyrimidin-2-amine
—— 1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one —— C24H25ClN4O2
1-[(2R)-2-[2-amino-5-(4-chlorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one —— C23H23FN4O
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one
—— 1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone —— C22H21FN4O2
1-[(2S)-2-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-phenoxyethanone