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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H29FN4
5-[[(3S)-3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— tert-butyl (4S)-4-(4-tert-butylphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H28N2O2S
tert-butyl (4S)-4-(4-tert-butylphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (2R)-2-[(4-cyclopentylpyrimidin-2-yl)amino]butan-1-ol —— C13H21N3O
(2R)-2-[(4-cyclopentylpyrimidin-2-yl)amino]butan-1-ol
—— 1-[4-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H26N6O
1-[4-[(8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— [(3S)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone —— C20H29N5O2
[(3S)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]-pyrrolidin-1-ylmethanone
—— (2S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]butan-1-ol —— C13H21N3O
(2S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]butan-1-ol
—— 4,6-dimethyl-1-[2-oxo-2-[(2S)-2-(trifluoromethyl)morpholin-4-yl]ethyl]pyrimidin-2-one —— C13H16F3N3O3
4,6-dimethyl-1-[2-oxo-2-[(2S)-2-(trifluoromethyl)morpholin-4-yl]ethyl]pyrimidin-2-one
—— 5-[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2-methylsulfanyl-1H-pyrimidin-6-one —— C14H16N4O2S
5-[(1R)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2-methylsulfanyl-1H-pyrimidin-6-one
—— 5-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2-methylsulfanyl-1H-pyrimidin-6-one —— C14H16N4O2S
5-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2-methylsulfanyl-1H-pyrimidin-6-one
—— (3S)-4-benzyl-3-ethyl-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C22H28N4O2
(3S)-4-benzyl-3-ethyl-1-(4-propylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— tert-butyl (4R)-4-(4-tert-butylphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H28N2O2S
tert-butyl (4R)-4-(4-tert-butylphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [(3S)-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone —— C21H31N5O3
[(3S)-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone
—— (3S)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]pyrrolidin-2-one —— C15H17N5O
(3S)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]pyrrolidin-2-one
—— (3R)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]pyrrolidin-2-one —— C15H17N5O
(3R)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]pyrrolidin-2-one
—— [(3R)-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone —— C21H31N5O3
[(3R)-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-3-yl]-morpholin-4-ylmethanone
—— N-[(3R)-1-(7-acetyl-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-yl]acetamide —— C20H24N6O2
N-[(3R)-1-(7-acetyl-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl)pyrrolidin-3-yl]acetamide
—— 2-(dimethylamino)-4-methyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidine-5-carboxamide —— C15H22N6O
2-(dimethylamino)-4-methyl-N-[(2R)-1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]pyrimidine-5-carboxamide
—— 4-cyclobutyl-6-methyl-N-[(1S)-1-(6-methylpyridin-2-yl)propyl]pyrimidin-2-amine —— C18H24N4
4-cyclobutyl-6-methyl-N-[(1S)-1-(6-methylpyridin-2-yl)propyl]pyrimidin-2-amine
—— ethyl (4R)-6-[(4-bromo-2-chlorophenoxy)methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H16BrClN2O4
ethyl (4R)-6-[(4-bromo-2-chlorophenoxy)methyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 5-(Benzyloxy)-6-methyl-2,4-pyrimidinediol —— C12H12N2O3
5-(Benzyloxy)-6-methyl-2,4-pyrimidinediol
—— 1-[2-pyridin-3-yl-4-[[(1R)-1-pyridin-3-ylethyl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H22N6O
1-[2-pyridin-3-yl-4-[[(1R)-1-pyridin-3-ylethyl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 5-[[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine —— C21H29FN4
5-[[(3R)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine
—— 5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine —— C21H29FN4
5-[[(3S)-3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propylpyrimidin-2-amine
—— (1R)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-phenylethanol —— C17H21N3O
(1R)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-phenylethanol
—— (1S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-phenylethanol —— C17H21N3O
(1S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-1-phenylethanol
—— 1-[2-pyridin-3-yl-4-[[(1S)-1-pyridin-3-ylethyl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C21H22N6O
1-[2-pyridin-3-yl-4-[[(1S)-1-pyridin-3-ylethyl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 4-cyclobutyl-6-methyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine —— C16H21N5
4-cyclobutyl-6-methyl-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine
—— 4-cyclobutyl-6-methyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine —— C16H21N5
4-cyclobutyl-6-methyl-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]pyrimidin-2-amine
—— [4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(3S)-oxolan-3-yl]methanone —— C19H23N5O2
[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(3S)-oxolan-3-yl]methanone
—— 4-[(3S)-3-propoxypiperidin-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine —— C20H27N5O
4-[(3S)-3-propoxypiperidin-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine
—— [4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(3R)-oxolan-3-yl]methanone —— C19H23N5O2
[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(3R)-oxolan-3-yl]methanone
—— 4-cyclobutyl-N-[[(2R)-1-ethylpiperidin-2-yl]methyl]-6-methylpyrimidin-2-amine —— C17H28N4
4-cyclobutyl-N-[[(2R)-1-ethylpiperidin-2-yl]methyl]-6-methylpyrimidin-2-amine
—— 6-(1-methylimidazol-2-yl)-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyridazin-3-amine —— C13H16N8
6-(1-methylimidazol-2-yl)-N-[(2R)-1-(1,2,4-triazol-1-yl)propan-2-yl]pyridazin-3-amine
—— 2-pyridin-2-yl-7-[(2R)-2-pyrrol-1-ylpentanoyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H23N5O2
2-pyridin-2-yl-7-[(2R)-2-pyrrol-1-ylpentanoyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (2S)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxybutan-1-one —— C19H25N5O2
(2S)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxybutan-1-one
—— 2-pyridin-2-yl-7-[(2S)-2-pyrrol-1-ylpentanoyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H23N5O2
2-pyridin-2-yl-7-[(2S)-2-pyrrol-1-ylpentanoyl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 4-[(3R)-3-propoxypiperidin-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine —— C20H27N5O
4-[(3R)-3-propoxypiperidin-1-yl]-2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[3,4-d]pyrimidine
—— N-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C15H20F3N5
N-[(1S)-2-methyl-1-(1-methylimidazol-2-yl)propyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 3-[6-(dimethylamino)pyrimidin-4-yl]-5-[2-[(2S)-piperidin-2-yl]ethyl]phenol —— C19H26N4O
3-[6-(dimethylamino)pyrimidin-4-yl]-5-[2-[(2S)-piperidin-2-yl]ethyl]phenol
—— 3-[6-(dimethylamino)pyrimidin-4-yl]-5-[2-[(2R)-piperidin-2-yl]ethyl]phenol —— C19H26N4O
3-[6-(dimethylamino)pyrimidin-4-yl]-5-[2-[(2R)-piperidin-2-yl]ethyl]phenol
—— N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C15H20F3N5
N-[(1R)-2-methyl-1-(1-methylimidazol-2-yl)propyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— (2R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxybutan-1-one —— C19H25N5O2
(2R)-1-[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxybutan-1-one
—— (2R)-2-[(3-methoxyphenyl)methyl]-4-(6-phenylpyridazin-3-yl)morpholine —— C22H23N3O2
(2R)-2-[(3-methoxyphenyl)methyl]-4-(6-phenylpyridazin-3-yl)morpholine
—— ethyl 2-methylsulfanyl-4-[(3R)-3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]pyrimidine-5-carboxylate —— C17H24N4O3S
ethyl 2-methylsulfanyl-4-[(3R)-3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]pyrimidine-5-carboxylate
—— 1-[4-[[(2R)-2,3-dihydroxypropyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C17H21N5O3
1-[4-[[(2R)-2,3-dihydroxypropyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— (2S)-2-[(3-methoxyphenyl)methyl]-4-(6-phenylpyridazin-3-yl)morpholine —— C22H23N3O2
(2S)-2-[(3-methoxyphenyl)methyl]-4-(6-phenylpyridazin-3-yl)morpholine
—— 6-methyl-5-[[(2S)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C16H27N3O3
6-methyl-5-[[(2S)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(2S)-1-pyridin-4-ylpropan-2-yl]pyrimidin-2-amine —— C19H21N5
4-(2,6-dimethylpyridin-3-yl)-N-[(2S)-1-pyridin-4-ylpropan-2-yl]pyrimidin-2-amine
—— 1-[4-[[(2S)-2,3-dihydroxypropyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C17H21N5O3
1-[4-[[(2S)-2,3-dihydroxypropyl]amino]-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— 5-[[(2R)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione —— C15H25N3O3
5-[[(2R)-2-(4-methylpentyl)morpholin-4-yl]methyl]-1H-pyrimidine-2,4-dione