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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-methyl-2-[(3R)-1-methylpyrrolidin-3-yl]-N-pyrazin-2-ylpyrimidin-4-amine —— C14H18N6
6-methyl-2-[(3R)-1-methylpyrrolidin-3-yl]-N-pyrazin-2-ylpyrimidin-4-amine
—— 4,6-dimethyl-N-[6-methyl-2-[(3S)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C18H26N6
4,6-dimethyl-N-[6-methyl-2-[(3S)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 4,6-dimethyl-N-[6-methyl-2-[(3R)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C21H25N7
4,6-dimethyl-N-[6-methyl-2-[(3R)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 4,6-dimethyl-N-[6-methyl-2-[(2R)-1-methylpyrrolidin-2-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C16H22N6
4,6-dimethyl-N-[6-methyl-2-[(2R)-1-methylpyrrolidin-2-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 2-hydroxy-1-[(2R)-2-(2-methylpyrimidin-4-yl)morpholin-4-yl]ethanone —— C11H15N3O3
2-hydroxy-1-[(2R)-2-(2-methylpyrimidin-4-yl)morpholin-4-yl]ethanone
—— 4-methyl-N-[6-methyl-2-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C15H21N5S
4-methyl-N-[6-methyl-2-[(2S)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 4,6-dimethyl-N-[6-methyl-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C21H25N7
4,6-dimethyl-N-[6-methyl-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 2-[(2S)-2-[4-methyl-6-(pyrimidin-2-ylamino)pyrimidin-2-yl]pyrrolidin-1-yl]ethanol —— C15H20N6O
2-[(2S)-2-[4-methyl-6-(pyrimidin-2-ylamino)pyrimidin-2-yl]pyrrolidin-1-yl]ethanol
—— 2-[(2R)-2-[4-methyl-6-(1,3-thiazol-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol —— C15H21N5OS
2-[(2R)-2-[4-methyl-6-(1,3-thiazol-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol
—— N-[6-methyl-2-(1-propan-2-ylazetidin-3-yl)pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C13H18N6S
N-[6-methyl-2-(1-propan-2-ylazetidin-3-yl)pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— N-[6-methyl-2-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C14H19N5S
N-[6-methyl-2-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 6-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-4-amine —— C17H24N6
6-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-4-amine
—— 1-[3-[4-Methyl-6-(1,3,4-thiadiazol-2-ylamino)pyrimidin-2-yl]azetidin-1-yl]ethanone —— C12H14N6OS
1-[3-[4-Methyl-6-(1,3,4-thiadiazol-2-ylamino)pyrimidin-2-yl]azetidin-1-yl]ethanone
—— 6-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine —— C17H24N6
6-methyl-2-[(2R)-1-propan-2-ylpiperidin-2-yl]-N-pyrimidin-2-ylpyrimidin-4-amine
—— 6-methyl-2-[(2S)-1-methylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-4-amine —— C15H19N5
6-methyl-2-[(2S)-1-methylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-4-amine
—— N-[2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,2-oxazol-3-amine —— C17H21N7O
N-[2-[(3R)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,2-oxazol-3-amine
—— 4-methyl-N-[2-methyl-6-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C15H21N5S
4-methyl-N-[2-methyl-6-[(2R)-1-methylpiperidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 2-[(2S)-2-[4-methyl-6-(pyrazin-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol —— C16H22N6O
2-[(2S)-2-[4-methyl-6-(pyrazin-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol
—— N-[2-[(2R)-1-(2-methoxyethyl)pyrrolidin-2-yl]-6-methylpyrimidin-4-yl]-4,6-dimethylpyrimidin-2-amine —— C18H26N6O
N-[2-[(2R)-1-(2-methoxyethyl)pyrrolidin-2-yl]-6-methylpyrimidin-4-yl]-4,6-dimethylpyrimidin-2-amine
—— 6-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-4-amine —— C17H24N6
6-methyl-2-[(2S)-1-propan-2-ylpiperidin-2-yl]-N-pyrazin-2-ylpyrimidin-4-amine
—— 5-ethyl-N-[6-methyl-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C19H23N7S
5-ethyl-N-[6-methyl-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]pyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 6-methyl-2-[(2S)-1-methylsulfonylpiperidin-2-yl]-N-pyridin-2-ylpyrimidin-4-amine —— C16H21N5O2S
6-methyl-2-[(2S)-1-methylsulfonylpiperidin-2-yl]-N-pyridin-2-ylpyrimidin-4-amine
—— Tert-butyl 3-[2-methyl-6-[(5-methyl-1,3-thiazol-2-yl)amino]pyrimidin-4-yl]azetidine-1-carboxylate —— C17H23N5O2S
Tert-butyl 3-[2-methyl-6-[(5-methyl-1,3-thiazol-2-yl)amino]pyrimidin-4-yl]azetidine-1-carboxylate
—— 5-ethyl-N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine —— C17H22N8S
5-ethyl-N-[2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methylpyrimidin-4-yl]-1,3,4-thiadiazol-2-amine
—— 2-Methoxy-1-[3-[2-methyl-6-(pyrimidin-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]ethanone —— C15H18N6O2
2-Methoxy-1-[3-[2-methyl-6-(pyrimidin-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]ethanone
—— 2-Methoxy-1-[3-[4-methyl-6-(pyrazin-2-ylamino)pyrimidin-2-yl]azetidin-1-yl]ethanone —— C15H18N6O2
2-Methoxy-1-[3-[4-methyl-6-(pyrazin-2-ylamino)pyrimidin-2-yl]azetidin-1-yl]ethanone
—— N-[2-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,3-thiazol-2-amine —— C17H25N5OS
N-[2-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,3-thiazol-2-amine
—— 2-[(2S)-2-[4-methyl-6-(pyrimidin-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol —— C16H22N6O
2-[(2S)-2-[4-methyl-6-(pyrimidin-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol
—— 2-[(2S)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]pyrrolidin-1-yl]ethanol —— C17H24N6O
2-[(2S)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]pyrrolidin-1-yl]ethanol
—— 6-methyl-2-[(3R)-1-methylpyrrolidin-3-yl]-N-pyrimidin-2-ylpyrimidin-4-amine —— C14H18N6
6-methyl-2-[(3R)-1-methylpyrrolidin-3-yl]-N-pyrimidin-2-ylpyrimidin-4-amine
—— N-[2-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-6-methylpyrimidin-4-yl]-4-methyl-1,3-thiazol-2-amine —— C17H25N5OS
N-[2-[(2R)-1-(2-methoxyethyl)piperidin-2-yl]-6-methylpyrimidin-4-yl]-4-methyl-1,3-thiazol-2-amine
—— 2-[(2S)-1-(2-methoxyethyl)piperidin-2-yl]-6-methyl-N-pyrazin-2-ylpyrimidin-4-amine —— C17H24N6O
2-[(2S)-1-(2-methoxyethyl)piperidin-2-yl]-6-methyl-N-pyrazin-2-ylpyrimidin-4-amine
—— 2-[(3R)-1-methylsulfonylpiperidin-3-yl]-3-(1H-pyrazol-4-yl)pyrazine —— C13H17N5O2S
2-[(3R)-1-methylsulfonylpiperidin-3-yl]-3-(1H-pyrazol-4-yl)pyrazine
—— 2-hydroxy-1-[(3S)-3-(4-methylpyrimidin-2-yl)morpholin-4-yl]ethanone —— C11H15N3O3
2-hydroxy-1-[(3S)-3-(4-methylpyrimidin-2-yl)morpholin-4-yl]ethanone
—— 2-[(2R)-2-[4-methyl-6-(pyrazin-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol —— C16H22N6O
2-[(2R)-2-[4-methyl-6-(pyrazin-2-ylamino)pyrimidin-2-yl]piperidin-1-yl]ethanol
—— 2-Methoxy-1-[3-[2-methyl-6-(1,3-thiazol-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]ethanone —— C14H17N5O2S
2-Methoxy-1-[3-[2-methyl-6-(1,3-thiazol-2-ylamino)pyrimidin-4-yl]azetidin-1-yl]ethanone
—— 6-methyl-N-(6-methylpyridin-2-yl)-2-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-amine —— C16H21N5O2S
6-methyl-N-(6-methylpyridin-2-yl)-2-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-amine
—— N-[2-[(2S)-1-(2-methoxyethyl)piperidin-2-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,3-thiazol-2-amine —— C17H25N5OS
N-[2-[(2S)-1-(2-methoxyethyl)piperidin-2-yl]-6-methylpyrimidin-4-yl]-5-methyl-1,3-thiazol-2-amine
—— 2-[(2R)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]pyrrolidin-1-yl]ethanol —— C17H24N6O
2-[(2R)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyrimidin-2-yl]pyrrolidin-1-yl]ethanol
—— (2S)-N,N-dimethyl-2-pyrazin-2-ylmorpholine-4-sulfonamide —— C10H16N4O3S
(2S)-N,N-dimethyl-2-pyrazin-2-ylmorpholine-4-sulfonamide
—— 2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-(3-methylpyridin-2-yl)pyrimidin-4-amine —— C19H23N7
2-[(3S)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-6-methyl-N-(3-methylpyridin-2-yl)pyrimidin-4-amine
—— 4,6-dimethyl-N-[6-methyl-2-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C18H26N6
4,6-dimethyl-N-[6-methyl-2-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 6-methyl-N-(3-methylpyridin-2-yl)-2-[(3S)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-amine —— C18H25N5
6-methyl-N-(3-methylpyridin-2-yl)-2-[(3S)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-amine
—— [(3R)-3-[4-methyl-6-(pyridin-2-ylamino)pyrimidin-2-yl]pyrrolidin-1-yl]-pyrazin-2-ylmethanone —— C19H19N7O
[(3R)-3-[4-methyl-6-(pyridin-2-ylamino)pyrimidin-2-yl]pyrrolidin-1-yl]-pyrazin-2-ylmethanone
—— 6-methyl-N-(3-methylpyridin-2-yl)-2-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-amine —— C18H25N5
6-methyl-N-(3-methylpyridin-2-yl)-2-[(3R)-1-propan-2-ylpyrrolidin-3-yl]pyrimidin-4-amine
—— 6-methyl-2-[(3R)-1-methylsulfonylpyrrolidin-3-yl]-N-pyridin-2-ylpyrimidin-4-amine —— C15H19N5O2S
6-methyl-2-[(3R)-1-methylsulfonylpyrrolidin-3-yl]-N-pyridin-2-ylpyrimidin-4-amine
—— 4,6-dimethyl-N-[6-methyl-2-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine —— C16H22N6O2S
4,6-dimethyl-N-[6-methyl-2-[(3S)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-yl]pyrimidin-2-amine
—— 4-methyl-N-[6-methyl-2-[(2S)-1-methylpyrrolidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine —— C14H19N5S
4-methyl-N-[6-methyl-2-[(2S)-1-methylpyrrolidin-2-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine
—— 2-methyl-N-(3-methylpyridin-2-yl)-6-[(3R)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-amine —— C16H21N5O2S
2-methyl-N-(3-methylpyridin-2-yl)-6-[(3R)-1-methylsulfonylpyrrolidin-3-yl]pyrimidin-4-amine
—— 6-methyl-2-[(2R)-1-methylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-4-amine —— C15H19N5
6-methyl-2-[(2R)-1-methylpyrrolidin-2-yl]-N-pyridin-2-ylpyrimidin-4-amine