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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C22H28N6O3
6-[1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— [(3S)-3-[6-methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]-pyrazin-2-ylmethanone —— C19H20N6O
[(3S)-3-[6-methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]-pyrazin-2-ylmethanone
—— 6-[1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide —— C22H28N6O3
6-[1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-N-[[(2R)-oxolan-2-yl]methyl]pyridine-3-carboxamide
—— N-(2-methoxyethyl)-6-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]pyridine-3-carboxamide —— C20H25N5O3
N-(2-methoxyethyl)-6-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]pyridine-3-carboxamide
—— N,N-dimethyl-6-[(3S)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl]pyridine-3-carboxamide —— C19H24N6O2
N,N-dimethyl-6-[(3S)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl]pyridine-3-carboxamide
—— (2,4-Dimethylpyrimidin-5-yl)-[4-[6-methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]piperidin-1-yl]methanone —— C22H26N6O
(2,4-Dimethylpyrimidin-5-yl)-[4-[6-methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]piperidin-1-yl]methanone
—— 4-[5-[(4,6-dimethylpyrimidin-2-yl)amino]pyridin-2-yl]-N,N-diethylpiperidine-1-sulfonamide —— C20H30N6O2S
4-[5-[(4,6-dimethylpyrimidin-2-yl)amino]pyridin-2-yl]-N,N-diethylpiperidine-1-sulfonamide
—— N,N-dimethyl-4-[5-(pyrazin-2-ylamino)pyridin-2-yl]piperidine-1-sulfonamide —— C16H22N6O2S
N,N-dimethyl-4-[5-(pyrazin-2-ylamino)pyridin-2-yl]piperidine-1-sulfonamide
—— 4-[5-[(4,6-dimethylpyrimidin-2-yl)amino]pyridin-2-yl]-N,N-dimethylpiperidine-1-sulfonamide —— C18H26N6O2S
4-[5-[(4,6-dimethylpyrimidin-2-yl)amino]pyridin-2-yl]-N,N-dimethylpiperidine-1-sulfonamide
—— (5-Methylpyrazin-2-yl)-[4-[5-[(6-methylpyridin-2-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone —— C22H24N6O
(5-Methylpyrazin-2-yl)-[4-[5-[(6-methylpyridin-2-yl)amino]pyridin-2-yl]piperidin-1-yl]methanone
—— N,N-dibutyl-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)acetamide —— C18H26N4O3
N,N-dibutyl-2-(4-cyano-1,3-dioxo-6,7-dihydro-5H-pyrrolo[1,2-c]pyrimidin-2-yl)acetamide
—— (2-Amino-5-methylpyridin-3-yl)-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]methanone —— C18H21N5O2
(2-Amino-5-methylpyridin-3-yl)-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]methanone
—— N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-2,2-dimethylpropanamide —— C15H19N3O3
N-[2-[3-(furan-2-yl)-6-oxopyridazin-1-yl]ethyl]-2,2-dimethylpropanamide
—— 6-(4-Methoxyphenyl)-2-(piperidin-4-ylmethyl)pyridazin-3-one —— C17H21N3O2
6-(4-Methoxyphenyl)-2-(piperidin-4-ylmethyl)pyridazin-3-one
—— N-(1-hydroxy-2-methylpropan-2-yl)-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide —— C23H30N4O3
N-(1-hydroxy-2-methylpropan-2-yl)-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide
—— (1R)-1-(2-chlorophenyl)-N'-[6-(1-ethylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethylethane-1,2-diamine —— C20H25ClN6
(1R)-1-(2-chlorophenyl)-N'-[6-(1-ethylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethylethane-1,2-diamine
—— (2-Amino-5-methylpyridin-3-yl)-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]methanone —— C19H23N5O2
(2-Amino-5-methylpyridin-3-yl)-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-4-yl]methanone
—— N-(2-hydroxyethyl)-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide —— C21H26N4O3
N-(2-hydroxyethyl)-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide
—— (1R)-N'-[6-(5-ethyl-2-methylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethyl-1-(4-methylphenyl)ethane-1,2-diamine —— C22H30N6
(1R)-N'-[6-(5-ethyl-2-methylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethyl-1-(4-methylphenyl)ethane-1,2-diamine
—— N-[1-(3-fluorophenyl)cyclopentyl]pyrimidine-5-carboxamide —— C16H16FN3O
N-[1-(3-fluorophenyl)cyclopentyl]pyrimidine-5-carboxamide
—— (1S)-1-(2-chlorophenyl)-N'-[6-(1-ethylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethylethane-1,2-diamine —— C20H25ClN6
(1S)-1-(2-chlorophenyl)-N'-[6-(1-ethylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethylethane-1,2-diamine
—— N-[2-(2,3-dimethylphenoxy)ethyl]-2-methyl-6-(4-methyl-2-morpholin-4-ylpyrimidin-5-yl)pyrimidin-4-amine —— C24H30N6O2
N-[2-(2,3-dimethylphenoxy)ethyl]-2-methyl-6-(4-methyl-2-morpholin-4-ylpyrimidin-5-yl)pyrimidin-4-amine
—— N-[3-(4-fluorophenyl)propyl]-2-methyl-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C23H30FN5
N-[3-(4-fluorophenyl)propyl]-2-methyl-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— N-[2-(diethylamino)ethyl]-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide —— C25H35N5O2
N-[2-(diethylamino)ethyl]-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide
—— 2-methyl-N-[(4-phenyloxan-4-yl)methyl]-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C26H35N5O
2-methyl-N-[(4-phenyloxan-4-yl)methyl]-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— N-(cyclopropylmethyl)-6-(5-ethyl-4-methyl-1H-pyrazol-3-yl)-2-methylpyrimidin-4-amine —— C15H21N5
N-(cyclopropylmethyl)-6-(5-ethyl-4-methyl-1H-pyrazol-3-yl)-2-methylpyrimidin-4-amine
—— (1S)-N'-[6-(5-ethyl-2-methylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethyl-1-(4-methylphenyl)ethane-1,2-diamine —— C22H30N6
(1S)-N'-[6-(5-ethyl-2-methylpyrazol-3-yl)-2-methylpyrimidin-4-yl]-N,N-dimethyl-1-(4-methylphenyl)ethane-1,2-diamine
—— 4-N-[(2S)-2-(4-fluorophenyl)-2-piperidin-1-ylethyl]-6-(1-methylpyrazol-4-yl)pyrimidine-2,4-diamine —— C21H26FN7
4-N-[(2S)-2-(4-fluorophenyl)-2-piperidin-1-ylethyl]-6-(1-methylpyrazol-4-yl)pyrimidine-2,4-diamine
—— 4-(2-Morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzoic acid —— C19H21N3O3
4-(2-Morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzoic acid
—— N-[3-(2-methoxyphenyl)propyl]-2-methyl-6-(4-methyl-2-morpholin-4-ylpyrimidin-5-yl)pyrimidin-4-amine —— C24H30N6O2
N-[3-(2-methoxyphenyl)propyl]-2-methyl-6-(4-methyl-2-morpholin-4-ylpyrimidin-5-yl)pyrimidin-4-amine
—— 2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C27H37N5O
2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— N-(3-hydroxy-2,2-dimethylpropyl)-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide —— C24H32N4O3
N-(3-hydroxy-2,2-dimethylpropyl)-4-(2-morpholin-4-yl-5,6,7,8-tetrahydroquinazolin-4-yl)benzamide
—— 6-(5-ethyl-2-methylpyrazol-3-yl)-2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]pyrimidin-4-amine —— C24H31N5O
6-(5-ethyl-2-methylpyrazol-3-yl)-2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]pyrimidin-4-amine
—— 2-methyl-N-[(4-phenyloxan-4-yl)methyl]-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C26H35N5O
2-methyl-N-[(4-phenyloxan-4-yl)methyl]-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— 6-(1-ethylpyrazol-4-yl)-4-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine —— C19H23FN6
6-(1-ethylpyrazol-4-yl)-4-N-[(2S)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine
—— 4-N-[(2R)-2-(4-fluorophenyl)-2-piperidin-1-ylethyl]-6-(1-methylpyrazol-4-yl)pyrimidine-2,4-diamine —— C21H26FN7
4-N-[(2R)-2-(4-fluorophenyl)-2-piperidin-1-ylethyl]-6-(1-methylpyrazol-4-yl)pyrimidine-2,4-diamine
—— 6-(1-ethylpyrazol-4-yl)-4-N-[(2R)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine —— C19H23FN6
6-(1-ethylpyrazol-4-yl)-4-N-[(2R)-4-(4-fluorophenyl)butan-2-yl]pyrimidine-2,4-diamine
—— 2-methyl-N-[[4-(4-methylphenyl)oxan-4-yl]methyl]-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C27H37N5O
2-methyl-N-[[4-(4-methylphenyl)oxan-4-yl]methyl]-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[[4-(4-methylphenyl)oxan-4-yl]methyl]-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C27H37N5O
2-methyl-N-[[4-(4-methylphenyl)oxan-4-yl]methyl]-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C27H37N5O
2-methyl-N-[[4-(3-methylphenyl)oxan-4-yl]methyl]-6-[(2R)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— N-[3-(4-fluorophenyl)propyl]-2-methyl-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine —— C23H30FN5
N-[3-(4-fluorophenyl)propyl]-2-methyl-6-[(2S)-1-(3,4,5-trimethylpyrazol-1-yl)propan-2-yl]pyrimidin-4-amine
—— N-[2-methyl-6-[(2R)-1-(3-phenylpropylsulfonyl)pyrrolidin-2-yl]pyridin-4-yl]pyrazin-2-amine —— C23H27N5O2S
N-[2-methyl-6-[(2R)-1-(3-phenylpropylsulfonyl)pyrrolidin-2-yl]pyridin-4-yl]pyrazin-2-amine
—— N-[2-methyl-6-[(2S)-1-(3-phenylpropylsulfonyl)pyrrolidin-2-yl]pyridin-4-yl]pyrazin-2-amine —— C23H27N5O2S
N-[2-methyl-6-[(2S)-1-(3-phenylpropylsulfonyl)pyrrolidin-2-yl]pyridin-4-yl]pyrazin-2-amine
—— N-[2-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]-4,6-dimethylpyrimidin-2-amine —— C21H26N6O3S
N-[2-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]-4,6-dimethylpyrimidin-2-amine
—— N-[2-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]-4,6-dimethylpyrimidin-2-amine —— C21H26N6O3S
N-[2-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]-4,6-dimethylpyrimidin-2-amine
—— N-[2-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]pyrazin-2-amine —— C19H22N6O3S
N-[2-[(2R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]pyrazin-2-amine
—— N-[2-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]pyrazin-2-amine —— C19H22N6O3S
N-[2-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]pyrrolidin-2-yl]-6-methylpyridin-4-yl]pyrazin-2-amine
—— (2S)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide —— C18H26N6O2S
(2S)-2-[4-[(4,6-dimethylpyrimidin-2-yl)amino]-6-methylpyridin-2-yl]-N,N-dimethylpyrrolidine-1-sulfonamide
—— (2R)-N,N-diethyl-2-[6-methyl-4-(pyrazin-2-ylamino)pyridin-2-yl]pyrrolidine-1-sulfonamide —— C18H26N6O2S
(2R)-N,N-diethyl-2-[6-methyl-4-(pyrazin-2-ylamino)pyridin-2-yl]pyrrolidine-1-sulfonamide
—— (2S)-N,N-diethyl-2-[6-methyl-4-(pyrazin-2-ylamino)pyridin-2-yl]pyrrolidine-1-sulfonamide —— C18H26N6O2S
(2S)-N,N-diethyl-2-[6-methyl-4-(pyrazin-2-ylamino)pyridin-2-yl]pyrrolidine-1-sulfonamide