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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1R)-1-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C16H15F3N6O
N-[(1R)-1-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— (4-methylpiperazin-1-yl)-[(3S)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone —— C21H32N6O2
(4-methylpiperazin-1-yl)-[(3S)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone
—— (4S)-4-[[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl]-1-propan-2-ylpyrrolidin-2-one —— C17H26N4O
(4S)-4-[[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl]-1-propan-2-ylpyrrolidin-2-one
—— N-[(1S)-1-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine —— C16H15F3N6O
N-[(1S)-1-(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
—— 3-(6-morpholin-4-ylpyrimidin-4-yl)-5-[2-[(2S)-piperidin-2-yl]ethyl]phenol —— C21H28N4O2
3-(6-morpholin-4-ylpyrimidin-4-yl)-5-[2-[(2S)-piperidin-2-yl]ethyl]phenol
—— (2S)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one —— C19H25N5OS
(2S)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one
—— (4-methylpiperazin-1-yl)-[(3R)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone —— C21H32N6O2
(4-methylpiperazin-1-yl)-[(3R)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidin-3-yl]methanone
—— (4R)-4-[[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl]-1-propan-2-ylpyrrolidin-2-one —— C17H26N4O
(4R)-4-[[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl]-1-propan-2-ylpyrrolidin-2-one
—— (2R)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one —— C19H25N5OS
(2R)-1-[4-(dimethylamino)-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-2-ethylsulfanylpropan-1-one
—— [4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(2R)-2-methyloxolan-2-yl]methanone —— C20H25N5O2
[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(2R)-2-methyloxolan-2-yl]methanone
—— N-methyl-N-[[(2S)-oxan-2-yl]methyl]-2-pyridin-2-ylpyrimidine-5-carboxamide —— C17H20N4O2
N-methyl-N-[[(2S)-oxan-2-yl]methyl]-2-pyridin-2-ylpyrimidine-5-carboxamide
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-thiophen-2-ylacetate —— C13H10N2O3S2
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 2-thiophen-2-ylacetate
—— N-methyl-2-propan-2-yl-N-[(1S)-1-pyridin-3-ylpropyl]pyrimidine-4-carboxamide —— C17H22N4O
N-methyl-2-propan-2-yl-N-[(1S)-1-pyridin-3-ylpropyl]pyrimidine-4-carboxamide
—— (2-amino-4-methylpyrimidin-5-yl)-[(3R)-3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl]methanone —— C20H26N4O2
(2-amino-4-methylpyrimidin-5-yl)-[(3R)-3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl]methanone
—— N-methyl-N-[[(2R)-oxan-2-yl]methyl]-2-pyridin-2-ylpyrimidine-5-carboxamide —— C17H20N4O2
N-methyl-N-[[(2R)-oxan-2-yl]methyl]-2-pyridin-2-ylpyrimidine-5-carboxamide
—— ethyl (4R)-4-[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C22H23FN2O5
ethyl (4R)-4-[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(2S)-2-methyloxolan-2-yl]methanone —— C20H25N5O2
[4-(dimethylamino)-2-pyridin-4-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-[(2S)-2-methyloxolan-2-yl]methanone
—— 5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3R)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
—— (3S)-4-benzyl-3-ethyl-1-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C21H26N4O2
(3S)-4-benzyl-3-ethyl-1-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— 5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine —— C16H21N5O2S
5-methylsulfonyl-4-[(3S)-piperidin-3-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
—— (3R)-4-benzyl-3-ethyl-1-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C21H26N4O2
(3R)-4-benzyl-3-ethyl-1-(2-ethylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— (3S)-N-(2-methoxyethyl)-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide —— C20H31N5O3
(3S)-N-(2-methoxyethyl)-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
—— 4-(2,6-dimethylpyridin-3-yl)-N-[[(3S)-1-ethylpiperidin-3-yl]methyl]-N-methylpyrimidin-2-amine —— C20H29N5
4-(2,6-dimethylpyridin-3-yl)-N-[[(3S)-1-ethylpiperidin-3-yl]methyl]-N-methylpyrimidin-2-amine
—— (4S)-4-(2-chlorophenyl)-6-methyl-5-(morpholine-4-carbonyl)-3,4-dihydro-1H-pyrimidin-2-one —— C16H18ClN3O3
(4S)-4-(2-chlorophenyl)-6-methyl-5-(morpholine-4-carbonyl)-3,4-dihydro-1H-pyrimidin-2-one
—— (3R)-N-(2-methoxyethyl)-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide —— C20H31N5O3
(3R)-N-(2-methoxyethyl)-1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidin-2-amine —— C19H25N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1S)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidin-2-amine
—— (3S)-4-benzyl-3-ethyl-1-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H24N4O3
(3S)-4-benzyl-3-ethyl-1-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— methyl (4R)-4-[4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21ClN2O5
methyl (4R)-4-[4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-methoxyethyl (4R)-6-methyl-4-(3-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H20N2O4
2-methoxyethyl (4R)-6-methyl-4-(3-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— N-[(2R)-1-amino-1-oxopropan-2-yl]-N-ethyl-4-methyl-2-pyridin-3-ylpyrimidine-5-carboxamide —— C16H19N5O2
N-[(2R)-1-amino-1-oxopropan-2-yl]-N-ethyl-4-methyl-2-pyridin-3-ylpyrimidine-5-carboxamide
—— 2-methoxyethyl (4S)-6-methyl-4-(3-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H20N2O4
2-methoxyethyl (4S)-6-methyl-4-(3-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4S)-4-[4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21ClN2O5
methyl (4S)-4-[4-[(2-chlorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (4R)-4-(2-fluorophenyl)-6-methyl-5-(morpholine-4-carbonyl)-3,4-dihydro-1H-pyrimidin-2-one —— C16H18FN3O3
(4R)-4-(2-fluorophenyl)-6-methyl-5-(morpholine-4-carbonyl)-3,4-dihydro-1H-pyrimidin-2-one
—— N-methyl-N-[(2R)-2-morpholin-4-ylpropyl]-2-phenylpyrimidine-5-carboxamide —— C19H24N4O2
N-methyl-N-[(2R)-2-morpholin-4-ylpropyl]-2-phenylpyrimidine-5-carboxamide
—— 4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidin-2-amine —— C19H25N7
4-(2,6-dimethylpyridin-3-yl)-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidin-2-amine
—— 4-(2,6-dimethylpyridin-3-yl)-N-[[(3R)-1-ethylpiperidin-3-yl]methyl]-N-methylpyrimidin-2-amine —— C20H29N5
4-(2,6-dimethylpyridin-3-yl)-N-[[(3R)-1-ethylpiperidin-3-yl]methyl]-N-methylpyrimidin-2-amine
—— N-methyl-N-[(2S)-2-morpholin-4-ylpropyl]-2-phenylpyrimidine-5-carboxamide —— C19H24N4O2
N-methyl-N-[(2S)-2-morpholin-4-ylpropyl]-2-phenylpyrimidine-5-carboxamide
—— (3S)-4-benzyl-3-ethyl-1-(2-methylsulfanylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H24N4O2S
(3S)-4-benzyl-3-ethyl-1-(2-methylsulfanylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— (3R)-4-benzyl-3-ethyl-1-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H24N4O3
(3R)-4-benzyl-3-ethyl-1-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— (4S)-4-(2-fluorophenyl)-6-methyl-5-(morpholine-4-carbonyl)-3,4-dihydro-1H-pyrimidin-2-one —— C16H18FN3O3
(4S)-4-(2-fluorophenyl)-6-methyl-5-(morpholine-4-carbonyl)-3,4-dihydro-1H-pyrimidin-2-one
—— (3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one —— C20H23FN4O2
(3S)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
—— (3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one —— C20H23FN4O2
(3R)-4-[(4-fluorophenyl)methyl]-3-propan-2-yl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
—— 5-[[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine —— C21H28F2N4
5-[[(3R)-3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl]methyl]-N-propan-2-ylpyrimidin-2-amine
—— 1-[4-[[(2R)-1-hydroxyhexan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone —— C20H27N5O2
1-[4-[[(2R)-1-hydroxyhexan-2-yl]amino]-2-pyridin-3-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]ethanone
—— ethyl (4R)-4-ethyl-2-oxo-6-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C15H21N5O3S2
ethyl (4R)-4-ethyl-2-oxo-6-[[5-(prop-2-enylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (3R)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]butanoate —— C17H22N4O2
ethyl (3R)-3-[[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino]butanoate
—— (3R)-4-benzyl-3-ethyl-1-(2-methylsulfanylpyrimidine-5-carbonyl)-1,4-diazepan-5-one —— C20H24N4O2S
(3R)-4-benzyl-3-ethyl-1-(2-methylsulfanylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
—— (2S)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-2-(trifluoromethyl)morpholine —— C16H17F3N4O
(2S)-4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-2-(trifluoromethyl)morpholine
—— 4-cyclopentyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine —— C18H24N4
4-cyclopentyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
—— methyl (4S)-4-[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H21FN2O5
methyl (4S)-4-[4-[(4-fluorophenyl)methoxy]-3-methoxyphenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate