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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[4-[[(2S)-2-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]methyl]phenyl]acetamide —— C25H28ClN5O
N-[4-[[(2S)-2-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]methyl]phenyl]acetamide
—— 4-[(3R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-5-(2-fluorophenyl)-N,N-dimethylpyrimidin-2-amine —— C23H29FN6
4-[(3R)-1-[(1,5-dimethylpyrazol-4-yl)methyl]piperidin-3-yl]-5-(2-fluorophenyl)-N,N-dimethylpyrimidin-2-amine
—— 2-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone —— C22H29N5O2
2-[(2R)-2-[2-amino-5-(3-methoxyphenyl)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone
—— N-[6-[(2R)-pyrrolidin-2-yl]pyridin-2-yl]pyrimidin-2-amine —— C13H15N5
N-[6-[(2R)-pyrrolidin-2-yl]pyridin-2-yl]pyrimidin-2-amine
—— 4-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]piperidin-2-yl]-5-(4-methoxyphenyl)-N,N-dimethylpyrimidin-2-amine —— C24H32N6O
4-[(2R)-1-[(1-ethylpyrazol-4-yl)methyl]piperidin-2-yl]-5-(4-methoxyphenyl)-N,N-dimethylpyrimidin-2-amine
—— 4-[2-(dimethylamino)-4-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide —— C22H29N5O2
4-[2-(dimethylamino)-4-[(3S)-1-(2-methylpropanoyl)piperidin-3-yl]pyrimidin-5-yl]benzamide
—— N-[4-[(2S)-piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C12H15N5S
N-[4-[(2S)-piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— 4-[(2S)-1-benzylpyrrolidin-2-yl]-5-(3-fluorophenyl)-N,N-dimethylpyrimidin-2-amine —— C23H25FN4
4-[(2S)-1-benzylpyrrolidin-2-yl]-5-(3-fluorophenyl)-N,N-dimethylpyrimidin-2-amine
—— [(2R)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(1-methylpyrazol-4-yl)methanone —— C21H23FN6O
[(2R)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(1-methylpyrazol-4-yl)methanone
—— 1-[4-[2-(Dimethylamino)-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(5-methyl-3,4-dihydropyrazol-2-yl)propan-1-one —— C24H31FN6O
1-[4-[2-(Dimethylamino)-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-3-(5-methyl-3,4-dihydropyrazol-2-yl)propan-1-one
—— 3-[4-[1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-2-(dimethylamino)pyrimidin-5-yl]benzamide —— C25H31N5O2
3-[4-[1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-2-(dimethylamino)pyrimidin-5-yl]benzamide
—— N-pyrazin-2-yl-4-[(2S)-pyrrolidin-2-yl]pyrimidin-2-amine —— C12H14N6
N-pyrazin-2-yl-4-[(2S)-pyrrolidin-2-yl]pyrimidin-2-amine
—— 4,6-dimethyl-N-[2-methyl-6-[(2S)-pyrrolidin-2-yl]pyridin-4-yl]pyrimidin-2-amine —— C16H21N5
4,6-dimethyl-N-[2-methyl-6-[(2S)-pyrrolidin-2-yl]pyridin-4-yl]pyrimidin-2-amine
—— 6-[(2S)-1-[(3-chlorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine —— C19H19ClN6O2S
6-[(2S)-1-[(3-chlorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyrazin-2-ylpyrazin-2-amine
—— 5-methyl-N-[6-[(2S)-pyrrolidin-2-yl]pyrazin-2-yl]-1,3,4-thiadiazol-2-amine —— C11H14N6S
5-methyl-N-[6-[(2S)-pyrrolidin-2-yl]pyrazin-2-yl]-1,3,4-thiadiazol-2-amine
—— 4,6-dimethyl-N-[6-[(2S)-pyrrolidin-2-yl]pyrazin-2-yl]pyrimidin-2-amine —— C14H18N6
4,6-dimethyl-N-[6-[(2S)-pyrrolidin-2-yl]pyrazin-2-yl]pyrimidin-2-amine
—— N-[6-[(2S)-pyrrolidin-2-yl]pyridin-2-yl]pyrimidin-2-amine —— C13H15N5
N-[6-[(2S)-pyrrolidin-2-yl]pyridin-2-yl]pyrimidin-2-amine
—— [(2R)-2-[5-(4-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]-(2-methylpyrazol-3-yl)methanone —— C21H23ClN6O
[(2R)-2-[5-(4-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]-(2-methylpyrazol-3-yl)methanone
—— [(3R)-3-[2-(dimethylamino)-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone —— C23H26FN5OS
[(3R)-3-[2-(dimethylamino)-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone
—— 1-[(3S)-3-[2-(dimethylamino)-5-phenylpyrimidin-4-yl]piperidin-1-yl]-3-(3-fluorophenoxy)propan-1-one —— C26H29FN4O2
1-[(3S)-3-[2-(dimethylamino)-5-phenylpyrimidin-4-yl]piperidin-1-yl]-3-(3-fluorophenoxy)propan-1-one
—— N-[4-[[(2R)-2-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]methyl]phenyl]acetamide —— C25H28ClN5O
N-[4-[[(2R)-2-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]methyl]phenyl]acetamide
—— 3-[2-(Dimethylamino)-4-[1-(dimethylsulfamoyl)piperidin-4-yl]pyrimidin-5-yl]benzamide —— C20H28N6O3S
3-[2-(Dimethylamino)-4-[1-(dimethylsulfamoyl)piperidin-4-yl]pyrimidin-5-yl]benzamide
—— [(3R)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-(2,4-dimethyl-1,3-oxazol-5-yl)methanone —— C23H26ClN5O2
[(3R)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-(2,4-dimethyl-1,3-oxazol-5-yl)methanone
—— 5-methyl-N-[6-[(2R)-pyrrolidin-2-yl]pyrazin-2-yl]-1,3,4-thiadiazol-2-amine —— C11H14N6S
5-methyl-N-[6-[(2R)-pyrrolidin-2-yl]pyrazin-2-yl]-1,3,4-thiadiazol-2-amine
—— 4-[(2R)-1-benzylpyrrolidin-2-yl]-5-(3-fluorophenyl)-N,N-dimethylpyrimidin-2-amine —— C23H25FN4
4-[(2R)-1-benzylpyrrolidin-2-yl]-5-(3-fluorophenyl)-N,N-dimethylpyrimidin-2-amine
—— [(3R)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-(1-ethylpyrazol-3-yl)methanone —— C23H27ClN6O
[(3R)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-(1-ethylpyrazol-3-yl)methanone
—— [(2S)-2-[5-(4-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]-(2-methylpyrazol-3-yl)methanone —— C21H23ClN6O
[(2S)-2-[5-(4-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]pyrrolidin-1-yl]-(2-methylpyrazol-3-yl)methanone
—— N-pyrimidin-2-yl-6-[(2R)-pyrrolidin-2-yl]pyrazin-2-amine —— C12H14N6
N-pyrimidin-2-yl-6-[(2R)-pyrrolidin-2-yl]pyrazin-2-amine
—— 1-[(2R)-2-[2-(dimethylamino)-5-phenylpyrimidin-4-yl]pyrrolidin-1-yl]ethanone —— C18H22N4O
1-[(2R)-2-[2-(dimethylamino)-5-phenylpyrimidin-4-yl]pyrrolidin-1-yl]ethanone
—— 4-[(2S)-1-(benzenesulfonyl)pyrrolidin-2-yl]-5-(3-methoxyphenyl)-N,N-dimethylpyrimidin-2-amine —— C23H26N4O3S
4-[(2S)-1-(benzenesulfonyl)pyrrolidin-2-yl]-5-(3-methoxyphenyl)-N,N-dimethylpyrimidin-2-amine
—— 6-[(2S)-1-[(3-fluorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine —— C20H20FN5O2S
6-[(2S)-1-[(3-fluorophenyl)methylsulfonyl]pyrrolidin-2-yl]-N-pyridin-2-ylpyrazin-2-amine
—— N-pyrazin-2-yl-6-[(2R)-pyrrolidin-2-yl]pyrazin-2-amine —— C12H14N6
N-pyrazin-2-yl-6-[(2R)-pyrrolidin-2-yl]pyrazin-2-amine
—— 6-N-methyl-4-N-[4-[(2S)-pyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine —— C13H17N7
6-N-methyl-4-N-[4-[(2S)-pyrrolidin-2-yl]pyrimidin-2-yl]pyrimidine-4,6-diamine
—— N-(3-methylpyridin-2-yl)-6-[(2S)-1-(3-phenylpropylsulfonyl)pyrrolidin-2-yl]pyrazin-2-amine —— C23H27N5O2S
N-(3-methylpyridin-2-yl)-6-[(2S)-1-(3-phenylpropylsulfonyl)pyrrolidin-2-yl]pyrazin-2-amine
—— 1-[(2S)-2-[2-(dimethylamino)-5-(3-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]propan-1-one —— C20H26N4O2
1-[(2S)-2-[2-(dimethylamino)-5-(3-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]propan-1-one
—— 2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol —— C16H19FN4O
2-[(2S)-2-[2-amino-5-(3-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]ethanol
—— 1-[(2R)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone —— C22H24FN5OS
1-[(2R)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethanone
—— 4,6-dimethyl-N-[2-methyl-6-[(2R)-pyrrolidin-2-yl]pyridin-4-yl]pyrimidin-2-amine —— C16H21N5
4,6-dimethyl-N-[2-methyl-6-[(2R)-pyrrolidin-2-yl]pyridin-4-yl]pyrimidin-2-amine
—— 2-[(3R)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone —— C23H30ClN5O
2-[(3R)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone
—— [(2S)-2-[2-(dimethylamino)-5-(3-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C22H25N5O2S
[(2S)-2-[2-(dimethylamino)-5-(3-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— N,N-dimethyl-4-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-5-phenylpyrimidin-2-amine —— C24H30N6
N,N-dimethyl-4-[(3R)-1-[[2-(methylamino)pyridin-3-yl]methyl]piperidin-3-yl]-5-phenylpyrimidin-2-amine
—— 1-[(2S)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone —— C19H23FN4O2
1-[(2S)-2-[2-(dimethylamino)-5-(2-fluorophenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-2-methoxyethanone
—— 4-[(2S)-piperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine —— C13H16N6
4-[(2S)-piperidin-2-yl]-N-pyrazin-2-ylpyrimidin-2-amine
—— [(2R)-2-[2-(dimethylamino)-5-(3-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone —— C22H25N5O2S
[(2R)-2-[2-(dimethylamino)-5-(3-methoxyphenyl)pyrimidin-4-yl]pyrrolidin-1-yl]-(4-methyl-1,3-thiazol-5-yl)methanone
—— [(3S)-3-[2-(dimethylamino)-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(2-methylpyrazol-3-yl)methanone —— C22H25FN6O
[(3S)-3-[2-(dimethylamino)-5-(3-fluorophenyl)pyrimidin-4-yl]piperidin-1-yl]-(2-methylpyrazol-3-yl)methanone
—— N,N-dimethyl-4-[(2S)-1-methylpyrrolidin-2-yl]-5-phenylpyrimidin-2-amine —— C17H22N4
N,N-dimethyl-4-[(2S)-1-methylpyrrolidin-2-yl]-5-phenylpyrimidin-2-amine
—— N-[4-[(2R)-piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine —— C12H15N5S
N-[4-[(2R)-piperidin-2-yl]pyrimidin-2-yl]-1,3-thiazol-2-amine
—— 2-[(3S)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone —— C23H30ClN5O
2-[(3S)-3-[5-(3-chlorophenyl)-2-(dimethylamino)pyrimidin-4-yl]piperidin-1-yl]-1-pyrrolidin-1-ylethanone
—— 4-[(2R)-1-[(2,8-dimethylimidazo[1,2-a]pyridin-3-yl)methyl]pyrrolidin-2-yl]-5-(3-fluorophenyl)-N,N-dimethylpyrimidin-2-amine —— C26H29FN6
4-[(2R)-1-[(2,8-dimethylimidazo[1,2-a]pyridin-3-yl)methyl]pyrrolidin-2-yl]-5-(3-fluorophenyl)-N,N-dimethylpyrimidin-2-amine
—— 4,6-dimethyl-N-[6-[(2R)-pyrrolidin-2-yl]pyrazin-2-yl]pyrimidin-2-amine —— C14H18N6
4,6-dimethyl-N-[6-[(2R)-pyrrolidin-2-yl]pyrazin-2-yl]pyrimidin-2-amine