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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-benzyl-4-chloro-5-[[(2S)-1-(furan-2-yl)propan-2-yl]amino]pyridazin-3-one —— C18H18ClN3O2
2-benzyl-4-chloro-5-[[(2S)-1-(furan-2-yl)propan-2-yl]amino]pyridazin-3-one
—— N-methyl-N-[(1R)-2-methyl-1-(2-methylphenyl)propyl]imidazo[1,2-a]pyrazine-8-carboxamide —— C19H22N4O
N-methyl-N-[(1R)-2-methyl-1-(2-methylphenyl)propyl]imidazo[1,2-a]pyrazine-8-carboxamide
—— N-(cyclopropylmethylsulfonyl)-2-phenylpyrimidine-5-carboxamide —— C15H15N3O3S
N-(cyclopropylmethylsulfonyl)-2-phenylpyrimidine-5-carboxamide
—— N-[(S)-cyano-(2,4-difluorophenyl)methyl]imidazo[1,2-a]pyrazine-8-carboxamide —— C15H9F2N5O
N-[(S)-cyano-(2,4-difluorophenyl)methyl]imidazo[1,2-a]pyrazine-8-carboxamide
—— 1-prop-2-ynyl-3-[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]urea —— C16H16N4O
1-prop-2-ynyl-3-[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]urea
—— 2-cyclopropyl-4-methyl-6-methylsulfanyl-N-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrimidine-5-carboxamide —— C16H20N4OS2
2-cyclopropyl-4-methyl-6-methylsulfanyl-N-[(1R)-1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrimidine-5-carboxamide
—— N-[(3-chlorophenyl)methyl]-2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]acetamide —— C17H17ClN4O2S2
N-[(3-chlorophenyl)methyl]-2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]acetamide
—— 3-N-[(2S)-4-(3,4-difluorophenyl)butan-2-yl]pyrazine-2,3-dicarboxamide —— C16H16F2N4O2
3-N-[(2S)-4-(3,4-difluorophenyl)butan-2-yl]pyrazine-2,3-dicarboxamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1S,2R)-2-methylcyclohexyl]acetamide —— C17H24N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1S,2R)-2-methylcyclohexyl]acetamide
—— 2-Ethyl-7-[(3-methylphenyl)methylsulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C16H17N3OS2
2-Ethyl-7-[(3-methylphenyl)methylsulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1R)-1-(4-ethylphenyl)ethyl]acetamide —— C20H24N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1R)-1-(4-ethylphenyl)ethyl]acetamide
—— 3-N-[(1S)-1-(1-benzothiophen-3-yl)ethyl]pyrazine-2,3-dicarboxamide —— C16H14N4O2S
3-N-[(1S)-1-(1-benzothiophen-3-yl)ethyl]pyrazine-2,3-dicarboxamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(2,2,2-trifluoroethyl)acetamide —— C12H13F3N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(2,2,2-trifluoroethyl)acetamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(2S)-3-methylbutan-2-yl]acetamide —— C15H22N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(2S)-3-methylbutan-2-yl]acetamide
—— 3-N-[(1R)-1-(1-benzothiophen-3-yl)ethyl]pyrazine-2,3-dicarboxamide —— C16H14N4O2S
3-N-[(1R)-1-(1-benzothiophen-3-yl)ethyl]pyrazine-2,3-dicarboxamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1R,2S)-2-methylcyclohexyl]acetamide —— C17H24N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1R,2S)-2-methylcyclohexyl]acetamide
—— 2-Ethyl-7-[(4-fluorophenyl)methylsulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C15H14FN3OS2
2-Ethyl-7-[(4-fluorophenyl)methylsulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(thiophen-2-ylmethyl)acetamide —— C15H16N4O2S3
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(thiophen-2-ylmethyl)acetamide
—— N-[(R)-cyano-(2,4-difluorophenyl)methyl]imidazo[1,2-a]pyrazine-8-carboxamide —— C15H9F2N5O
N-[(R)-cyano-(2,4-difluorophenyl)methyl]imidazo[1,2-a]pyrazine-8-carboxamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(2S)-pentan-2-yl]acetamide —— C15H22N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(2S)-pentan-2-yl]acetamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1R,2R)-2-methylcyclohexyl]acetamide —— C17H24N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(1R,2R)-2-methylcyclohexyl]acetamide
—— ethyl (4S)-4-ethyl-2-oxo-6-[(4-pentyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H27N5O3S
ethyl (4S)-4-ethyl-2-oxo-6-[(4-pentyl-1,2,4-triazol-3-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 7-[(2-Bromophenyl)methylsulfanylmethyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C15H14BrN3OS2
7-[(2-Bromophenyl)methylsulfanylmethyl]-2-ethyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 2-Ethyl-7-[(2-fluorophenyl)methylsulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C15H14FN3OS2
2-Ethyl-7-[(2-fluorophenyl)methylsulfanylmethyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N,N-dimethylacetamide —— C12H16N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N,N-dimethylacetamide
—— (2S)-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide —— C16H20N4O
(2S)-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide
—— (2R)-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide —— C16H20N4O
(2R)-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide
—— N-[(2S)-butan-2-yl]-2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]acetamide —— C14H20N4O2S2
N-[(2S)-butan-2-yl]-2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]acetamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(3-phenylpropyl)acetamide —— C19H22N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(3-phenylpropyl)acetamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(3-methylbutyl)acetamide —— C15H22N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(3-methylbutyl)acetamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(3-methoxypropyl)acetamide —— C14H20N4O3S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(3-methoxypropyl)acetamide
—— ethyl (4R)-4-[4-[bis(2-chloroethyl)amino]-2-chlorophenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H22Cl3N3O3
ethyl (4R)-4-[4-[bis(2-chloroethyl)amino]-2-chlorophenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (2R)-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide —— C16H20N4O
(2R)-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(4-fluorophenyl)methyl]acetamide —— C17H17FN4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-[(4-fluorophenyl)methyl]acetamide
—— (2S)-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide —— C16H20N4O
(2S)-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]butanamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-pentan-3-ylacetamide —— C15H22N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-pentan-3-ylacetamide
—— (2S)-N-tert-butyl-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide —— C19H26N4O
(2S)-N-tert-butyl-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(2-phenylethyl)acetamide —— C18H20N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-(2-phenylethyl)acetamide
—— (2R)-N-tert-butyl-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide —— C19H26N4O
(2R)-N-tert-butyl-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide
—— (2S)-N-tert-butyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide —— C19H26N4O
(2S)-N-tert-butyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide
—— (3S)-1-methyl-3-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]pyrrolidin-2-one —— C17H20N4O
(3S)-1-methyl-3-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]pyrrolidin-2-one
—— (3R)-1-methyl-3-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]pyrrolidin-2-one —— C17H20N4O
(3R)-1-methyl-3-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]pyrrolidin-2-one
—— (3R)-1-methyl-3-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]pyrrolidin-2-one —— C17H20N4O
(3R)-1-methyl-3-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]pyrrolidin-2-one
—— N'-[(2S)-2,3-dihydro-1-benzofuran-2-carbonyl]pyrazine-2-carbohydrazide —— C14H12N4O3
N'-[(2S)-2,3-dihydro-1-benzofuran-2-carbonyl]pyrazine-2-carbohydrazide
—— (2S)-2-phenyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]acetamide —— C20H20N4O
(2S)-2-phenyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]acetamide
—— (2R)-2-phenyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]acetamide —— C20H20N4O
(2R)-2-phenyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]acetamide
—— (2R)-N-tert-butyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide —— C19H26N4O
(2R)-N-tert-butyl-2-[[(1S)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]propanamide
—— (2S)-2-phenyl-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]acetamide —— C20H20N4O
(2S)-2-phenyl-2-[[(1R)-1-(4-pyrimidin-5-ylphenyl)ethyl]amino]acetamide
—— N-[(1R)-1-(2-chlorophenyl)ethyl]-2-cyclopropyl-4-methyl-6-methylsulfanylpyrimidine-5-carboxamide —— C18H20ClN3OS
N-[(1R)-1-(2-chlorophenyl)ethyl]-2-cyclopropyl-4-methyl-6-methylsulfanylpyrimidine-5-carboxamide
—— 2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-propan-2-ylacetamide —— C13H18N4O2S2
2-[(2-ethyl-5-oxo-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl)methylsulfanyl]-N-propan-2-ylacetamide