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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-methyl-7-[[[(2R,3S)-3-pyrazol-1-ylbutan-2-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H19N5OS
3-methyl-7-[[[(2R,3S)-3-pyrazol-1-ylbutan-2-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide —— C23H25ClN4O3
N-[(2R)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide
—— 7-[[4-[3-[(2S)-oxolan-2-yl]propanoyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H24N4O3S
7-[[4-[3-[(2S)-oxolan-2-yl]propanoyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide —— C23H25ClN4O3
N-[(2S)-2-(2-chlorophenyl)-2-morpholin-4-ylethyl]-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide
—— [4-[(2S)-2-hydroxybutyl]piperazin-1-yl]-(2-methylpyrimidin-4-yl)methanone —— C14H22N4O2
[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]-(2-methylpyrimidin-4-yl)methanone
—— [4-[(2R)-2-hydroxybutyl]piperazin-1-yl]-(2-methylpyrimidin-4-yl)methanone —— C14H22N4O2
[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]-(2-methylpyrimidin-4-yl)methanone
—— 7-[[4-[3-[(2R)-oxolan-2-yl]propanoyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H24N4O3S
7-[[4-[3-[(2R)-oxolan-2-yl]propanoyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 2-[(2R)-2-(2-chlorophenyl)-2-hydroxyethyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile —— C17H18ClN3O2
2-[(2R)-2-(2-chlorophenyl)-2-hydroxyethyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile
—— 2-[(2S)-2-(2-chlorophenyl)-2-hydroxyethyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile —— C17H18ClN3O2
2-[(2S)-2-(2-chlorophenyl)-2-hydroxyethyl]-5,6-diethyl-3-oxopyridazine-4-carbonitrile
—— ethyl (4R)-4-ethyl-2-oxo-6-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H19N5O4S
ethyl (4R)-4-ethyl-2-oxo-6-[(5-pyridin-3-yl-1,3,4-oxadiazol-2-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1,3-dimethyl-6-[[(2R)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]pyrimidine-2,4-dione —— C17H25N5O2
1,3-dimethyl-6-[[(2R)-2-(1,3,5-trimethylpyrazol-4-yl)pyrrolidin-1-yl]methyl]pyrimidine-2,4-dione
—— ethyl (4R)-4-ethyl-2-oxo-6-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H25N5O3S
ethyl (4R)-4-ethyl-2-oxo-6-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 1,3-dimethyl-6-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C15H22N6O2
1,3-dimethyl-6-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— ethyl (4S)-4-ethyl-2-oxo-6-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H25N5O3S
ethyl (4S)-4-ethyl-2-oxo-6-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylsulfanylmethyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 3-methyl-7-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H20N6OS
3-methyl-7-[[(2S)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 1,3-dimethyl-6-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C15H22N6O2
1,3-dimethyl-6-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— 3-methyl-7-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H21N5OS
3-methyl-7-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 3-methyl-7-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H20N6OS
3-methyl-7-[[(2R)-2-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 3-methyl-7-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H21N5OS
3-methyl-7-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 1,3-dimethyl-6-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C17H25N5O2
1,3-dimethyl-6-[[(2R)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— 1,3-dimethyl-6-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C17H25N5O2
1,3-dimethyl-6-[[(2S)-2-[(4-methylpyrazol-1-yl)methyl]piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— (6S)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H19N7
(6S)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 1,3-dimethyl-6-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C15H22N6O2
1,3-dimethyl-6-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— 1,3-dimethyl-6-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione —— C15H22N6O2
1,3-dimethyl-6-[[(3R)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]pyrimidine-2,4-dione
—— (6R)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H19N7
(6R)-2-methyl-N-(6-methyl-2-pyridin-4-ylpyrimidin-4-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— N-[(2R)-butan-2-yl]-N-butyl-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide —— C19H27N3O2
N-[(2R)-butan-2-yl]-N-butyl-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide
—— N-[(2R)-butan-2-yl]-N-butyl-5-methylpyrazine-2-carboxamide —— C14H23N3O
N-[(2R)-butan-2-yl]-N-butyl-5-methylpyrazine-2-carboxamide
—— N-[(2S)-butan-2-yl]-N-butyl-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide —— C19H27N3O2
N-[(2S)-butan-2-yl]-N-butyl-6-oxo-1-phenyl-4,5-dihydropyridazine-3-carboxamide
—— N-[(2S)-butan-2-yl]-N-butyl-5-methylpyrazine-2-carboxamide —— C14H23N3O
N-[(2S)-butan-2-yl]-N-butyl-5-methylpyrazine-2-carboxamide
—— N-[(2S)-butan-2-yl]-N-butyl-2-[1-(4,6-dimethylpyrimidin-2-yl)-3,5-dimethylpyrazol-4-yl]acetamide —— C21H33N5O
N-[(2S)-butan-2-yl]-N-butyl-2-[1-(4,6-dimethylpyrimidin-2-yl)-3,5-dimethylpyrazol-4-yl]acetamide
—— N-[(2R)-butan-2-yl]-N-butyl-2-[1-(4,6-dimethylpyrimidin-2-yl)-3,5-dimethylpyrazol-4-yl]acetamide —— C21H33N5O
N-[(2R)-butan-2-yl]-N-butyl-2-[1-(4,6-dimethylpyrimidin-2-yl)-3,5-dimethylpyrazol-4-yl]acetamide
—— (3-aminopyrazin-2-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C14H18N6O
(3-aminopyrazin-2-yl)-[(2S)-2-[(4-methylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— 3-methyl-7-[[[(2R)-1-(4-methylpyrazol-1-yl)propan-2-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H19N5OS
3-methyl-7-[[[(2R)-1-(4-methylpyrazol-1-yl)propan-2-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 3-methyl-7-[[[(2S)-1-(4-methylpyrazol-1-yl)propan-2-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H19N5OS
3-methyl-7-[[[(2S)-1-(4-methylpyrazol-1-yl)propan-2-yl]amino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (3-aminopyrazin-2-yl)-[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone —— C15H20N6O
(3-aminopyrazin-2-yl)-[(2S)-2-[(3,5-dimethylpyrazol-1-yl)methyl]pyrrolidin-1-yl]methanone
—— (3-aminopyrazin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C14H18N6O
(3-aminopyrazin-2-yl)-[(2R)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (3-aminopyrazin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone —— C14H18N6O
(3-aminopyrazin-2-yl)-[(2S)-2-(pyrazol-1-ylmethyl)piperidin-1-yl]methanone
—— (3-aminopyrazin-2-yl)-[4-[(2S)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]methanone —— C15H25N5O2
(3-aminopyrazin-2-yl)-[4-[(2S)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]methanone
—— (3-aminopyrazin-2-yl)-[4-[(2R)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]methanone —— C15H25N5O2
(3-aminopyrazin-2-yl)-[4-[(2R)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone —— C15H23ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2R)-2-hydroxypropyl]piperazin-1-yl]methanone
—— (5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone —— C15H23ClN4O2
(5-chloro-2-propan-2-ylpyrimidin-4-yl)-[4-[(2S)-2-hydroxypropyl]piperazin-1-yl]methanone
—— N-(cyclohexen-1-yl)-2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-(furan-2-ylmethyl)acetamide —— C17H17Cl2N3O3
N-(cyclohexen-1-yl)-2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-(furan-2-ylmethyl)acetamide
—— {5-Oxo-5H-[1,3]thiazolo[3,2-A]pyrimidin-7-YL}methyl 2-phenylacetate —— C15H12N2O3S
{5-Oxo-5H-[1,3]thiazolo[3,2-A]pyrimidin-7-YL}methyl 2-phenylacetate
—— ethyl (4S)-6-[[5-(benzylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H21N5O3S2
ethyl (4S)-6-[[5-(benzylamino)-1,3,4-thiadiazol-2-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— [2-[Cyclohexen-1-yl(furan-2-ylmethyl)amino]-2-oxoethyl] 5-methylpyrazine-2-carboxylate —— C19H21N3O4
[2-[Cyclohexen-1-yl(furan-2-ylmethyl)amino]-2-oxoethyl] 5-methylpyrazine-2-carboxylate
—— [(1S)-1-(furan-2-yl)-2-[(2-pyridin-3-ylquinazolin-4-yl)amino]ethyl]-dimethylazanium —— C21H22N5O+
[(1S)-1-(furan-2-yl)-2-[(2-pyridin-3-ylquinazolin-4-yl)amino]ethyl]-dimethylazanium
—— (4-methylpyrimidin-5-yl)-[(2R)-2-[(2R)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methanone —— C15H22N4O
(4-methylpyrimidin-5-yl)-[(2R)-2-[(2R)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methanone
—— ethyl (4R)-6-[3-(benzenesulfonyl)propanoyloxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H22N2O7S
ethyl (4R)-6-[3-(benzenesulfonyl)propanoyloxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (4-methylpyrimidin-5-yl)-[(2R)-2-[(2S)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methanone —— C15H22N4O
(4-methylpyrimidin-5-yl)-[(2R)-2-[(2S)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methanone
—— (4-methylpyrimidin-5-yl)-[(2S)-2-[(2S)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methanone —— C15H22N4O
(4-methylpyrimidin-5-yl)-[(2S)-2-[(2S)-1-methylpyrrolidin-2-yl]pyrrolidin-1-yl]methanone