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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-(2,5-dimethylphenyl)-2-[(2S)-3-[(2-fluorophenyl)methoxy]-2-hydroxypropyl]phthalazin-1-one —— C26H25FN2O3
4-(2,5-dimethylphenyl)-2-[(2S)-3-[(2-fluorophenyl)methoxy]-2-hydroxypropyl]phthalazin-1-one
—— 4-(trifluoromethyl)-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrimidin-2-amine —— C13H16F3N5
4-(trifluoromethyl)-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrimidin-2-amine
—— 1,3-dimethyl-2,4-dioxo-6-[[(2R)-1-(2,2,2-trifluoroethoxy)propan-2-yl]amino]pyrimidine-5-carbonitrile —— C12H15F3N4O3
1,3-dimethyl-2,4-dioxo-6-[[(2R)-1-(2,2,2-trifluoroethoxy)propan-2-yl]amino]pyrimidine-5-carbonitrile
—— 4-(trifluoromethyl)-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrimidin-2-amine —— C13H16F3N5
4-(trifluoromethyl)-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyrimidin-2-amine
—— 1,3-dimethyl-2,4-dioxo-6-[[(2S)-1-(2,2,2-trifluoroethoxy)propan-2-yl]amino]pyrimidine-5-carbonitrile —— C12H15F3N4O3
1,3-dimethyl-2,4-dioxo-6-[[(2S)-1-(2,2,2-trifluoroethoxy)propan-2-yl]amino]pyrimidine-5-carbonitrile
—— methyl (4R)-4-(6-bromo-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17BrN2O4S
methyl (4R)-4-(6-bromo-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— methyl (4S)-4-(6-bromo-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H17BrN2O4S
methyl (4S)-4-(6-bromo-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 7-[[4-[(3S)-oxolane-3-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H20N4O3S
7-[[4-[(3S)-oxolane-3-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 2-[(2S)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-4-(4-methylphenyl)phthalazin-1-one —— C24H20Cl2N2O3
2-[(2S)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-4-(4-methylphenyl)phthalazin-1-one
—— 7-[[4-[(3R)-oxolane-3-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C16H20N4O3S
7-[[4-[(3R)-oxolane-3-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— ethyl (4S)-4-ethyl-6-(4-methylpentanoyloxymethyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H26N2O5
ethyl (4S)-4-ethyl-6-(4-methylpentanoyloxymethyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— 2-[(2R)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-4-(4-methylphenyl)phthalazin-1-one —— C24H20Cl2N2O3
2-[(2R)-3-(2,6-dichlorophenoxy)-2-hydroxypropyl]-4-(4-methylphenyl)phthalazin-1-one
—— N-[(2R)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]tetrazolo[1,5-b]pyridazin-6-amine —— C16H18FN7O
N-[(2R)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]tetrazolo[1,5-b]pyridazin-6-amine
—— 7-ethyl-2-[[(2S,3S)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C13H20N4OS
7-ethyl-2-[[(2S,3S)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-ethyl-2-[[(2R,3R)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C13H20N4OS
7-ethyl-2-[[(2R,3R)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-ethyl-2-[[(2R,3S)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C13H20N4OS
7-ethyl-2-[[(2R,3S)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— N-[(2S)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]tetrazolo[1,5-b]pyridazin-6-amine —— C16H18FN7O
N-[(2S)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]tetrazolo[1,5-b]pyridazin-6-amine
—— 7-ethyl-2-[[(2S,3R)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C13H20N4OS
7-ethyl-2-[[(2S,3R)-3-methylpentan-2-yl]amino]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— N-[[(1R)-cyclohex-3-en-1-yl]methyl]-2-(4-methyl-6-oxo-2-pyridin-4-yl-1H-pyrimidin-5-yl)acetamide —— C19H22N4O2
N-[[(1R)-cyclohex-3-en-1-yl]methyl]-2-(4-methyl-6-oxo-2-pyridin-4-yl-1H-pyrimidin-5-yl)acetamide
—— N-[[(1S)-cyclohex-3-en-1-yl]methyl]-2-(4-methyl-6-oxo-2-pyridin-4-yl-1H-pyrimidin-5-yl)acetamide —— C19H22N4O2
N-[[(1S)-cyclohex-3-en-1-yl]methyl]-2-(4-methyl-6-oxo-2-pyridin-4-yl-1H-pyrimidin-5-yl)acetamide
—— (3S)-1-[5-chloro-2-(diethylamino)pyrimidine-4-carbonyl]pyrrolidine-3-carboxamide —— C14H20ClN5O2
(3S)-1-[5-chloro-2-(diethylamino)pyrimidine-4-carbonyl]pyrrolidine-3-carboxamide
—— 6-cyclopropyl-4-(trifluoromethyl)-2-[[(6R)-2,2,6-trimethylmorpholin-4-yl]methyl]pyridazin-3-one —— C16H22F3N3O2
6-cyclopropyl-4-(trifluoromethyl)-2-[[(6R)-2,2,6-trimethylmorpholin-4-yl]methyl]pyridazin-3-one
—— 1-cyclopropyl-3-[2-[(2S)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile —— C16H20N4O4
1-cyclopropyl-3-[2-[(2S)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile
—— 1-cyclopropyl-3-[2-[(2R)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile —— C16H20N4O4
1-cyclopropyl-3-[2-[(2R)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile
—— 2-[2-[(2R)-2-ethylmorpholin-4-yl]-2-oxoethyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile —— C15H20N4O3
2-[2-[(2R)-2-ethylmorpholin-4-yl]-2-oxoethyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile
—— 2-[2-[(2S)-2-ethylmorpholin-4-yl]-2-oxoethyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile —— C15H20N4O3
2-[2-[(2S)-2-ethylmorpholin-4-yl]-2-oxoethyl]-5,6-dimethyl-3-oxopyridazine-4-carbonitrile
—— (3-aminopyrazin-2-yl)-[(3R)-3-[(2S,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]methanone —— C16H25N5O
(3-aminopyrazin-2-yl)-[(3R)-3-[(2S,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]methanone
—— 1-ethyl-3-[2-[(2S)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile —— C15H20N4O4
1-ethyl-3-[2-[(2S)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile
—— 2-methyl-7-[[(3R)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C15H20N6O2S
2-methyl-7-[[(3R)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— (3-aminopyrazin-2-yl)-[(3R)-3-[(2R,5R)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]methanone —— C16H25N5O
(3-aminopyrazin-2-yl)-[(3R)-3-[(2R,5R)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]methanone
—— [(3R)-3-[(2S,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C17H26N4O
[(3R)-3-[(2S,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— 1-ethyl-3-[2-[(2R)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile —— C15H20N4O4
1-ethyl-3-[2-[(2R)-2-ethylmorpholin-4-yl]-2-oxoethyl]-2,4-dioxopyrimidine-5-carbonitrile
—— [(3R)-3-[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C17H26N4O
[(3R)-3-[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3S)-3-[(2S,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C17H26N4O
[(3S)-3-[(2S,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3S)-3-[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone —— C17H26N4O
[(3S)-3-[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]piperidin-1-yl]-(5-methylpyrazin-2-yl)methanone
—— 7-[[(3R)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H19N5O2S
7-[[(3R)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 2-methyl-7-[[(3S)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one —— C15H20N6O2S
2-methyl-7-[[(3S)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
—— 7-[[(3S)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H19N5O2S
7-[[(3S)-3-(2-oxoimidazolidin-1-yl)piperidin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (3R,6S)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide —— C14H18N4O3S
(3R,6S)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide
—— (3R,6R)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide —— C14H18N4O3S
(3R,6R)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide
—— (3S,6S)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide —— C14H18N4O3S
(3S,6S)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide
—— (3S,6R)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide —— C14H18N4O3S
(3S,6R)-6-methyl-1-(5-oxo-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl)piperidine-3-carboxamide
—— ethyl (4S)-6-[[4-amino-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C12H15F3N6O3S
ethyl (4S)-6-[[4-amino-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[4-amino-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C12H15F3N6O3S
ethyl (4R)-6-[[4-amino-5-(trifluoromethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (3-aminopyrazin-2-yl)-[4-[(2R)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone —— C15H23N5O2
(3-aminopyrazin-2-yl)-[4-[(2R)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone
—— (3-aminopyrazin-2-yl)-[4-[(2S)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone —— C15H23N5O2
(3-aminopyrazin-2-yl)-[4-[(2S)-2-methylmorpholin-4-yl]piperidin-1-yl]methanone
—— 2-(2-bromobenzyl)-4,5-dichloropyridazin-3(2H)-one —— C11H7BrCl2N2O
2-(2-bromobenzyl)-4,5-dichloropyridazin-3(2H)-one
—— 2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(2R)-1-methoxypropan-2-yl]acetamide —— C10H13Cl2N3O3
2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(2R)-1-methoxypropan-2-yl]acetamide
—— N-[(1R)-1-cyano-1-cyclopropylethyl]-2-(4,5-dichloro-6-oxopyridazin-1-yl)acetamide —— C12H12Cl2N4O2
N-[(1R)-1-cyano-1-cyclopropylethyl]-2-(4,5-dichloro-6-oxopyridazin-1-yl)acetamide
—— 2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(2S)-1-methoxypropan-2-yl]acetamide —— C10H13Cl2N3O3
2-(4,5-dichloro-6-oxopyridazin-1-yl)-N-[(2S)-1-methoxypropan-2-yl]acetamide