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二嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(2S)-2-[2-methyl-6-[2-[(S)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C14H22N4O3S
1-[(2S)-2-[2-methyl-6-[2-[(S)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— 2-methyl-6-[(2S)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C13H18N6O2
2-methyl-6-[(2S)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine —— C15H21N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-(5-methylpyrazol-1-yl)ethyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine —— C15H22N6O
2-methyl-N-[2-(5-methylpyrazol-1-yl)ethyl]-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-(6-amino-2-methylpyrimidin-4-yl)morpholin-4-yl]-3-phenylpropan-1-one —— C18H22N4O2
1-[(2R)-2-(6-amino-2-methylpyrimidin-4-yl)morpholin-4-yl]-3-phenylpropan-1-one
—— N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine —— C14H20N6O2
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-6-[(2S)-morpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-6-[(2S)-4-methylmorpholin-2-yl]-N-[2-[(R)-methylsulfinyl]ethyl]pyrimidin-4-amine —— C13H22N4O2S
2-methyl-6-[(2S)-4-methylmorpholin-2-yl]-N-[2-[(R)-methylsulfinyl]ethyl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2R)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C15H21N5OS
N,2-dimethyl-6-[(2R)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine —— C18H27N5O2
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-methyl-6-[(2S)-4-propan-2-ylmorpholin-2-yl]pyrimidin-4-amine
—— 2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-[(R)-methylsulfinyl]ethyl]pyrimidin-4-amine —— C13H22N4O2S
2-methyl-6-[(2R)-4-methylmorpholin-2-yl]-N-[2-[(R)-methylsulfinyl]ethyl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2S)-4-[[2-(methylamino)pyridin-3-yl]methyl]morpholin-2-yl]pyrimidin-4-amine —— C17H24N6O
N,2-dimethyl-6-[(2S)-4-[[2-(methylamino)pyridin-3-yl]methyl]morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2S)-2-[2-methyl-6-[2-[(R)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C14H22N4O3S
1-[(2S)-2-[2-methyl-6-[2-[(R)-methylsulfinyl]ethylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— 2-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[(2S)-1-methylsulfonylazetidin-2-yl]pyrimidin-4-amine —— C13H18N6O3S
2-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[(2S)-1-methylsulfonylazetidin-2-yl]pyrimidin-4-amine
—— 2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine —— C12H20N4O2S
2-methyl-N-[2-[(S)-methylsulfinyl]ethyl]-6-[(2R)-morpholin-2-yl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2S)-4-(oxan-4-yl)morpholin-2-yl]pyrimidin-4-amine —— C15H24N4O2
N,2-dimethyl-6-[(2S)-4-(oxan-4-yl)morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-[2-methyl-6-[(4-methylthiadiazol-5-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone —— C15H20N6O2S
1-[(2R)-2-[2-methyl-6-[(4-methylthiadiazol-5-yl)methylamino]pyrimidin-4-yl]morpholin-4-yl]ethanone
—— 1-[(2R)-2-[2-methyl-6-(2-pyrazin-2-ylethylamino)pyrimidin-4-yl]morpholin-4-yl]ethanone —— C17H22N6O2
1-[(2R)-2-[2-methyl-6-(2-pyrazin-2-ylethylamino)pyrimidin-4-yl]morpholin-4-yl]ethanone
—— N,2-dimethyl-6-[(2S)-4-methylsulfonylmorpholin-2-yl]pyrimidin-4-amine —— C11H18N4O3S
N,2-dimethyl-6-[(2S)-4-methylsulfonylmorpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-(6-amino-2-methylpyrimidin-4-yl)morpholin-4-yl]-2-pyrazol-1-ylethanone —— C14H18N6O2
1-[(2R)-2-(6-amino-2-methylpyrimidin-4-yl)morpholin-4-yl]-2-pyrazol-1-ylethanone
—— 2-methyl-6-[(2S)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C14H20N6O
2-methyl-6-[(2S)-4-[(1-methylpyrazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N-(2-methoxyethyl)-2-methyl-6-[(2R)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine —— C17H25N5O3
N-(2-methoxyethyl)-2-methyl-6-[(2R)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-2-yl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2R)-4-[[2-(methylamino)pyridin-3-yl]methyl]morpholin-2-yl]pyrimidin-4-amine —— C17H24N6O
N,2-dimethyl-6-[(2R)-4-[[2-(methylamino)pyridin-3-yl]methyl]morpholin-2-yl]pyrimidin-4-amine
—— N,2-dimethyl-6-[(2R)-4-(1H-pyrazol-4-ylsulfonyl)morpholin-2-yl]pyrimidin-4-amine —— C13H18N6O3S
N,2-dimethyl-6-[(2R)-4-(1H-pyrazol-4-ylsulfonyl)morpholin-2-yl]pyrimidin-4-amine
—— 6-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]azetidin-2-yl]-N,2-dimethylpyrimidin-4-amine —— C14H19N5O3S
6-[(2S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]azetidin-2-yl]-N,2-dimethylpyrimidin-4-amine
—— [(2R)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]azetidin-1-yl]-(oxan-4-yl)methanone —— C15H22N4O2
[(2R)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]azetidin-1-yl]-(oxan-4-yl)methanone
—— 2-methyl-6-[(2R)-4-methylsulfonylmorpholin-2-yl]pyrimidin-4-amine —— C10H16N4O3S
2-methyl-6-[(2R)-4-methylsulfonylmorpholin-2-yl]pyrimidin-4-amine
—— 1-[(2S)-2-[6-(cyclopentylamino)-2-methylpyrimidin-4-yl]azetidin-1-yl]propan-1-one —— C16H24N4O
1-[(2S)-2-[6-(cyclopentylamino)-2-methylpyrimidin-4-yl]azetidin-1-yl]propan-1-one
—— 1-[(2R)-2-[2-methyl-6-[(4-methylthiadiazol-5-yl)methylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone —— C14H18N6OS
1-[(2R)-2-[2-methyl-6-[(4-methylthiadiazol-5-yl)methylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone
—— 2-methyl-6-[(2S)-4-methylsulfonylmorpholin-2-yl]pyrimidin-4-amine —— C10H16N4O3S
2-methyl-6-[(2S)-4-methylsulfonylmorpholin-2-yl]pyrimidin-4-amine
—— 1-[(2S)-2-[2-methyl-6-[2-[(R)-methylsulfinyl]ethylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone —— C13H20N4O2S
1-[(2S)-2-[2-methyl-6-[2-[(R)-methylsulfinyl]ethylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone
—— N,2-dimethyl-6-[(2R)-1-(1-methylpyrazol-4-yl)sulfonylazetidin-2-yl]pyrimidin-4-amine —— C13H18N6O2S
N,2-dimethyl-6-[(2R)-1-(1-methylpyrazol-4-yl)sulfonylazetidin-2-yl]pyrimidin-4-amine
—— N-(2-methoxyethyl)-2-methyl-6-[(2R)-4-(oxan-4-yl)morpholin-2-yl]pyrimidin-4-amine —— C17H28N4O3
N-(2-methoxyethyl)-2-methyl-6-[(2R)-4-(oxan-4-yl)morpholin-2-yl]pyrimidin-4-amine
—— 1-[(2R)-2-[2-methyl-6-[2-[(S)-methylsulfinyl]ethylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone —— C13H20N4O2S
1-[(2R)-2-[2-methyl-6-[2-[(S)-methylsulfinyl]ethylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone
—— [(2S)-2-(6-amino-2-methylpyrimidin-4-yl)azetidin-1-yl]-pyrazin-2-ylmethanone —— C13H14N6O
[(2S)-2-(6-amino-2-methylpyrimidin-4-yl)azetidin-1-yl]-pyrazin-2-ylmethanone
—— [(2R)-2-[6-(cyclopentylamino)-2-methylpyrimidin-4-yl]azetidin-1-yl]-pyrazin-2-ylmethanone —— C18H22N6O
[(2R)-2-[6-(cyclopentylamino)-2-methylpyrimidin-4-yl]azetidin-1-yl]-pyrazin-2-ylmethanone
—— 6-[(2R)-4-(1H-imidazol-5-ylmethyl)morpholin-2-yl]-N-(2-methoxyethyl)-2-methylpyrimidin-4-amine —— C16H24N6O2
6-[(2R)-4-(1H-imidazol-5-ylmethyl)morpholin-2-yl]-N-(2-methoxyethyl)-2-methylpyrimidin-4-amine
—— N,2-dimethyl-6-[(2S)-1-(1-methylimidazol-4-yl)sulfonylazetidin-2-yl]pyrimidin-4-amine —— C13H18N6O2S
N,2-dimethyl-6-[(2S)-1-(1-methylimidazol-4-yl)sulfonylazetidin-2-yl]pyrimidin-4-amine
—— N-cyclopentyl-2-methyl-6-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]azetidin-2-yl]pyrimidin-4-amine —— C18H26N6
N-cyclopentyl-2-methyl-6-[(2R)-1-[(1-methylpyrazol-4-yl)methyl]azetidin-2-yl]pyrimidin-4-amine
—— 6-[[(3S)-1-propan-2-ylpiperidin-3-yl]methyl]-N-(2-pyridin-4-ylethyl)pyridazin-3-amine —— C20H29N5
6-[[(3S)-1-propan-2-ylpiperidin-3-yl]methyl]-N-(2-pyridin-4-ylethyl)pyridazin-3-amine
—— N,2-dimethyl-6-[(2S)-1-methylsulfonylazetidin-2-yl]pyrimidin-4-amine —— C10H16N4O2S
N,2-dimethyl-6-[(2S)-1-methylsulfonylazetidin-2-yl]pyrimidin-4-amine
—— 6-[(2S)-1-cyclohexylazetidin-2-yl]-2-methylpyrimidin-4-amine —— C14H22N4
6-[(2S)-1-cyclohexylazetidin-2-yl]-2-methylpyrimidin-4-amine
—— N-cyclopentyl-6-[(2R)-1-(2-methoxyethyl)azetidin-2-yl]-2-methylpyrimidin-4-amine —— C16H26N4O
N-cyclopentyl-6-[(2R)-1-(2-methoxyethyl)azetidin-2-yl]-2-methylpyrimidin-4-amine
—— 6-[(2S)-1-(2-methoxyethyl)azetidin-2-yl]-2-methylpyrimidin-4-amine —— C11H18N4O
6-[(2S)-1-(2-methoxyethyl)azetidin-2-yl]-2-methylpyrimidin-4-amine
—— 6-[(2R)-1-cyclohexylazetidin-2-yl]-2-methylpyrimidin-4-amine —— C14H22N4
6-[(2R)-1-cyclohexylazetidin-2-yl]-2-methylpyrimidin-4-amine
—— 6-[(2R)-1-(2-methoxyethyl)azetidin-2-yl]-2-methylpyrimidin-4-amine —— C11H18N4O
6-[(2R)-1-(2-methoxyethyl)azetidin-2-yl]-2-methylpyrimidin-4-amine
—— 6-[[(3S)-1-(1H-pyrazol-4-ylsulfonyl)piperidin-3-yl]methyl]pyridazin-3-amine —— C13H18N6O2S
6-[[(3S)-1-(1H-pyrazol-4-ylsulfonyl)piperidin-3-yl]methyl]pyridazin-3-amine
—— [(2S)-2-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)azetidin-1-yl]-pyrazin-2-ylmethanone —— C17H20N6O
[(2S)-2-(2-methyl-6-pyrrolidin-1-ylpyrimidin-4-yl)azetidin-1-yl]-pyrazin-2-ylmethanone
—— 1-[(2R)-2-[2-methyl-6-[2-(5-methylpyrazol-1-yl)ethylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone —— C16H22N6O
1-[(2R)-2-[2-methyl-6-[2-(5-methylpyrazol-1-yl)ethylamino]pyrimidin-4-yl]azetidin-1-yl]ethanone
—— 1-[(2S)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]azetidin-1-yl]-2-pyrazol-1-ylethanone —— C14H18N6O
1-[(2S)-2-[2-methyl-6-(methylamino)pyrimidin-4-yl]azetidin-1-yl]-2-pyrazol-1-ylethanone
—— 2-methyl-6-[(2S)-1-(oxan-4-yl)azetidin-2-yl]pyrimidin-4-amine —— C13H20N4O
2-methyl-6-[(2S)-1-(oxan-4-yl)azetidin-2-yl]pyrimidin-4-amine