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—— 5-[(R)-(3-bromophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C16H17BrN4OS
5-[(R)-(3-bromophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-7-methyl-2-[2-(3-methylphenyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C23H26N2O2
(5R)-7-methyl-2-[2-(3-methylphenyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H26N4OS
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5-chlorofuran-2-yl)-[(3R)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone —— C15H22ClNO4
(5-chlorofuran-2-yl)-[(3R)-3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methanone
—— 5-[(R)-(2-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22ClN4OS+
5-[(R)-(2-chlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one —— C17H26N2OS
(5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one
—— 5-[(S)-(2-chlorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H22ClN5OS+2
5-[(S)-(2-chlorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-fluorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H24FN5O2S+2
5-[(S)-(2-fluorophenyl)-[4-(2-hydroxyethyl)piperazine-1,4-diium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-7-methyl-2-[2-(3-methylphenyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C23H26N2O2
(5S)-7-methyl-2-[2-(3-methylphenyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(S)-(2-chlorophenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C17H19ClN4OS
5-[(S)-(2-chlorophenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(2-chlorophenyl)-(1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H22ClN4O3S+
5-[(R)-(2-chlorophenyl)-(1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-N-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C16H21N3O3S
(5S)-N-[2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[(R)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H22ClN5O2S
5-[(R)-(2-chlorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5S)-5-[4-[1-[2-(dimethylamino)ethyl]imidazol-2-yl]piperidine-1-carbonyl]piperidin-2-one —— C18H29N5O2
(5S)-5-[4-[1-[2-(dimethylamino)ethyl]imidazol-2-yl]piperidine-1-carbonyl]piperidin-2-one
—— (5S)-7-ethyl-2-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O2
(5S)-7-ethyl-2-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(R)-(4-ethylpiperazin-1-ium-1-yl)-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H22FN5OS
5-[(R)-(4-ethylpiperazin-1-ium-1-yl)-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-(4-ethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O2S+
5-[(S)-(4-ethoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-difluorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C16H17F2N4O2S+
5-[(R)-(3,4-difluorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-2-(5-fluoro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H22FN3O2
(5S)-2-(5-fluoro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(S)-(4-ethoxy-3-methoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(S)-(4-ethoxy-3-methoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-ethoxycarbonylpiperidin-1-ium-1-yl)-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H23FN4O3S
5-[(S)-(4-ethoxycarbonylpiperidin-1-ium-1-yl)-(2-fluorophenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(3,4-dichlorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C16H17Cl2N4O2S+
5-[(R)-(3,4-dichlorophenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2-chlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C17H20ClN5OS
5-[(R)-(2-chlorophenyl)-(4-methylpiperazin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O2S+
5-[(S)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-dichlorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C16H17Cl2N4OS+
5-[(S)-(3,4-dichlorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-dichlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H20Cl2N4OS
5-[(R)-(3,4-dichlorophenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-2-(5-fluoro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H22FN3O2
(5R)-2-(5-fluoro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-isoquinolin-1-yl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C22H27N3O2
(5S)-2-isoquinolin-1-yl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(R)-(3,4-difluorophenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H20F2N4O2S
5-[(R)-(3,4-difluorophenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-chlorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C16H17ClN4OS
5-[(S)-(2-chlorophenyl)-pyrrolidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-7-ethyl-2-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O2
(5R)-7-ethyl-2-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(S)-(3,4-difluorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H22F2N4OS
5-[(S)-(3,4-difluorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(4-ethoxy-3-methoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H26N4O3S
5-[(R)-(4-ethoxy-3-methoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(2-fluorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H22FN5O2S
5-[(R)-(2-fluorophenyl)-[4-(2-hydroxyethyl)piperazin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(2-chlorophenyl)-[(2R,6S)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22ClN4O2S+
5-[(R)-(2-chlorophenyl)-[(2R,6S)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-difluorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H21F2N5OS+2
5-[(S)-(3,4-difluorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-chlorophenyl)-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H21ClN4O3S
5-[(S)-(2-chlorophenyl)-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-ethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O2S+
5-[(S)-(4-ethoxyphenyl)-piperidin-1-ium-1-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-5-[4-[1-[2-(dimethylamino)ethyl]imidazol-2-yl]piperidine-1-carbonyl]piperidin-2-one —— C18H29N5O2
(5R)-5-[4-[1-[2-(dimethylamino)ethyl]imidazol-2-yl]piperidine-1-carbonyl]piperidin-2-one
—— 5-[(R)-(3,4-dichlorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H21Cl2N5OS+2
5-[(R)-(3,4-dichlorophenyl)-(4-methylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(3,4-difluorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C18H20F2N4OS
5-[(S)-(3,4-difluorophenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— (5R)-5-methyl-N-[2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C15H19N3O3S
(5R)-5-methyl-N-[2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(2-methylsulfonylethyl)piperidin-2-one —— C17H23NO5S
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(2-methylsulfonylethyl)piperidin-2-one
—— 5-[(S)-(2-chlorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C19H23ClN4OS
5-[(S)-(2-chlorophenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate —— C20H24N4O3S
5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(3-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-olate
—— 5-[(R)-(2-chlorophenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C16H17ClN4O2S
5-[(R)-(2-chlorophenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(4-ethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O2S+
5-[(R)-(4-ethoxyphenyl)-(4-methylpiperidin-1-ium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O3S+
5-[(R)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(4-ethoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(3,4-difluorophenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H21F2N4O2S+
5-[(R)-(3,4-difluorophenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-2-[(4-chloro-5-methyl-1H-pyrazol-3-yl)methyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27ClN4O
(5S)-2-[(4-chloro-5-methyl-1H-pyrazol-3-yl)methyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one