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—— (5R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one —— C19H25N3O
(5R)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-7-(3-methoxypropyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2S
(5R)-7-(3-methoxypropyl)-2-thieno[3,2-d]pyrimidin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(morpholine-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one —— C19H26N2O3
(5S)-5-(morpholine-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
—— (5S)-7-(cyclopropylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O4S
(5S)-7-(cyclopropylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O4S
(5R)-7-(cyclopropylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclopentyl-2-[[2-(methoxymethyl)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5S)-7-cyclopentyl-2-[[2-(methoxymethyl)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(1-benzylpyrazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C22H28N4O2
(5R)-2-(1-benzylpyrazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one —— C17H18F3N3O2
(5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one
—— 5-[(2R)-2-methyl-4-phenylpiperazine-1-carbonyl]-2-thiophen-2-yl-1H-pyrimidin-6-one —— C20H20N4O2S
5-[(2R)-2-methyl-4-phenylpiperazine-1-carbonyl]-2-thiophen-2-yl-1H-pyrimidin-6-one
—— (5S)-7-(3-methoxypropyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3S
(5S)-7-(3-methoxypropyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(3-methoxypropyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3S
(5R)-7-(3-methoxypropyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-chlorophenyl)-N-[(S)-cyclopropyl-(2-methyl-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide —— C18H17ClN4O2
5-(2-chlorophenyl)-N-[(S)-cyclopropyl-(2-methyl-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide
—— (5S)-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O3
(5S)-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1R)-1-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C14H14N6OS
5-[(1R)-1-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— (5R)-2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C17H27N7O
(5R)-2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-ethyl-2-(4-phenylmethoxybutanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3
(5S)-7-ethyl-2-(4-phenylmethoxybutanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S)-2-methyl-4-phenylpiperazine-1-carbonyl]-2-thiophen-2-yl-1H-pyrimidin-6-one —— C20H20N4O2S
5-[(2S)-2-methyl-4-phenylpiperazine-1-carbonyl]-2-thiophen-2-yl-1H-pyrimidin-6-one
—— (5R)-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O3
(5R)-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O3
(5S)-2-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-(3-imidazol-1-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2
(5R)-7-(cyclopropylmethyl)-2-(3-imidazol-1-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-methyl-3-phenylpiperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione —— C16H19N3O4S
5-[(3S)-3-methyl-3-phenylpiperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione
—— 5-[(1S)-1-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C14H14N6OS
5-[(1S)-1-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— (5S)-7-(cyclopropylmethyl)-2-(3-imidazol-1-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2
(5S)-7-(cyclopropylmethyl)-2-(3-imidazol-1-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one —— C17H18F3N3O2
(5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[[3-(trifluoromethyl)phenyl]methyl]piperidin-2-one
—— (5S)-2-(1-benzylpyrazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C22H28N4O2
(5S)-2-(1-benzylpyrazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-aminopyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one —— C16H16Cl2N4O2
5-[(3R)-3-aminopyrrolidine-1-carbonyl]-2-[(2,6-dichlorophenyl)methyl]-1H-pyrimidin-6-one
—— (5S)-7-(3-methoxypropyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O3
(5S)-7-(3-methoxypropyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-N-(imidazo[1,2-a]pyrimidin-2-ylmethyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H18N4OS
(5S)-N-(imidazo[1,2-a]pyrimidin-2-ylmethyl)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— [5-[(2S)-oxolan-2-yl]thiophen-2-yl]-[4-(1,3-thiazol-2-yl)piperazin-1-yl]methanone —— C16H19N3O2S2
[5-[(2S)-oxolan-2-yl]thiophen-2-yl]-[4-(1,3-thiazol-2-yl)piperazin-1-yl]methanone
—— (5R)-7-ethyl-2-(4-phenylmethoxybutanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3
(5R)-7-ethyl-2-(4-phenylmethoxybutanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(methoxymethyl)thiophen-2-yl]-[(2S)-2-(2-pyrrolidin-1-ylethyl)piperidin-1-yl]methanone —— C18H28N2O2S
[5-(methoxymethyl)thiophen-2-yl]-[(2S)-2-(2-pyrrolidin-1-ylethyl)piperidin-1-yl]methanone
—— (5R)-7-(3-methoxypropyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O3
(5R)-7-(3-methoxypropyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-chlorophenyl)-N-[(R)-cyclopropyl-(2-methyl-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide —— C18H17ClN4O2
5-(2-chlorophenyl)-N-[(R)-cyclopropyl-(2-methyl-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide
—— (5R)-7-cyclopentyl-2-[[2-(methoxymethyl)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5R)-7-cyclopentyl-2-[[2-(methoxymethyl)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O3
(5R)-2-[2-(5-amino-3-methylpyrazol-1-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-methyl-3-phenylpiperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione —— C16H19N3O4S
5-[(3R)-3-methyl-3-phenylpiperidin-1-yl]sulfonyl-1H-pyrimidine-2,4-dione
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[1-(hydroxymethyl)cyclopropyl]methyl]-5-methylpiperidin-2-one —— C19H25NO4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[1-(hydroxymethyl)cyclopropyl]methyl]-5-methylpiperidin-2-one
—— (5S)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one —— C20H24N6O3
(5S)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one
—— (5S)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22FN3O3
(5S)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-2-[(2,5-dimethyl-1,2,4-triazol-3-yl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H27N5O
(5S)-2-[(2,5-dimethyl-1,2,4-triazol-3-yl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one —— C20H33N5O3
(5R)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one
—— (5R)-7-cyclohexyl-2-(3-pyrazol-1-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5R)-7-cyclohexyl-2-(3-pyrazol-1-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one —— C19H22FN3O3
(5R)-9-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,9-diazaspiro[4.6]undecan-2-one
—— (5S)-2-(2-methylsulfanylacetyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H26N2O3S
(5S)-2-(2-methylsulfanylacetyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one —— C20H33N5O3
(5S)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one
—— (5S)-2-(2-methyl-1,3-benzothiazole-6-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N3O2S
(5S)-2-(2-methyl-1,3-benzothiazole-6-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-3-fluoro-2-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine —— C19H19ClFN5
5-chloro-3-fluoro-2-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine
—— (5R)-9-[2-(5-methylfuran-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H21NO3
(5R)-9-[2-(5-methylfuran-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[1-(hydroxymethyl)cyclopropyl]methyl]-5-methylpiperidin-2-one —— C19H25NO4
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[1-(hydroxymethyl)cyclopropyl]methyl]-5-methylpiperidin-2-one
—— (5R)-2-(2-methylsulfanylacetyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H26N2O3S
(5R)-2-(2-methylsulfanylacetyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one