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—— (5-bromopyridin-3-yl)methyl (1R,2R)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate —— C17H13BrF3NO2
(5-bromopyridin-3-yl)methyl (1R,2R)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate
—— (5S)-1-(2,5-dimethoxyphenyl)-5-(2-piperidin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H26N4O4S
(5S)-1-(2,5-dimethoxyphenyl)-5-(2-piperidin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R,7R)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H23F3N4O2
(5R,7R)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S)-5-(2-morpholin-4-ylethyliminomethyl)-1-(4-propan-2-ylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H26N4O3S
(5S)-5-(2-morpholin-4-ylethyliminomethyl)-1-(4-propan-2-ylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[(3aS,7aS)-2,3,3a,4,5,6,7,7a-octahydroindol-1-yl]-4-chloro-2-methylpyridazin-3-one —— C13H18ClN3O
5-[(3aS,7aS)-2,3,3a,4,5,6,7,7a-octahydroindol-1-yl]-4-chloro-2-methylpyridazin-3-one
—— (5S)-5-(2-piperidin-1-ylethyliminomethyl)-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C15H22N4O2S
(5S)-5-(2-piperidin-1-ylethyliminomethyl)-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S,7S)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C20H23F3N4O2
(5S,7S)-5-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S)-1-(3-methoxyphenyl)-5-(2-morpholin-4-ium-4-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H23N4O4S+
(5S)-1-(3-methoxyphenyl)-5-(2-morpholin-4-ium-4-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-1-phenyl-5-(2-piperazin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H21N5O2S
(5S)-1-phenyl-5-(2-piperazin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5-bromopyridin-3-yl)methyl (1R,2S)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate —— C17H13BrF3NO2
(5-bromopyridin-3-yl)methyl (1R,2S)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate
—— [(5S,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-morpholin-4-ylmethanone —— C19H21F3N4O3
[(5S,7R)-5-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-morpholin-4-ylmethanone
—— (5R)-1-cyclohexyl-5-(2-morpholin-4-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H26N4O3S
(5R)-1-cyclohexyl-5-(2-morpholin-4-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[3-(Dimethylamino)propyliminomethyl]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C13H20N4O2S
5-[3-(Dimethylamino)propyliminomethyl]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-1-hexyl-4-[hydroxy(phenyl)methylidene]-5-(3-nitrophenyl)pyrrolidine-2,3-dione —— C23H24N2O5
(5S)-1-hexyl-4-[hydroxy(phenyl)methylidene]-5-(3-nitrophenyl)pyrrolidine-2,3-dione
—— (5S)-1-phenyl-5-(2-piperazine-1,4-diium-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H23N5O2S+2
(5S)-1-phenyl-5-(2-piperazine-1,4-diium-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-5-[2-(dimethylamino)ethyliminomethyl]-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C10H16N4O2S
(5R)-5-[2-(dimethylamino)ethyliminomethyl]-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R,7R)-5-phenyl-N-[(1S)-1-phenylethyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H21F3N4O
(5R,7R)-5-phenyl-N-[(1S)-1-phenylethyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5-bromopyridin-3-yl)methyl (1S,2S)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate —— C17H13BrF3NO2
(5-bromopyridin-3-yl)methyl (1S,2S)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate
—— (5-bromopyridin-3-yl)methyl (1S,2R)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate —— C17H13BrF3NO2
(5-bromopyridin-3-yl)methyl (1S,2R)-2-[2-(trifluoromethyl)phenyl]cyclopropane-1-carboxylate
—— (5R)-1-(2-chlorophenyl)-5-(2-morpholin-4-ium-4-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H20ClN4O3S+
(5R)-1-(2-chlorophenyl)-5-(2-morpholin-4-ium-4-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[2-(Diethylamino)ethyliminomethyl]-1-(4-propan-2-ylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H28N4O2S
5-[2-(Diethylamino)ethyliminomethyl]-1-(4-propan-2-ylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S,7R)-3-bromo-N-[(2-pyrazol-1-ylpyridin-4-yl)methyl]adamantane-1-carboxamide —— C20H23BrN4O
(5S,7R)-3-bromo-N-[(2-pyrazol-1-ylpyridin-4-yl)methyl]adamantane-1-carboxamide
—— (5R,10bS)-1',5'-dimethyl-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one —— C25H21N3O2
(5R,10bS)-1',5'-dimethyl-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one
—— (5R,10bS)-2-naphthalen-1-yl-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H20N2O
(5R,10bS)-2-naphthalen-1-yl-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-1-(4-fluorophenyl)-5-(2-piperidin-1-ium-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H22FN4O2S+
(5R)-1-(4-fluorophenyl)-5-(2-piperidin-1-ium-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S,10bS)-5-(4-tert-butylphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H28N2O2
(5S,10bS)-5-(4-tert-butylphenyl)-2-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,7R)-3-chloro-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cycloheptyl]adamantane-1-carboxamide —— C21H30ClN3O2
(5S,7R)-3-chloro-N-[1-(5-methyl-1,2,4-oxadiazol-3-yl)cycloheptyl]adamantane-1-carboxamide
—— 5-(2-Piperazin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C11H17N5O2S
5-(2-Piperazin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S,10bS)-2-naphthalen-2-yl-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C26H20N2O
(5S,10bS)-2-naphthalen-2-yl-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(9aR)-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-4-chloro-2-methylpyridazin-3-one —— C13H19ClN4O
5-[(9aR)-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepin-2-yl]-4-chloro-2-methylpyridazin-3-one
—— (5R)-1-(2,5-dimethoxyphenyl)-5-(3-imidazol-1-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H21N5O4S
(5R)-1-(2,5-dimethoxyphenyl)-5-(3-imidazol-1-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-3-(2,4-dichlorophenyl)-N-(5-methyl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C13H11Cl2N5O2
(5R)-3-(2,4-dichlorophenyl)-N-(5-methyl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R,10bS)-2-(4-methoxyphenyl)-1'-methylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one —— C25H21N3O3
(5R,10bS)-2-(4-methoxyphenyl)-1'-methylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one
—— (5S)-1-(2-methoxyphenyl)-5-(2-piperidin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H24N4O3S
(5S)-1-(2-methoxyphenyl)-5-(2-piperidin-1-ylethyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R,10bS)-5-(4-butoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C27H28N2O2
(5R,10bS)-5-(4-butoxyphenyl)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(1-Benzylpiperidin-4-yl)iminomethyl]-1-phenyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C23H24N4O2S
5-[(1-Benzylpiperidin-4-yl)iminomethyl]-1-phenyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[(3aR,7aS)-2,3,3a,4,5,6,7,7a-octahydroindol-1-yl]-4-chloro-2-methylpyridazin-3-one —— C13H18ClN3O
5-[(3aR,7aS)-2,3,3a,4,5,6,7,7a-octahydroindol-1-yl]-4-chloro-2-methylpyridazin-3-one
—— (5S)-3-(2,4-dichlorophenyl)-N-(5-methyl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C13H11Cl2N5O2
(5S)-3-(2,4-dichlorophenyl)-N-(5-methyl-1H-1,2,4-triazol-3-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5Z)-5-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C20H19ClN2O3S
(5Z)-5-[[5-(2-chlorophenyl)furan-2-yl]methylidene]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— 5-[5-(Diethylsulfamoyl)-2-methoxyanilino]-5-oxopentanoate —— C16H23N2O6S-
5-[5-(Diethylsulfamoyl)-2-methoxyanilino]-5-oxopentanoate
—— 5-amino-1-[(6R)-6-methyl-2-propylsulfanyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]pyrazole-4-carbonitrile —— C18H20N6S2
5-amino-1-[(6R)-6-methyl-2-propylsulfanyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]pyrazole-4-carbonitrile
—— (5Z)-5-[[(1R)-cyclohex-3-en-1-yl]methylidene]-3-[(3R)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C14H17NO3S3
(5Z)-5-[[(1R)-cyclohex-3-en-1-yl]methylidene]-3-[(3R)-1,1-dioxothiolan-3-yl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R,7R)-N-[(4-fluorophenyl)methyl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H16F4N4O2
(5R,7R)-N-[(4-fluorophenyl)methyl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-bromo-2-[[(2R)-2-(3-chlorophenoxy)propanoyl]amino]benzoate —— C16H12BrClNO4-
5-bromo-2-[[(2R)-2-(3-chlorophenoxy)propanoyl]amino]benzoate
—— [(5S)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone —— C20H25ClN2O2
[(5S)-3-(4-chlorophenyl)-4,5-dihydro-1,2-oxazol-5-yl]-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]methanone
—— 5-chloro-4-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]amino]-1H-pyridazin-6-one —— C14H14ClN3O3
5-chloro-4-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]amino]-1H-pyridazin-6-one
—— 5-[(1R)-1-[2-(3,4-dimethoxyphenyl)ethylamino]ethyl]-1,3-dihydrobenzimidazol-2-one —— C19H23N3O3
5-[(1R)-1-[2-(3,4-dimethoxyphenyl)ethylamino]ethyl]-1,3-dihydrobenzimidazol-2-one
—— 5-[(1S)-1-[2-(3,4-dimethoxyphenyl)ethylamino]ethyl]-1,3-dihydrobenzimidazol-2-one —— C19H23N3O3
5-[(1S)-1-[2-(3,4-dimethoxyphenyl)ethylamino]ethyl]-1,3-dihydrobenzimidazol-2-one
—— (5S)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(5-methyl-1,2-oxazol-3-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H16ClN3O5
(5S)-3-(5-chloro-2,4-dimethoxyphenyl)-N-(5-methyl-1,2-oxazol-3-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(4-butylphenyl)sulfamoyl]-N-[(2S)-1-hydroxypropan-2-yl]-2-methylbenzamide —— C21H28N2O4S
5-[(4-butylphenyl)sulfamoyl]-N-[(2S)-1-hydroxypropan-2-yl]-2-methylbenzamide