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—— 5-chloro-N-[(3R)-1-(2-methoxyethyl)piperidin-3-yl]pyridin-2-amine —— C13H20ClN3O
5-chloro-N-[(3R)-1-(2-methoxyethyl)piperidin-3-yl]pyridin-2-amine
—— (5R)-5-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1-benzylpiperidin-2-one —— C19H24N2O2
(5R)-5-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1-benzylpiperidin-2-one
—— 5-chloro-6-[[(1S)-1-cyclohexyl-3-hydroxypropyl]amino]-N,N-dimethylpyridine-3-carboxamide —— C17H26ClN3O2
5-chloro-6-[[(1S)-1-cyclohexyl-3-hydroxypropyl]amino]-N,N-dimethylpyridine-3-carboxamide
—— (5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (E)-3-thiophen-3-ylprop-2-enoate —— C14H10N2O3S2
(5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl (E)-3-thiophen-3-ylprop-2-enoate
—— (5R)-5-methyl-2-[4-[2-(1,2,4-triazol-1-yl)ethyl]piperazin-1-yl]-4,5-dihydro-1,3-thiazole —— C12H20N6S
(5R)-5-methyl-2-[4-[2-(1,2,4-triazol-1-yl)ethyl]piperazin-1-yl]-4,5-dihydro-1,3-thiazole
—— 5-[(3aS,7aR)-1,3,3a,4,5,6,7,7a-octahydroisoindol-2-yl]-4-chloro-2-methylpyridazin-3-one —— C13H18ClN3O
5-[(3aS,7aR)-1,3,3a,4,5,6,7,7a-octahydroisoindol-2-yl]-4-chloro-2-methylpyridazin-3-one
—— 5-fluoro-2-hydroxy-N-[(3S)-3-(2-oxopyrrolidin-1-yl)pentyl]benzamide —— C16H21FN2O3
5-fluoro-2-hydroxy-N-[(3S)-3-(2-oxopyrrolidin-1-yl)pentyl]benzamide
—— 5-Tert-butyl-2-[(4-methoxy-2-nitrophenoxy)methyl]-1,3-dimethylbenzene —— C20H25NO4
5-Tert-butyl-2-[(4-methoxy-2-nitrophenoxy)methyl]-1,3-dimethylbenzene
—— (5S)-4-[hydroxy-(4-propan-2-yloxyphenyl)methylidene]-1-(2-methoxyethyl)-5-(2-methoxyphenyl)pyrrolidine-2,3-dione —— C24H27NO6
(5S)-4-[hydroxy-(4-propan-2-yloxyphenyl)methylidene]-1-(2-methoxyethyl)-5-(2-methoxyphenyl)pyrrolidine-2,3-dione
—— 5-chloro-N-[(3S)-1-(4-ethoxyphenyl)-5-oxopyrrolidin-3-yl]-2-methoxybenzamide —— C20H21ClN2O4
5-chloro-N-[(3S)-1-(4-ethoxyphenyl)-5-oxopyrrolidin-3-yl]-2-methoxybenzamide
—— (5-chloropyrimidin-4-yl)-[(1R,5S)-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-3-yl]methanone —— C12H14ClN3O
(5-chloropyrimidin-4-yl)-[(1R,5S)-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-3-yl]methanone
—— (5-methylpyrazin-2-yl)-[(3S)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone —— C19H23N3O2
(5-methylpyrazin-2-yl)-[(3S)-3-(3-phenylpropoxy)pyrrolidin-1-yl]methanone
—— (5S,6R)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H15N3O2S2
(5S,6R)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— 5-chloro-N-[(1R)-2-(diethylamino)-2-oxo-1-phenylethyl]pyrimidine-4-carboxamide —— C17H19ClN4O2
5-chloro-N-[(1R)-2-(diethylamino)-2-oxo-1-phenylethyl]pyrimidine-4-carboxamide
—— (5R,6R)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H15N3O2S2
(5R,6R)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S,6S)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H15N3O2S2
(5S,6S)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5R,6S)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H15N3O2S2
(5R,6S)-1-methyl-6-thiophen-2-yl-5-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— 5-[(2S)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]thiophene-3-carbonitrile —— C16H19N3OS
5-[(2S)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]thiophene-3-carbonitrile
—— 5-chloro-N-[(1S)-2-(diethylamino)-2-oxo-1-phenylethyl]pyrimidine-4-carboxamide —— C17H19ClN4O2
5-chloro-N-[(1S)-2-(diethylamino)-2-oxo-1-phenylethyl]pyrimidine-4-carboxamide
—— 5-(3-chloro-4-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide —— C11H9ClFN3O
5-(3-chloro-4-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
—— 5-[(2R)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]thiophene-3-carbonitrile —— C16H19N3OS
5-[(2R)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]thiophene-3-carbonitrile
—— 5-[3-[(2R)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]propyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C18H23N5OS
5-[3-[(2R)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]propyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-[(2R)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]furan-2-carbonitrile —— C16H19N3O2
5-[(2R)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]furan-2-carbonitrile
—— [5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2S)-2-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)piperidin-1-yl]methanone —— C23H25FN4O3
[5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2S)-2-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)piperidin-1-yl]methanone
—— 5-[(2S)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]furan-2-carbonitrile —— C16H19N3O2
5-[(2S)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]furan-2-carbonitrile
—— 5-[3-[(2S)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]propyl]-3-thiophen-2-yl-1,2,4-oxadiazole —— C18H23N5OS
5-[3-[(2S)-2-[(2-methylimidazol-1-yl)methyl]pyrrolidin-1-yl]propyl]-3-thiophen-2-yl-1,2,4-oxadiazole
—— 5-chloro-N-[[(2R)-5-oxopyrrolidin-2-yl]methyl]-2-propoxybenzamide —— C15H19ClN2O3
5-chloro-N-[[(2R)-5-oxopyrrolidin-2-yl]methyl]-2-propoxybenzamide
—— [5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2R)-2-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)piperidin-1-yl]methanone —— C23H25FN4O3
[5-[(4-fluorophenoxy)methyl]furan-2-yl]-[(2R)-2-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)piperidin-1-yl]methanone
—— 5-methyl-N-[4-methyl-3-[(3S)-oxolan-3-yl]oxyphenyl]-1,2-oxazole-3-carboxamide —— C16H18N2O4
5-methyl-N-[4-methyl-3-[(3S)-oxolan-3-yl]oxyphenyl]-1,2-oxazole-3-carboxamide
—— 5-[4-[(1S)-1-phenylpropyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide —— C19H24N4O2
5-[4-[(1S)-1-phenylpropyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide
—— 5-methyl-N-[4-methyl-3-[(3R)-oxolan-3-yl]oxyphenyl]-1,2-oxazole-3-carboxamide —— C16H18N2O4
5-methyl-N-[4-methyl-3-[(3R)-oxolan-3-yl]oxyphenyl]-1,2-oxazole-3-carboxamide
—— 5-[(1R)-1-propyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1H-pyrrole-3-carboxamide —— C18H21N3O2
5-[(1R)-1-propyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1H-pyrrole-3-carboxamide
—— 5-[4-[(1R)-1-phenylpropyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide —— C19H24N4O2
5-[4-[(1R)-1-phenylpropyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide
—— (5S)-5-methyl-2-[4-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperazin-1-yl]-4,5-dihydro-1,3-thiazole —— C14H19N7S
(5S)-5-methyl-2-[4-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperazin-1-yl]-4,5-dihydro-1,3-thiazole
—— 5-chloro-N-[[(2S)-5-oxopyrrolidin-2-yl]methyl]-2-propoxybenzamide —— C15H19ClN2O3
5-chloro-N-[[(2S)-5-oxopyrrolidin-2-yl]methyl]-2-propoxybenzamide
—— 5-[4-[(1R)-1-(2-fluorophenyl)ethyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide —— C18H21FN4O2
5-[4-[(1R)-1-(2-fluorophenyl)ethyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide
—— 5-nitro-2-[[(2R)-1-piperidin-1-ylpropan-2-yl]amino]benzamide —— C15H22N4O3
5-nitro-2-[[(2R)-1-piperidin-1-ylpropan-2-yl]amino]benzamide
—— 5-fluoro-2-[[(3S)-oxolan-3-yl]methyl]isoindole-1,3-dione —— C13H12FNO3
5-fluoro-2-[[(3S)-oxolan-3-yl]methyl]isoindole-1,3-dione
—— 5-bromo-N-methyl-N-[[4-[(R)-methylsulfinyl]phenyl]methyl]pyridin-3-amine —— C14H15BrN2OS
5-bromo-N-methyl-N-[[4-[(R)-methylsulfinyl]phenyl]methyl]pyridin-3-amine
—— 5-[(1S)-1-propyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1H-pyrrole-3-carboxamide —— C18H21N3O2
5-[(1S)-1-propyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1H-pyrrole-3-carboxamide
—— 5-[4-[(1S)-1-(2-fluorophenyl)ethyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide —— C18H21FN4O2
5-[4-[(1S)-1-(2-fluorophenyl)ethyl]piperazine-1-carbonyl]-1H-pyrrole-3-carboxamide
—— 5-bromo-N-methyl-N-[[4-[(S)-methylsulfinyl]phenyl]methyl]pyridin-3-amine —— C14H15BrN2OS
5-bromo-N-methyl-N-[[4-[(S)-methylsulfinyl]phenyl]methyl]pyridin-3-amine
—— 5-nitro-2-[[(2S)-1-piperidin-1-ylpropan-2-yl]amino]benzamide —— C15H22N4O3
5-nitro-2-[[(2S)-1-piperidin-1-ylpropan-2-yl]amino]benzamide
—— 5-[[2-[amino(butylsulfanyl)methylidene]hydrazinyl]methylidene]-6-oxocyclohexa-1,3-diene-1-carboxylate —— C13H16N3O3S-
5-[[2-[amino(butylsulfanyl)methylidene]hydrazinyl]methylidene]-6-oxocyclohexa-1,3-diene-1-carboxylate
—— (5R)-5-methyl-2-[4-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperazin-1-yl]-4,5-dihydro-1,3-thiazole —— C14H19N7S
(5R)-5-methyl-2-[4-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperazin-1-yl]-4,5-dihydro-1,3-thiazole
—— (5E)-5-(2H-chromen-3-ylmethylidene)-2-[(E)-2-(4-methylphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C23H17N3O2S
(5E)-5-(2H-chromen-3-ylmethylidene)-2-[(E)-2-(4-methylphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— 5-chloro-N-cyclopentyl-6-[[(2S)-1-hydroxypropan-2-yl]amino]pyridine-3-carboxamide —— C14H20ClN3O2
5-chloro-N-cyclopentyl-6-[[(2S)-1-hydroxypropan-2-yl]amino]pyridine-3-carboxamide
—— 5-(Cyclohexylmethyl)-1-phenylpyrazolo[3,4-d]pyrimidin-4-one —— C18H20N4O
5-(Cyclohexylmethyl)-1-phenylpyrazolo[3,4-d]pyrimidin-4-one
—— 5-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylquinoline —— C15H18N2O3S
5-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylquinoline
—— 5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylquinoline —— C15H18N2O3S
5-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonylquinoline