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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-7-ethyl-2-(5-ethyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5R)-7-ethyl-2-(5-ethyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O3S
(5R)-2-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O2
(5R)-7-(cyclobutylmethyl)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-2-methyl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine —— C21H26N6
5-ethyl-2-methyl-4-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine
—— (5S)-5-methyl-5-(4-methylpent-3-enyl)-1-(pyridin-4-ylmethyl)piperidin-2-one —— C18H26N2O
(5S)-5-methyl-5-(4-methylpent-3-enyl)-1-(pyridin-4-ylmethyl)piperidin-2-one
—— (5S)-7-(cyclobutylmethyl)-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H33N3O3
(5S)-7-(cyclobutylmethyl)-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-2-methyl-4-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine —— C21H26N6
5-ethyl-2-methyl-4-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidine
—— (5R)-2-[2-(2-ethoxyphenyl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O4
(5R)-2-[2-(2-ethoxyphenyl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-2-(2-phenylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C20H21N3O2S
5-[(2R)-2-(2-phenylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (5R)-5-methyl-1-[(3-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one —— C19H22N2O
(5R)-5-methyl-1-[(3-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one
—— (5S)-2-[2-(2-ethoxyphenyl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O4
(5S)-2-[2-(2-ethoxyphenyl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O2
(5S)-7-(cyclobutylmethyl)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-cyclopropyl-N-[(3R)-3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1,3,4-oxadiazol-2-amine —— C18H18FN3O2
5-cyclopropyl-N-[(3R)-3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1,3,4-oxadiazol-2-amine
—— (5S)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H27N3O4S
(5S)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-chlorothiophen-2-yl)-[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C17H25ClN2O3S
(5-chlorothiophen-2-yl)-[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— (5R)-7-(cyclobutylmethyl)-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H33N3O3
(5R)-7-(cyclobutylmethyl)-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-methyl-1-[(3-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one —— C19H22N2O
(5S)-5-methyl-1-[(3-methylpyridin-4-yl)methyl]-5-phenylpiperidin-2-one
—— (5S)-2-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H25N3O3S
(5S)-2-[2-(2,4-dimethyl-1,3-thiazol-5-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1S)-1-[4-[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]triazol-1-yl]ethyl]-2H-tetrazole —— C16H16FN9
5-[(1S)-1-[4-[2-(3,5-dimethylpyrazol-1-yl)-5-fluorophenyl]triazol-1-yl]ethyl]-2H-tetrazole
—— (5R)-2-(3-chloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H22ClN3O2
(5R)-2-(3-chloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-chlorothiophen-2-yl)-[(4S)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C17H25ClN2O3S
(5-chlorothiophen-2-yl)-[(4S)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— 5-[(2S)-2-(2-phenylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C20H21N3O2S
5-[(2S)-2-(2-phenylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— 5-cyclopropyl-N-[(3S)-3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1,3,4-oxadiazol-2-amine —— C18H18FN3O2
5-cyclopropyl-N-[(3S)-3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1,3,4-oxadiazol-2-amine
—— 5-[4-[(3S)-oxolan-3-yl]triazol-1-yl]pentan-1-ol —— C11H19N3O2
5-[4-[(3S)-oxolan-3-yl]triazol-1-yl]pentan-1-ol
—— 5-cyclopropyl-N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide —— C22H25N5O
5-cyclopropyl-N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide
—— 5-[(2R)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide —— C17H17N5O2S
5-[(2R)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide
—— (5S)-2-[2-(1-methylpyrazol-4-yl)ethyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C17H28N4O
(5S)-2-[2-(1-methylpyrazol-4-yl)ethyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O3S
(5S)-7-(2-hydroxyethyl)-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-[4-(1H-pyrazol-4-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H32N4O2
(5R)-7-cyclohexyl-2-[4-(1H-pyrazol-4-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-methyl-1-[(4-methylpyridin-2-yl)methyl]-5-phenylpiperidin-2-one —— C19H22N2O
(5R)-5-methyl-1-[(4-methylpyridin-2-yl)methyl]-5-phenylpiperidin-2-one
—— 5-(imidazol-1-ylmethyl)-N-methyl-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]furan-2-carboxamide —— C21H24N4O2
5-(imidazol-1-ylmethyl)-N-methyl-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]furan-2-carboxamide
—— 5-(imidazol-1-ylmethyl)-N-methyl-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]furan-2-carboxamide —— C21H24N4O2
5-(imidazol-1-ylmethyl)-N-methyl-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]furan-2-carboxamide
—— (5R)-2-(furan-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N2O4
(5R)-2-(furan-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(3-methoxyphenyl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H26N2O4S
(5S)-2-(3-methoxyphenyl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(2,5-dimethyl-1,3-oxazol-4-yl)methyl]-5-methylpiperidin-2-one —— C20H24N2O4
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(2,5-dimethyl-1,3-oxazol-4-yl)methyl]-5-methylpiperidin-2-one
—— 5-[4-[(3R)-oxolan-3-yl]triazol-1-yl]pentan-1-ol —— C11H19N3O2
5-[4-[(3R)-oxolan-3-yl]triazol-1-yl]pentan-1-ol
—— 5-acetyl-N-[[(3R)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]thiophene-2-carboxamide —— C18H19NO4S
5-acetyl-N-[[(3R)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]thiophene-2-carboxamide
—— (5S)-7-ethyl-2-(5-ethyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5S)-7-ethyl-2-(5-ethyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2S
(5S)-7-(cyclobutylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(furan-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N2O4
(5S)-2-(furan-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(3-methoxyphenyl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H26N2O4S
(5R)-2-(3-methoxyphenyl)sulfonyl-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclopentyl-2-[3-(tetrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H28N6O
(5S)-7-cyclopentyl-2-[3-(tetrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-methyl-1-[(4-methylpyridin-2-yl)methyl]-5-phenylpiperidin-2-one —— C19H22N2O
(5S)-5-methyl-1-[(4-methylpyridin-2-yl)methyl]-5-phenylpiperidin-2-one
—— (5S)-7-cyclohexyl-2-[4-(1H-pyrazol-4-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H32N4O2
(5S)-7-cyclohexyl-2-[4-(1H-pyrazol-4-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O2
(5R)-7-cyclohexyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-[(2S)-oxolan-2-yl]thiophen-2-yl]-[4-(thian-4-yl)piperazin-1-yl]methanone —— C18H26N2O2S2
[5-[(2S)-oxolan-2-yl]thiophen-2-yl]-[4-(thian-4-yl)piperazin-1-yl]methanone
—— (5R)-7-(cyclobutylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2S
(5R)-7-(cyclobutylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(2,5-dimethyl-1,3-oxazol-4-yl)methyl]-5-methylpiperidin-2-one —— C20H24N2O4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(2,5-dimethyl-1,3-oxazol-4-yl)methyl]-5-methylpiperidin-2-one
—— (5R)-7-cyclopentyl-2-[3-(tetrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H28N6O
(5R)-7-cyclopentyl-2-[3-(tetrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-[(4-propan-2-ylthiadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H30N4OS
(5S)-7-(cyclobutylmethyl)-2-[(4-propan-2-ylthiadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one