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—— 5-ethyl-4-[(3S)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-2,6-dimethylpyrimidine —— C19H29N5O
5-ethyl-4-[(3S)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidin-1-yl]-2,6-dimethylpyrimidine
—— (5S)-7-(2-methoxyethyl)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H25N3O3
(5S)-7-(2-methoxyethyl)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[1-(hydroxymethyl)cyclobutyl]methyl]-5-methylpiperidin-2-one —— C20H27NO4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[1-(hydroxymethyl)cyclobutyl]methyl]-5-methylpiperidin-2-one
—— (5R,6R)-5-(4-methoxyphenyl)-3-oxo-2-[(1S)-1,2,3,4-tetrahydroisoquinolin-2-ium-1-yl]-6-(1,2,4-triazol-1-yl)cyclohexen-1-olate —— C24H24N4O3
(5R,6R)-5-(4-methoxyphenyl)-3-oxo-2-[(1S)-1,2,3,4-tetrahydroisoquinolin-2-ium-1-yl]-6-(1,2,4-triazol-1-yl)cyclohexen-1-olate
—— (5S)-N-(3-chloro-4-fluorophenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide —— C18H23ClFN3O2
(5S)-N-(3-chloro-4-fluorophenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-(3-methoxy-2,2-dimethylpropyl)-5-methylpiperidin-2-one —— C20H29NO4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-(3-methoxy-2,2-dimethylpropyl)-5-methylpiperidin-2-one
—— (5S)-2-[2-(2-methylimidazol-1-yl)ethyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C17H28N4O
(5S)-2-[2-(2-methylimidazol-1-yl)ethyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-(2-morpholin-4-ylethyl)-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H26N4O3
(5R)-1-(2-morpholin-4-ylethyl)-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— 5-[(4R)-2,2-dimethyloxan-4-yl]-3-(2-methoxyethyl)-1-methyl-1,2,4-triazole —— C13H23N3O2
5-[(4R)-2,2-dimethyloxan-4-yl]-3-(2-methoxyethyl)-1-methyl-1,2,4-triazole
—— (5R)-7-(2-methoxyethyl)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H25N3O3
(5R)-7-(2-methoxyethyl)-2-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1S)-1-(1,3-benzodioxol-5-yloxy)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C15H12N4O4
5-[(1S)-1-(1,3-benzodioxol-5-yloxy)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— 5-[(3R)-3-(4-phenylbenzoyl)piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C22H21N3O3
5-[(3R)-3-(4-phenylbenzoyl)piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— 5-[(2R)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C18H19N3O2S2
5-[(2R)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(3-methoxypropyl)-5-phenylpyrrolidine-2,3-dione —— C24H25NO5
(5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(3-methoxypropyl)-5-phenylpyrrolidine-2,3-dione
—— (5R)-N-(3-chloro-4-fluorophenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide —— C18H23ClFN3O2
(5R)-N-(3-chloro-4-fluorophenyl)-6-oxo-7-propan-2-yl-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-7-(cyclopropylmethyl)-2-[[6-(dimethylamino)pyridin-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O
(5S)-7-(cyclopropylmethyl)-2-[[6-(dimethylamino)pyridin-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-ethyl-5-(4-pyrimidin-2-ylpiperazine-1-carbonyl)piperidin-2-one —— C16H23N5O2
(5R)-1-ethyl-5-(4-pyrimidin-2-ylpiperazine-1-carbonyl)piperidin-2-one
—— (5R,7R)-N-(1-adamantyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H25F3N4OS
(5R,7R)-N-(1-adamantyl)-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R)-9-(2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C13H15N5O3
(5R)-9-(2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl)-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C18H19N3O2S2
5-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (5R)-4-(5-chloro-1,3-dimethylpyrazol-4-yl)sulfonyl-5-methyl-1-phenylpiperazin-2-one —— C16H19ClN4O3S
(5R)-4-(5-chloro-1,3-dimethylpyrazol-4-yl)sulfonyl-5-methyl-1-phenylpiperazin-2-one
—— (5S)-1-(2-morpholin-4-ylethyl)-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H26N4O3
(5S)-1-(2-morpholin-4-ylethyl)-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-(3-methoxy-2,2-dimethylpropyl)-5-methylpiperidin-2-one —— C20H29NO4
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-(3-methoxy-2,2-dimethylpropyl)-5-methylpiperidin-2-one
—— (5R)-9-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C14H23N3O3S
(5R)-9-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-7-(2-hydroxyethyl)-2-(3-phenyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H23N3O4
(5R)-7-(2-hydroxyethyl)-2-(3-phenyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H23N3O3
(5S)-7-(cyclopropylmethyl)-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-(4-phenylbenzoyl)piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one —— C22H21N3O3
5-[(3S)-3-(4-phenylbenzoyl)piperidine-1-carbonyl]-1,2-dihydropyrazol-3-one
—— (5R)-7-(cyclopropylmethyl)-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H23N3O3
(5R)-7-(cyclopropylmethyl)-2-(6-oxo-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(3S)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C19H22N6O2
[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(3S)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— [5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C19H22N6O2
[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— (5S)-2-(2,4-dimethyl-6-oxo-1H-pyridine-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O3
(5S)-2-(2,4-dimethyl-6-oxo-1H-pyridine-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C14H23N3O3S
(5S)-9-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-2-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O2S2
(5R)-2-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-(3-phenyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H23N3O4
(5S)-7-(2-hydroxyethyl)-2-(3-phenyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)-5-(3-methoxyphenyl)pyrrolidine-2,3-dione —— C24H25NO6
(5R)-4-[hydroxy-[(2R)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)-5-(3-methoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-2-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O2S2
(5S)-2-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione —— C29H27NO6
(5S)-4-[hydroxy-[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methylidene]-1-(2-methoxyethyl)-5-(3-phenoxyphenyl)pyrrolidine-2,3-dione
—— 5-[(5R)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile —— C21H28N4O2
5-[(5R)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile
—— 5-[(5S)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile —— C21H28N4O2
5-[(5S)-7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile
—— (5E)-3-ethyl-2-(3-methyl-5-oxo-1-phenylpyrazol-4-ylidene)-5-(1,3,3-trimethylindol-2-ylidene)-1,3-thiazolidin-4-one —— C26H26N4O2S
(5E)-3-ethyl-2-(3-methyl-5-oxo-1-phenylpyrazol-4-ylidene)-5-(1,3,3-trimethylindol-2-ylidene)-1,3-thiazolidin-4-one
—— (5S)-9-[(2-chloro-6-fluorophenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H17ClFNO2
(5S)-9-[(2-chloro-6-fluorophenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-4-[(4-fluorophenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-(3-propoxyphenyl)pyrrolidine-2,3-dione —— C25H22FNO5
(5R)-4-[(4-fluorophenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-(3-propoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-7-(cyclobutylmethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one —— C18H28N2O
(5S)-7-(cyclobutylmethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1,3,8,8-tetramethyl-5-(4-nitrophenyl)-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione —— C21H22N4O5
(5S)-1,3,8,8-tetramethyl-5-(4-nitrophenyl)-5,7,9,10-tetrahydropyrimido[4,5-b]quinoline-2,4,6-trione
—— (5R)-9-[(2-chloro-6-fluorophenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H17ClFNO2
(5R)-9-[(2-chloro-6-fluorophenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(cyclobutylmethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one —— C18H28N2O
(5R)-7-(cyclobutylmethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-methoxyethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H27N3O3
(5S)-7-(2-methoxyethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-methoxyethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H27N3O3
(5R)-7-(2-methoxyethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S,7R)-N-(furan-2-ylmethyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H17F3N4O2
(5S,7R)-N-(furan-2-ylmethyl)-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1-methylpyrrole-3-carbonitrile —— C19H28N4O3
5-[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1-methylpyrrole-3-carbonitrile