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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(6S)-6-methyl-2-phenyldiazinane-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C21H21N5O2
5-[(6S)-6-methyl-2-phenyldiazinane-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one —— C19H22N2O3S
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one
—— (5R)-1-[(3-methoxyphenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C20H26N4O4
(5R)-1-[(3-methoxyphenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5R)-5-(1,3-benzodioxol-5-yl)-2-propylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione —— C21H21N3O4S
(5R)-5-(1,3-benzodioxol-5-yl)-2-propylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione
—— (5S)-7-(cyclopropylmethyl)-2-[2-(4-ethyl-3,5-dimethylpyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H32N4O2
(5S)-7-(cyclopropylmethyl)-2-[2-(4-ethyl-3,5-dimethylpyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-[[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methyl]-2-propan-2-yloxyphenyl]methanol —— C20H31NO3
[5-[[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methyl]-2-propan-2-yloxyphenyl]methanol
—— (5-methylpyrazin-2-yl)-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C20H22N6O
(5-methylpyrazin-2-yl)-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5R)-9-(3-pyridin-3-yloxypropyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H22N2O3
(5R)-9-(3-pyridin-3-yloxypropyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-[(2R)-2-(4-fluorophenyl)azetidine-1-carbonyl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C19H15FN4O2
5-[(2R)-2-(4-fluorophenyl)azetidine-1-carbonyl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— (5-methylpyrazin-2-yl)-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C20H22N6O
(5-methylpyrazin-2-yl)-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5R)-2-[(2-methylphenyl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2
(5R)-2-[(2-methylphenyl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[[2-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl]-1,3-oxazolidin-2-one —— C18H26N4O4
(5S)-5-[[2-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl]-1,3-oxazolidin-2-one
—— 5-fluoro-N-[(1S)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]quinazolin-4-amine —— C16H19FN6
5-fluoro-N-[(1S)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]quinazolin-4-amine
—— (5S)-7-(cyclopropylmethyl)-2-(3-phenoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O3
(5S)-7-(cyclopropylmethyl)-2-(3-phenoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-N-[(1R)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]-6-oxo-1H-pyridine-3-carboxamide —— C19H19ClN4O3
5-chloro-N-[(1R)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]-6-oxo-1H-pyridine-3-carboxamide
—— (5S)-9-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H22F2N2O2
(5S)-9-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(cyclopropylmethyl)-2-[2-(4-ethyl-3,5-dimethylpyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H32N4O2
(5R)-7-(cyclopropylmethyl)-2-[2-(4-ethyl-3,5-dimethylpyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-[[2-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl]-1,3-oxazolidin-2-one —— C18H26N4O4
(5R)-5-[[2-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl]-1,3-oxazolidin-2-one
—— [5-[[(3S)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methyl]-2-propan-2-yloxyphenyl]methanol —— C20H31NO3
[5-[[(3S)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methyl]-2-propan-2-yloxyphenyl]methanol
—— (5S,10bR)-9-methoxy-2,5-diphenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H20N2O2
(5S,10bR)-9-methoxy-2,5-diphenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-9-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H22F2N2O2
(5R)-9-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-(4-methylpiperazin-4-ium-1-yl)-2-nitro-N-(2-phenoxyethyl)aniline —— C19H25N4O3+
5-(4-methylpiperazin-4-ium-1-yl)-2-nitro-N-(2-phenoxyethyl)aniline
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(1H-imidazol-5-yl)ethyl]-5-methylpiperidin-2-one —— C19H23N3O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(1H-imidazol-5-yl)ethyl]-5-methylpiperidin-2-one
—— (5S)-9-(3-pyridin-3-yloxypropyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H22N2O3
(5S)-9-(3-pyridin-3-yloxypropyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(furan-2-ylmethyl)azanium —— C17H19N2O2+
(5,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(furan-2-ylmethyl)azanium
—— (5S)-2-[(2-methylphenyl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2
(5S)-2-[(2-methylphenyl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-[1-[(2S)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]triazol-4-yl]furan-2-yl]methanol —— C16H20N4O2S
[5-[1-[(2S)-2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]triazol-4-yl]furan-2-yl]methanol
—— (5R)-7-(2-hydroxyethyl)-2-[3-(1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3
(5R)-7-(2-hydroxyethyl)-2-[3-(1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-11-benzyl-5-(1-benzyl-2-methylindol-3-yl)-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7)-dien-3-one —— C32H31N4OS+
(5R)-11-benzyl-5-(1-benzyl-2-methylindol-3-yl)-8-thia-4,6-diaza-11-azoniatricyclo[7.4.0.02,7]trideca-1(9),2(7)-dien-3-one
—— (5S)-7-(2-hydroxyethyl)-2-[3-(1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3
(5S)-7-(2-hydroxyethyl)-2-[3-(1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[(3-methoxyphenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C20H26N4O4
(5S)-1-[(3-methoxyphenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5R)-2-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N3O4
(5R)-2-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-methoxyethyl)-2-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O2
(5S)-7-(2-methoxyethyl)-2-[(6-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-N-[(1S)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]-6-oxo-1H-pyridine-3-carboxamide —— C19H19ClN4O3
5-chloro-N-[(1S)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]-6-oxo-1H-pyridine-3-carboxamide
—— 5-(5-methylindol-2-ylidene)-3-pyridazin-3-yl-2H-1,2,4-oxadiazole —— C15H11N5O
5-(5-methylindol-2-ylidene)-3-pyridazin-3-yl-2H-1,2,4-oxadiazole
—— (5S)-2-(morpholine-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H29N3O4
(5S)-2-(morpholine-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N3O4
(5S)-2-[2-(3,5-dimethyl-1,2-oxazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(4-chloro-1-methylpyrazole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23ClN4O3
(5R)-2-(4-chloro-1-methylpyrazole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-N-cyclopropyl-5-methyl-N-[(1-methylpyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H23N3OS
(5R)-N-cyclopropyl-5-methyl-N-[(1-methylpyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-ethyl-4-methyl-6-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]pyrimidin-2-amine —— C18H31N5O
5-ethyl-4-methyl-6-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]pyrimidin-2-amine
—— (5S)-N-cyclopropyl-5-methyl-N-[(1-methylpyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C18H23N3OS
(5S)-N-cyclopropyl-5-methyl-N-[(1-methylpyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-2-(morpholine-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H29N3O4
(5R)-2-(morpholine-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-fluoro-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]quinazolin-4-amine —— C16H19FN6
5-fluoro-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]quinazolin-4-amine
—— (5S)-7-(cyclopropylmethyl)-2-[3-(2-oxopyridin-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H27N3O3
(5S)-7-(cyclopropylmethyl)-2-[3-(2-oxopyridin-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-2-one —— C23H33N3O2
(5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-2-one
—— (5S)-2-(4-chloro-1-methylpyrazole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23ClN4O3
(5S)-2-(4-chloro-1-methylpyrazole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]piperidin-2-one —— C18H22N4O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]piperidin-2-one
—— (5S)-7-(cyclobutylmethyl)-2-(4-imidazol-1-ylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5S)-7-(cyclobutylmethyl)-2-(4-imidazol-1-ylbutanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(3,5-dichloro-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H18Cl2N2O2
(5S)-2-(3,5-dichloro-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-2-one —— C23H33N3O2
(5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidin-2-one