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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-5-methyl-5-(4-methylpent-3-enyl)-1-(1,2-oxazol-3-ylmethyl)piperidin-2-one —— C16H24N2O2
(5R)-5-methyl-5-(4-methylpent-3-enyl)-1-(1,2-oxazol-3-ylmethyl)piperidin-2-one
—— (5S)-7-cyclopentyl-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O
(5S)-7-cyclopentyl-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propyl-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H21F3N4O2
(5S)-7-propyl-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-(3-chlorophenyl)-4-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-5-methylpiperazin-2-one —— C17H21ClN4O3
(5S)-1-(3-chlorophenyl)-4-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-5-methylpiperazin-2-one
—— (5S)-7-methyl-2-(1-propylpyrazol-4-yl)sulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O3S
(5S)-7-methyl-2-(1-propylpyrazol-4-yl)sulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one —— C14H15ClF3N3O
(5S)-2-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[3-(dimethylamino)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2
(5S)-7-(cyclopropylmethyl)-2-[3-(dimethylamino)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(5-fluoro-2-methylphenyl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25FN2O2
(5R)-2-[(5-fluoro-2-methylphenyl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H18FN3O3
(5S)-7-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-5-benzyl-4-(3-hydroxypropyl)-1-(3-phenylphenyl)piperazin-2-one —— C26H28N2O2
(5R)-5-benzyl-4-(3-hydroxypropyl)-1-(3-phenylphenyl)piperazin-2-one
—— (5S)-2-[(5-fluoro-2-methylphenyl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25FN2O2
(5S)-2-[(5-fluoro-2-methylphenyl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(4-chloro-3-fluorobenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H22ClFN2O2
(5S)-2-(4-chloro-3-fluorobenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C17H18FN3O3
(5R)-7-[(8-fluoro-4-oxo-1H-quinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R)-7-cyclopentyl-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O
(5R)-7-cyclopentyl-2-pyridin-4-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclopentyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H28N2O3S
(5S)-7-cyclopentyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-fluoro-N-[(2S)-1-imidazol-1-ylbutan-2-yl]quinazolin-4-amine —— C15H16FN5
5-fluoro-N-[(2S)-1-imidazol-1-ylbutan-2-yl]quinazolin-4-amine
—— (5R)-7-cyclopentyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H28N2O3S
(5R)-7-cyclopentyl-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-1-(2-amino-2-oxoethyl)piperidine-3-carbonyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C16H22N4O3S
5-[(3S)-1-(2-amino-2-oxoethyl)piperidine-3-carbonyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— (5R)-2-[(2-chloro-3,4-dimethoxyphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H25ClN2O3
(5R)-2-[(2-chloro-3,4-dimethoxyphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-amino-2-[(E)-2-(4-nitro-2-sulfonatophenyl)ethenyl]benzenesulfonate —— C14H10N2O8S2-2
5-amino-2-[(E)-2-(4-nitro-2-sulfonatophenyl)ethenyl]benzenesulfonate
—— (5S)-7-(cyclobutylmethyl)-2-[4-(1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O2
(5S)-7-(cyclobutylmethyl)-2-[4-(1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H25N3O2
(5R)-2-[2-(3,4-dihydro-1H-isoquinolin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propan-2-yl-2-(3-pyridin-2-yl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5S)-7-propan-2-yl-2-(3-pyridin-2-yl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(4-chloro-3-fluorobenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H22ClFN2O2
(5R)-2-(4-chloro-3-fluorobenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(4-Chloro-3-methylphenyl)-5-oxopentanoate —— C12H12ClO3-
5-(4-Chloro-3-methylphenyl)-5-oxopentanoate
—— [5-[1-[(3S)-1-benzylpyrrolidin-3-yl]triazol-4-yl]furan-2-yl]methanol —— C18H20N4O2
[5-[1-[(3S)-1-benzylpyrrolidin-3-yl]triazol-4-yl]furan-2-yl]methanol
—— (5S)-7-ethyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O2
(5S)-7-ethyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloro-3-phenyl-1H-indol-2-yl)-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methanone —— C22H23ClN2O2
(5-chloro-3-phenyl-1H-indol-2-yl)-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methanone
—— 5-[[4-[5-[(2S)-oxan-2-yl]furan-2-yl]triazol-1-yl]methyl]-3-pyridin-3-yl-1,2-oxazole —— C20H19N5O3
5-[[4-[5-[(2S)-oxan-2-yl]furan-2-yl]triazol-1-yl]methyl]-3-pyridin-3-yl-1,2-oxazole
—— 5-[[(5S)-6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl]sulfonyl]-1H-pyrimidine-2,4-dione —— C15H22N4O5S
5-[[(5S)-6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl]sulfonyl]-1H-pyrimidine-2,4-dione
—— (5-chloro-3-phenyl-1H-indol-2-yl)-[(3S)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methanone —— C22H23ClN2O2
(5-chloro-3-phenyl-1H-indol-2-yl)-[(3S)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methanone
—— (5R)-2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C21H25N3O3
(5R)-2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2S
(5R)-7-cyclohexyl-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-cycloheptyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C21H25N5O2
(5R)-1-cycloheptyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-7-cyclohexyl-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2S
(5S)-7-cyclohexyl-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C21H25N3O3
(5S)-2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3R)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide —— C17H26N2O3
5-[[(3R)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide
—— (5S)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-prop-2-enylpiperidin-2-one —— C15H17N5O2
(5S)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-prop-2-enylpiperidin-2-one
—— 5-[[(3S)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide —— C17H26N2O3
5-[[(3S)-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl]-N-methylfuran-2-carboxamide
—— (5-methyl-4-phenylthiophen-3-yl)-[(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone —— C20H23NO2S
(5-methyl-4-phenylthiophen-3-yl)-[(5S)-2-oxa-9-azaspiro[4.5]decan-9-yl]methanone
—— (5R)-2-(5-chloro-2-methoxybenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25ClN2O3
(5R)-2-(5-chloro-2-methoxybenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-bromo-N-(4-(2,3-dihydroimidazo[2,1-b]thiazol-6-yl)phenyl)furan-2-carboxamide —— C16H12BrN3O2S
5-bromo-N-(4-(2,3-dihydroimidazo[2,1-b]thiazol-6-yl)phenyl)furan-2-carboxamide
—— (5S)-1-cycloheptyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C21H25N5O2
(5S)-1-cycloheptyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-2-[(2-chloro-3,4-dimethoxyphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H25ClN2O3
(5S)-2-[(2-chloro-3,4-dimethoxyphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-cyclopentyl-5-[3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C21H34N4O2
(5S)-1-cyclopentyl-5-[3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-[(6R)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]pyridine-2-carbonitrile —— C20H27N5O2
5-[(6R)-2-[2-(dimethylamino)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]pyridine-2-carbonitrile
—— 5-[(1R)-1-[4-[2-(2-phenylethynyl)phenyl]triazol-1-yl]ethyl]-2H-tetrazole —— C19H15N7
5-[(1R)-1-[4-[2-(2-phenylethynyl)phenyl]triazol-1-yl]ethyl]-2H-tetrazole
—— (5S)-2-(5-chloro-2-methoxybenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25ClN2O3
(5S)-2-(5-chloro-2-methoxybenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-[4-(1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O2
(5R)-7-(cyclobutylmethyl)-2-[4-(1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-[1-[(3R)-1-benzylpyrrolidin-3-yl]triazol-4-yl]furan-2-yl]methanol —— C18H20N4O2
[5-[1-[(3R)-1-benzylpyrrolidin-3-yl]triazol-4-yl]furan-2-yl]methanol