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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-2-(4-methoxypiperidin-1-yl)sulfonyl-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C17H31N3O4S
(5S)-2-(4-methoxypiperidin-1-yl)sulfonyl-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-(2-ethylsulfonylethyl)-5-methylpiperidin-2-one —— C18H25NO5S
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-(2-ethylsulfonylethyl)-5-methylpiperidin-2-one
—— (5R)-5-[(2R,4S)-2-hexyl-1,3-dioxolan-4-yl]-3-hydroxyoxolane-2,4-dione —— C13H20O6
(5R)-5-[(2R,4S)-2-hexyl-1,3-dioxolan-4-yl]-3-hydroxyoxolane-2,4-dione
—— (5Z)-3-(4-fluorophenyl)-5-(3-methyl-1,3-benzothiazol-2-ylidene)-2-[(1S)-1-phenylethyl]imino-1,3-thiazolidin-4-one —— C25H20FN3OS2
(5Z)-3-(4-fluorophenyl)-5-(3-methyl-1,3-benzothiazol-2-ylidene)-2-[(1S)-1-phenylethyl]imino-1,3-thiazolidin-4-one
—— (5R,8S,8aR)-6-imino-8-(3-methoxy-4-propan-2-yloxyphenyl)-2-methyl-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile —— C23H25N5O2
(5R,8S,8aR)-6-imino-8-(3-methoxy-4-propan-2-yloxyphenyl)-2-methyl-3,5,8,8a-tetrahydro-1H-isoquinoline-5,7,7-tricarbonitrile
—— 5-(3-Ethylphenoxy)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene —— C9H9N4O-
5-(3-Ethylphenoxy)-1,2,3-triaza-4-azanidacyclopenta-2,5-diene
—— (5R)-2-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H26N4O3
(5R)-2-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[4-(butylsulfanylmethyl)-5-methylfuran-2-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H30N2O3S
(5S)-2-[4-(butylsulfanylmethyl)-5-methylfuran-2-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O3S
(5S)-7-(2-hydroxyethyl)-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[2-(3-amino-1H-1,2,4-triazol-5-yl)ethyl]-5-(1,3-benzodioxol-5-ylmethyl)-5-methylpiperidin-2-one —— C18H23N5O3
(5S)-1-[2-(3-amino-1H-1,2,4-triazol-5-yl)ethyl]-5-(1,3-benzodioxol-5-ylmethyl)-5-methylpiperidin-2-one
—— (5R)-7-(cyclopropylmethyl)-2-(5-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5R)-7-(cyclopropylmethyl)-2-(5-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[4-(butylsulfanylmethyl)-5-methylfuran-2-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H30N2O3S
(5R)-2-[4-(butylsulfanylmethyl)-5-methylfuran-2-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-fluorophenyl)-N-[(1R)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide —— C17H12F4N4O
5-(3-fluorophenyl)-N-[(1R)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide
—— (5R)-7-cyclohexyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O4
(5R)-7-cyclohexyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-(5-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5S)-7-(cyclopropylmethyl)-2-(5-propyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N3OS
(5S)-2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O3S
(5R)-7-(2-hydroxyethyl)-2-(3-thiophen-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H28N4O
(5R)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-(2-ethylpyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H27N3O2
(5R)-7-(cyclopropylmethyl)-2-(2-ethylpyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3
(5S)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-N-[(1R)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide —— C17H16ClN5O2
5-chloro-N-[(1R)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide
—— (5R)-2-[2-(azepan-1-yl)-2-oxoethyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H35N3O2
(5R)-2-[2-(azepan-1-yl)-2-oxoethyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H26N4O3
(5S)-2-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-[[2-(dimethylamino)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O
(5R)-7-(cyclopropylmethyl)-2-[[2-(dimethylamino)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-N,5-dimethyl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H21N3O2S
(5S)-N,5-dimethyl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-9-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H23NO2S
(5S)-9-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5,8-dimethyl-2-[[[(1R)-1-(1-methylpyrazol-4-yl)propyl]amino]methyl]-1H-quinolin-4-one —— C19H24N4O
5,8-dimethyl-2-[[[(1R)-1-(1-methylpyrazol-4-yl)propyl]amino]methyl]-1H-quinolin-4-one
—— (5R)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3
(5R)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3R)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-amine —— C16H18N2O2
5-[[(3R)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-amine
—— (5R)-1-[2-(4-hydroxypiperidin-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C19H28N2O2
(5R)-1-[2-(4-hydroxypiperidin-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-9-[[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H23N3O5
(5R)-9-[[3-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-methyl-N-[(1S)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide —— C21H27N5O
5-methyl-N-[(1S)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide
—— (5S)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H28N4O
(5S)-7-(cyclopropylmethyl)-2-[(2-pyrazol-1-ylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-3-butyl-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-(3-methylphenyl)methanone —— C16H19F3N2O2
[(5S)-3-butyl-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-(3-methylphenyl)methanone
—— (5S)-1-[2-(4-hydroxypiperidin-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C19H28N2O2
(5S)-1-[2-(4-hydroxypiperidin-1-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— 5-[(6S)-2-cyclopropyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile —— C20H24N4O3
5-[(6S)-2-cyclopropyl-3-oxo-2,8-diazaspiro[5.5]undecane-8-carbonyl]-6-methyl-2-oxo-1H-pyridine-3-carbonitrile
—— (5R)-N,5-dimethyl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H21N3O2S
(5R)-N,5-dimethyl-N-[(3-pyridin-4-yl-1,2-oxazol-5-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-1-[2-(3-amino-1H-1,2,4-triazol-5-yl)ethyl]-5-(1,3-benzodioxol-5-ylmethyl)-5-methylpiperidin-2-one —— C18H23N5O3
(5R)-1-[2-(3-amino-1H-1,2,4-triazol-5-yl)ethyl]-5-(1,3-benzodioxol-5-ylmethyl)-5-methylpiperidin-2-one
—— (5R)-2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N3OS
(5R)-2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-N-[(1R)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide —— C21H27N5O
5-methyl-N-[(1R)-3-(2-methylimidazol-1-yl)-1-phenylpropyl]-1-propylpyrazole-4-carboxamide
—— 5-(3-fluorophenyl)-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide —— C17H12F4N4O
5-(3-fluorophenyl)-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1H-pyrazole-4-carboxamide
—— (5S)-7-(cyclopropylmethyl)-2-[[2-(dimethylamino)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H29N5O
(5S)-7-(cyclopropylmethyl)-2-[[2-(dimethylamino)pyrimidin-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[2-(azepan-1-yl)-2-oxoethyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H35N3O2
(5S)-2-[2-(azepan-1-yl)-2-oxoethyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-N-[(1S)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide —— C17H16ClN5O2
5-chloro-N-[(1S)-1-(5-methyl-1-pyridin-2-ylpyrazol-4-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide
—— 5-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-amine —— C16H18N2O2
5-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]pyridin-3-amine
—— (5S)-2-(3-benzylsulfanylpropanoyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H26N2O2S
(5S)-2-(3-benzylsulfanylpropanoyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-methyl-2-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H24N2O4
(5S)-7-methyl-2-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N6O
(5R)-7-cyclohexyl-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclohexyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O4
(5S)-7-cyclohexyl-2-(6-methyl-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)-1H-pyrimidin-6-one —— C20H20N4O3
5-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)-1H-pyrimidin-6-one