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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-butyl-4-methyl-6-[(5S)-7-methyl-2,7-diazaspiro[4.4]nonan-2-yl]pyrimidin-2-amine —— C17H29N5
5-butyl-4-methyl-6-[(5S)-7-methyl-2,7-diazaspiro[4.4]nonan-2-yl]pyrimidin-2-amine
—— 5,7-dimethyl-4-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrido[2,3-d]pyrimidine —— C20H30N6
5,7-dimethyl-4-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrido[2,3-d]pyrimidine
—— 5-[(S)-1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H24N4O4S
5-[(S)-1,4-dioxa-8-azaspiro[4.5]decan-8-yl-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-2-(5-chloropyridin-2-yl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one —— C18H24ClN3O
(5R)-2-(5-chloropyridin-2-yl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-5-methoxy-1-oxa-9-azaspiro[5.5]undecane —— C16H26N2O3
(5R)-9-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
—— 5-[(S)-(2,4-dimethoxyphenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O4S
5-[(S)-(2,4-dimethoxyphenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-ethyl-N-[(1R)-1-(4-methylsulfonylphenyl)propyl]-1,3,4-oxadiazol-2-amine —— C14H19N3O3S
5-ethyl-N-[(1R)-1-(4-methylsulfonylphenyl)propyl]-1,3,4-oxadiazol-2-amine
—— 5-[(R)-(2-methoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O2S+
5-[(R)-(2-methoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5-chloropyridin-3-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H20ClN7O
(5-chloropyridin-3-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— 5-[(R)-(2,4-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O3S+
5-[(R)-(2,4-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O4S
5-[(R)-(2,4-dimethoxyphenyl)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,5-dimethoxyphenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H29N5O3S+2
5-[(S)-(2,5-dimethoxyphenyl)-(4-ethylpiperazine-1,4-diium-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,4-dimethoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H23N4O4S+
5-[(S)-(2,4-dimethoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-[(2S,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O2S+
5-[(S)-[(2S,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(4-ethylpiperazine-1,4-diium-1-yl)-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H27N5O2S+2
5-[(S)-(4-ethylpiperazine-1,4-diium-1-yl)-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(S)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-3-phenyl-1,2,4-oxadiazole —— C21H25N5O
5-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(R)-(4-ethylpiperazin-1-yl)-(5-methylfuran-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C17H23N5O2S
5-[(R)-(4-ethylpiperazin-1-yl)-(5-methylfuran-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2-methoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O2S+
5-[(S)-(2-methoxyphenyl)-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-morpholin-4-yl-2-[[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]methyl]pyridazin-3-one —— C15H19N5O4
5-morpholin-4-yl-2-[[5-[(2S)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl]methyl]pyridazin-3-one
—— 5-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-3-phenyl-1,2,4-oxadiazole —— C21H25N5O
5-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidin-1-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(S)-(2,5-dimethoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H23N4O4S+
5-[(S)-(2,5-dimethoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— [(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(4,5,6,7-tetrahydro-2-benzothiophen-1-yl)methanone —— C19H27NO3S
[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(4,5,6,7-tetrahydro-2-benzothiophen-1-yl)methanone
—— 5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(5-methylfuran-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H25N4O2S+
5-[(R)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]-(5-methylfuran-2-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5,7-dimethyl-4-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrido[2,3-d]pyrimidine —— C20H30N6
5,7-dimethyl-4-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrido[2,3-d]pyrimidine
—— 5-[(R)-(4-ethylpiperazine-1,4-diium-1-yl)-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H27N5OS+2
5-[(R)-(4-ethylpiperazine-1,4-diium-1-yl)-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-cyclopropyl-N-[(1S)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-1,3,4-oxadiazol-2-amine —— C17H19N5O2
5-cyclopropyl-N-[(1S)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-1,3,4-oxadiazol-2-amine
—— 5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C19H25N4O2S+
5-[(S)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]-(2-methylphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H22N4O4S
5-[(R)-(2,4-dimethoxyphenyl)-morpholin-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5S)-3-(5-chlorothiophen-2-yl)-N-[(2-morpholin-4-ylphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H20ClN3O3S
(5S)-3-(5-chlorothiophen-2-yl)-N-[(2-morpholin-4-ylphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione —— C13H21N3O5S
5-[(2S,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione
—— 5-[4-[(3R)-1-acetylpiperidine-3-carbonyl]piperazin-1-yl]-2-methylpyridazin-3-one —— C17H25N5O3
5-[4-[(3R)-1-acetylpiperidine-3-carbonyl]piperazin-1-yl]-2-methylpyridazin-3-one
—— 5-[4-[(3S)-1-acetylpiperidine-3-carbonyl]piperazin-1-yl]-2-methylpyridazin-3-one —— C17H25N5O3
5-[4-[(3S)-1-acetylpiperidine-3-carbonyl]piperazin-1-yl]-2-methylpyridazin-3-one
—— 5-[(R)-(2,5-dimethoxyphenyl)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O4S
5-[(R)-(2,5-dimethoxyphenyl)-[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(R)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H26N4O3S
5-[(R)-(2,4-dimethoxyphenyl)-(4-methylpiperidin-1-yl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-cyclopropyl-N-[(1R)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-1,3,4-oxadiazol-2-amine —— C17H19N5O2
5-cyclopropyl-N-[(1R)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-1,3,4-oxadiazol-2-amine
—— 5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H25N4O4S+
5-[(R)-1,4-dioxa-8-azoniaspiro[4.5]decan-8-yl-(2-methoxyphenyl)methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,5-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O3S+
5-[(S)-(2,5-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,4-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H29N4O3S+
5-[(S)-(2,4-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-ium-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5R)-7-cyclopentyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H31N5O2
(5R)-7-cyclopentyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-bromo-3-chloro-N-[(2S)-1-morpholin-4-yl-1-oxopropan-2-yl]-1H-indole-2-carboxamide —— C16H17BrClN3O3
5-bromo-3-chloro-N-[(2S)-1-morpholin-4-yl-1-oxopropan-2-yl]-1H-indole-2-carboxamide
—— 5-[(S)-(2,4-dimethoxyphenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C20H27N4O4S+
5-[(S)-(2,4-dimethoxyphenyl)-[(2R,6R)-2,6-dimethylmorpholin-4-ium-4-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione —— C14H23N3O4S
5-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-1,3,6-trimethylpyrimidine-2,4-dione
—— (5S)-7-cyclopentyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H31N5O2
(5S)-7-cyclopentyl-2-(5-methyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-Methyl-2-phenylpyrazol-3-yl) 2,4,5-trimethylbenzenesulfonate —— C19H20N2O3S
(5-Methyl-2-phenylpyrazol-3-yl) 2,4,5-trimethylbenzenesulfonate
—— 5-bromo-N-[(2R)-1-[cyclopropyl-(4-methylcyclohexyl)amino]-1-oxopropan-2-yl]thiophene-2-carboxamide —— C18H25BrN2O2S
5-bromo-N-[(2R)-1-[cyclopropyl-(4-methylcyclohexyl)amino]-1-oxopropan-2-yl]thiophene-2-carboxamide
—— 5-[(R)-(2,4-dimethoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C18H23N4O4S+
5-[(R)-(2,4-dimethoxyphenyl)-morpholin-4-ium-4-ylmethyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— 5-[(S)-(2,4-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol —— C21H28N4O3S
5-[(S)-(2,4-dimethoxyphenyl)-[(3S,5S)-3,5-dimethylpiperidin-1-yl]methyl]-2-methyl-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-ol
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]methanone —— C19H26N4O3
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(5R)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]methanone
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]methanone —— C19H26N4O3
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-[(5S)-5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]methanone