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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-(2-chlorophenyl)-N-[(1R)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide —— C18H19ClN4O2
5-(2-chlorophenyl)-N-[(1R)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
—— (5R)-7-propan-2-yl-2-(3-pyridin-4-yl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5R)-7-propan-2-yl-2-(3-pyridin-4-yl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(6-methoxy-1H-benzimidazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H23N3O3
(5S)-9-[2-(6-methoxy-1H-benzimidazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-4-benzyl-12-(methoxymethyl)-1-aza-4-azoniatetracyclo[7.6.1.05,16.010,15]hexadeca-9(16),10(15),11,13-tetraene —— C23H27N2O+
(5R)-4-benzyl-12-(methoxymethyl)-1-aza-4-azoniatetracyclo[7.6.1.05,16.010,15]hexadeca-9(16),10(15),11,13-tetraene
—— (5R)-2-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2S2
(5R)-2-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(2-pyrimidin-2-yl-1,3-thiazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H18N4O2S
(5R)-9-[(2-pyrimidin-2-yl-1,3-thiazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(2-methoxyethyl)-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N3O3S
(5R)-7-(2-methoxyethyl)-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-chlorophenyl)-N-[(1S)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide —— C18H19ClN4O2
5-(2-chlorophenyl)-N-[(1S)-1-(4-propyl-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
—— (5S)-5-methyl-1-(4-methylphenyl)-4-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-2-one —— C17H22N4O2S
(5S)-5-methyl-1-(4-methylphenyl)-4-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]piperazin-2-one
—— 5-[[(1R)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]pyridine-2-carbonitrile —— C15H13N3O
5-[[(1R)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]pyridine-2-carbonitrile
—— 5-[[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl]-2-ethylpyrimidine —— C21H27N3O2
5-[[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl]-2-ethylpyrimidine
—— (5S)-7-cyclohexyl-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O
(5S)-7-cyclohexyl-2-(pyridin-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2
(5S)-7-(cyclopropylmethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methanone —— C20H28N4O3
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(2S)-2-(2-morpholin-4-ylethyl)piperidin-1-yl]methanone
—— (5S)-2-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2S2
(5S)-2-[2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[3-[2-(cyclopropylmethyl)-4-oxo-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-7-yl]-3-oxopropyl]imidazolidine-2,4-dione —— C17H21N5O4
(5S)-5-[3-[2-(cyclopropylmethyl)-4-oxo-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-7-yl]-3-oxopropyl]imidazolidine-2,4-dione
—— (5S)-2-(6-morpholin-4-ylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O2
(5S)-2-(6-morpholin-4-ylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O3
(5R)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]pyridine-2-carbonitrile —— C15H13N3O
5-[[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]amino]pyridine-2-carbonitrile
—— 5-(3-fluorophenyl)-N-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]-1H-pyrazole-4-carboxamide —— C20H18FN3O
5-(3-fluorophenyl)-N-[(2R)-1,2,3,4-tetrahydronaphthalen-2-yl]-1H-pyrazole-4-carboxamide
—— (5R)-2-(2-ethyl-6-oxo-1H-pyridine-4-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O4
(5R)-2-(2-ethyl-6-oxo-1H-pyridine-4-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[4-(methylamino)pyrimidin-2-yl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O2
(5R)-2-[4-(methylamino)pyrimidin-2-yl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-ethyl-2-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5S)-7-ethyl-2-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O3
(5S)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(2S)-1-morpholin-4-yl-1-oxopropan-2-yl]amino]pyridine-2-carbonitrile —— C13H16N4O2
5-[[(2S)-1-morpholin-4-yl-1-oxopropan-2-yl]amino]pyridine-2-carbonitrile
—— (5R)-7-ethyl-2-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5R)-7-ethyl-2-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(2R)-1-morpholin-4-yl-1-oxopropan-2-yl]amino]pyridine-2-carbonitrile —— C13H16N4O2
5-[[(2R)-1-morpholin-4-yl-1-oxopropan-2-yl]amino]pyridine-2-carbonitrile
—— (5R)-9-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H19F2NO3
(5R)-9-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-2-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3
(5R)-2-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propan-2-yl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2
(5S)-7-propan-2-yl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(oxan-4-yl)-2-(6-oxo-1H-pyrazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O4
(5R)-7-(oxan-4-yl)-2-(6-oxo-1H-pyrazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-(azepan-1-yl)piperidin-1-yl]pyridine-2-carbonitrile —— C17H24N4
5-[(3R)-3-(azepan-1-yl)piperidin-1-yl]pyridine-2-carbonitrile
—— (5S)-2-[4-(methylamino)pyrimidin-2-yl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O2
(5S)-2-[4-(methylamino)pyrimidin-2-yl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-(azepan-1-yl)piperidin-1-yl]pyridine-2-carbonitrile —— C17H24N4
5-[(3S)-3-(azepan-1-yl)piperidin-1-yl]pyridine-2-carbonitrile
—— 5-(Azepan-1-ylsulfonyl)-2-chlorobenzoate —— C13H15ClNO4S-
5-(Azepan-1-ylsulfonyl)-2-chlorobenzoate
—— 5-[(2R)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile —— C18H19N3OS
5-[(2R)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile
—— 5-fluoro-2-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]benzonitrile —— C15H15FN4
5-fluoro-2-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]benzonitrile
—— (5S)-7-(2-methoxyethyl)-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N3O3S
(5S)-7-(2-methoxyethyl)-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(2S)-2-cyclopropyl-2-(dimethylamino)ethyl]amino]pyridine-2-carbonitrile —— C13H18N4
5-[[(2S)-2-cyclopropyl-2-(dimethylamino)ethyl]amino]pyridine-2-carbonitrile
—— (5R)-7-(cyclopropylmethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2
(5R)-7-(cyclopropylmethyl)-2-[2-(methylamino)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-fluoro-2-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]benzonitrile —— C15H15FN4
5-fluoro-2-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]benzonitrile
—— 5-chloro-2-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]pyridine —— C13H15ClN4
5-chloro-2-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]pyridine
—— (5S)-7-(cyclopropylmethyl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O2S
(5S)-7-(cyclopropylmethyl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-O'-tert-butyl 3-O'-prop-2-enyl (3S)-2'-amino-6'-methyl-2-oxospiro[1H-indole-3,4'-pyran]-3',5'-dicarboxylate —— C22H24N2O6
5-O'-tert-butyl 3-O'-prop-2-enyl (3S)-2'-amino-6'-methyl-2-oxospiro[1H-indole-3,4'-pyran]-3',5'-dicarboxylate
—— (5S)-2-[(Z)-[4-[(4-fluorophenyl)methoxy]phenyl]methylidenehydrazinylidene]-5-propan-2-yl-1,3-thiazolidin-4-one —— C20H20FN3O2S
(5S)-2-[(Z)-[4-[(4-fluorophenyl)methoxy]phenyl]methylidenehydrazinylidene]-5-propan-2-yl-1,3-thiazolidin-4-one
—— (5S,7R)-5-(4-bromophenyl)-7-(2-methylphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine —— C18H18BrN5
(5S,7R)-5-(4-bromophenyl)-7-(2-methylphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine
—— (5S,7S)-5-(2-chlorophenyl)-7-(4-phenylmethoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C24H21ClN4O
(5S,7S)-5-(2-chlorophenyl)-7-(4-phenylmethoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (5R)-5-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-3-phenyl-2-sulfanylidene-5,6-dihydro-4H-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C24H17Cl2N3O2S2
(5R)-5-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-3-phenyl-2-sulfanylidene-5,6-dihydro-4H-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 5-chloro-2-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]pyridine —— C13H15ClN4
5-chloro-2-[(3S)-3-(1H-imidazol-2-yl)piperidin-1-yl]pyridine
—— (5S)-9-[(3,5-dimethyl-1-propylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H27N3O2
(5S)-9-[(3,5-dimethyl-1-propylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one