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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-1-ethyl-5-[4-(2-pyrrol-1-ylethyl)piperazine-1-carbonyl]piperidin-2-one —— C18H28N4O2
(5R)-1-ethyl-5-[4-(2-pyrrol-1-ylethyl)piperazine-1-carbonyl]piperidin-2-one
—— (5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(2-fluorophenyl)methyl]piperidin-2-one —— C16H18FN3O2
(5R)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(2-fluorophenyl)methyl]piperidin-2-one
—— 5-acetyl-N-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]thiophene-2-carboxamide —— C18H19NO4S
5-acetyl-N-[[(3S)-7-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]thiophene-2-carboxamide
—— 5-butyl-4-[(3R)-3-methoxypyrrolidin-1-yl]-6-methylpyrimidin-2-amine —— C14H24N4O
5-butyl-4-[(3R)-3-methoxypyrrolidin-1-yl]-6-methylpyrimidin-2-amine
—— (5R)-7-(2-hydroxyethyl)-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O3S
(5R)-7-(2-hydroxyethyl)-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— [5-[(2R)-oxolan-2-yl]thiophen-2-yl]-[4-(thian-4-yl)piperazin-1-yl]methanone —— C18H26N2O2S2
[5-[(2R)-oxolan-2-yl]thiophen-2-yl]-[4-(thian-4-yl)piperazin-1-yl]methanone
—— (5S)-1-ethyl-5-[4-(2-pyrrol-1-ylethyl)piperazine-1-carbonyl]piperidin-2-one —— C18H28N4O2
(5S)-1-ethyl-5-[4-(2-pyrrol-1-ylethyl)piperazine-1-carbonyl]piperidin-2-one
—— (5R)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H27N3O4S
(5R)-7-(cyclobutylmethyl)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-cyclopropyl-N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide —— C22H25N5O
5-cyclopropyl-N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-1H-pyrazole-3-carboxamide
—— (5S)-7-methyl-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O
(5S)-7-methyl-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C16H25N5O2S
(5R)-2-[2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-methoxyethyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O3
(5R)-7-(2-methoxyethyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide —— C17H17N5O2S
5-[(2S)-oxolan-2-yl]-N-[(1-phenyltetrazol-5-yl)methyl]thiophene-2-carboxamide
—— (5R)-2-[2-(1-methylpyrazol-4-yl)ethyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C17H28N4O
(5R)-2-[2-(1-methylpyrazol-4-yl)ethyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C20H22N6O2
5-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— (5S)-N,5-dimethyl-N-[2-(2-methylimidazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H23N3OS
(5S)-N,5-dimethyl-N-[2-(2-methylimidazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1,2-oxazol-5-ylmethyl)piperidin-2-one —— C18H20N2O4
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1,2-oxazol-5-ylmethyl)piperidin-2-one
—— (5S)-9-(imidazo[1,2-a]pyrimidin-2-ylmethyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H18N4O2
(5S)-9-(imidazo[1,2-a]pyrimidin-2-ylmethyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(2-methoxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H21F3N4O3
(5R)-7-(2-methoxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O
(5R)-7-methyl-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-methoxyethyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O3
(5S)-7-(2-methoxyethyl)-2-[2-(N-methylanilino)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclohexyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O2
(5S)-7-cyclohexyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C17H19N5O2S
5-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— 5-butyl-4-[(3S)-3-methoxypyrrolidin-1-yl]-6-methylpyrimidin-2-amine —— C14H24N4O
5-butyl-4-[(3S)-3-methoxypyrrolidin-1-yl]-6-methylpyrimidin-2-amine
—— (5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(2-fluorophenyl)methyl]piperidin-2-one —— C16H18FN3O2
(5S)-5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(2-fluorophenyl)methyl]piperidin-2-one
—— (5R)-2-[3-(benzenesulfonyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H22N2O4S
(5R)-2-[3-(benzenesulfonyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-(1-ethylpyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5R)-7-(cyclobutylmethyl)-2-(1-ethylpyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-[(4-propan-2-ylthiadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H30N4OS
(5R)-7-(cyclobutylmethyl)-2-[(4-propan-2-ylthiadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-ethyl-1H-pyrrol-2-yl)-[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C19H31N3O3
(5-ethyl-1H-pyrrol-2-yl)-[(4R)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— (5S)-2-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N5O2
(5S)-2-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C17H19N5O2S
5-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (5S)-2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O
(5S)-2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(7-chloro-4-oxo-1H-quinoline-3-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H20ClN3O3
(5S)-2-(7-chloro-4-oxo-1H-quinoline-3-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(7-chloro-4-oxo-1H-quinoline-3-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H20ClN3O3
(5R)-2-(7-chloro-4-oxo-1H-quinoline-3-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-(1-ethylpyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O2
(5S)-7-(cyclobutylmethyl)-2-(1-ethylpyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-2-pyridin-2-yl-1H-pyrimidin-6-one —— C20H22N6O2
5-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-2-pyridin-2-yl-1H-pyrimidin-6-one
—— (5R)-2-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N5O2
(5R)-2-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-methoxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H21F3N4O3
(5S)-7-(2-methoxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(6-aminopyridine-3-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2
(5S)-2-(6-aminopyridine-3-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O
(5R)-2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-N,5-dimethyl-N-[2-(2-methylimidazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H23N3OS
(5R)-N,5-dimethyl-N-[2-(2-methylimidazol-1-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-9-[(3-methyl-1-benzofuran-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H21NO3
(5R)-9-[(3-methyl-1-benzofuran-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-2-(2-amino-6-propan-2-ylpyrimidine-4-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H29N5O2
(5R)-2-(2-amino-6-propan-2-ylpyrimidine-4-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(5-methoxy-4-oxopyran-2-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H24N2O5
(5R)-2-(5-methoxy-4-oxopyran-2-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(5-methoxy-4-oxopyran-2-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C18H24N2O5
(5S)-2-(5-methoxy-4-oxopyran-2-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(4aR)-9-bromo-5,11-dioxo-2,4,4a,6-tetrahydro-1H-pyrazino[2,1-c][1,4]benzodiazepin-3-yl]-5-oxopentanoate —— C17H17BrN3O5-
5-[(4aR)-9-bromo-5,11-dioxo-2,4,4a,6-tetrahydro-1H-pyrazino[2,1-c][1,4]benzodiazepin-3-yl]-5-oxopentanoate
—— (5-ethyl-1H-pyrrol-2-yl)-[(4S)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C19H31N3O3
(5-ethyl-1H-pyrrol-2-yl)-[(4S)-4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1,2-oxazol-5-ylmethyl)piperidin-2-one —— C18H20N2O4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1,2-oxazol-5-ylmethyl)piperidin-2-one
—— (5S)-9-[(3-methyl-1-benzofuran-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H21NO3
(5S)-9-[(3-methyl-1-benzofuran-2-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-9-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H24N2O3
(5R)-9-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one