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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-1-(2-morpholin-4-ylethyl)-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C16H26N4O3
(5S)-1-(2-morpholin-4-ylethyl)-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5R)-7-(2-methoxyethyl)-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O3
(5R)-7-(2-methoxyethyl)-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propyl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5S)-7-propyl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclopentyl-2-[3-(1,2,4-triazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O2
(5S)-7-cyclopentyl-2-[3-(1,2,4-triazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one —— C16H21N5O4
5-[(3R)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl]-2-methyl-1H-pyrimidin-6-one
—— (5R)-7-(2-hydroxyethyl)-2-[(4-methyl-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C14H23N5O2
(5R)-7-(2-hydroxyethyl)-2-[(4-methyl-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3R)-1-(2-methoxyacetyl)pyrrolidin-3-yl]methyl]-1H-pyridin-2-one —— C13H18N2O3
5-[[(3R)-1-(2-methoxyacetyl)pyrrolidin-3-yl]methyl]-1H-pyridin-2-one
—— (5S)-2-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H24N4O
(5S)-2-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-methoxyethyl)-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O3
(5S)-7-(2-methoxyethyl)-2-(1-propan-2-ylpyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(3,4-dihydro-2H-chromen-6-ylmethyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H23NO3
(5R)-9-(3,4-dihydro-2H-chromen-6-ylmethyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H26N4O3
(5R)-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H30N4O
(5S)-7-(cyclobutylmethyl)-2-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidine-1-carbonyl]-1-methylpyrrole-3-carboxamide —— C17H17F2N3O3
5-[(2S,4R)-2-(2,5-difluorophenyl)-4-hydroxypyrrolidine-1-carbonyl]-1-methylpyrrole-3-carboxamide
—— (5S)-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)-1-(2-pyridin-2-ylethyl)piperidin-2-one —— C21H20N6O2
(5S)-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)-1-(2-pyridin-2-ylethyl)piperidin-2-one
—— (5R)-7-(2-hydroxyethyl)-2-(2-methylthieno[3,2-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H22N4O2S
(5R)-7-(2-hydroxyethyl)-2-(2-methylthieno[3,2-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(4-methoxypyrimidin-2-yl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O2
(5R)-2-(4-methoxypyrimidin-2-yl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O2
(5R)-7-cyclohexyl-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(2,5-dimethyl-1,2,4-triazol-3-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H29N5O2
(5R)-2-[(2,5-dimethyl-1,2,4-triazol-3-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H30N4O
(5R)-7-(cyclobutylmethyl)-2-[(3-methylimidazo[1,5-a]pyridin-1-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-2-[6-methyl-2-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C20H24N4O2
(5R)-7-methyl-2-[6-methyl-2-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1S)-1-[4-(6-chloro-1,3-benzodioxol-5-yl)triazol-1-yl]ethyl]-2H-tetrazole —— C12H10ClN7O2
5-[(1S)-1-[4-(6-chloro-1,3-benzodioxol-5-yl)triazol-1-yl]ethyl]-2H-tetrazole
—— (5S)-2-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H30N2O3
(5S)-2-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-cyclohexyl-2-(1,2-dimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O2
(5S)-7-cyclohexyl-2-(1,2-dimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H30N2O3
(5R)-2-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one —— C15H24N2O2
(5S)-7-(2-hydroxyethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H25N3O4S
(5R)-2-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-(propoxymethyl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C18H22N4O3
5-[(3S)-3-(propoxymethyl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— (5R)-2-[2-(4-fluorophenoxy)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H25FN2O4
(5R)-2-[2-(4-fluorophenoxy)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[(4-chloro-2-pyrrolidin-1-yl-1,3-thiazol-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C17H25ClN4OS
(5S)-2-[(4-chloro-2-pyrrolidin-1-yl-1,3-thiazol-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H22N4O2
(5R)-9-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(2-hydroxyethyl)-2-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H24N4O4
(5R)-7-(2-hydroxyethyl)-2-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[4-[(3S)-oxolan-3-yl]triazol-1-yl]methyl]-4-propan-2-ylthiadiazole —— C12H17N5OS
5-[[4-[(3S)-oxolan-3-yl]triazol-1-yl]methyl]-4-propan-2-ylthiadiazole
—— (5S)-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)-1-(pyridin-2-ylmethyl)piperidin-2-one —— C16H20N4O2
(5S)-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)-1-(pyridin-2-ylmethyl)piperidin-2-one
—— (5S)-7-cyclohexyl-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O2
(5S)-7-cyclohexyl-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-propyl-1H-pyrazol-3-yl)-[(2S)-2-(trifluoromethyl)pyrrolidin-1-yl]methanone —— C12H16F3N3O
(5-propyl-1H-pyrazol-3-yl)-[(2S)-2-(trifluoromethyl)pyrrolidin-1-yl]methanone
—— (5R)-7-cyclohexyl-2-(1,2-dimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H31N3O2
(5R)-7-cyclohexyl-2-(1,2-dimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(5-cyclohexylsulfanylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H28N2O2S
(5R)-2-[(5-cyclohexylsulfanylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one —— C15H24N2O2
(5R)-7-(2-hydroxyethyl)-2-pent-2-ynyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-N-benzyl-5-hydroxy-N-methyl-1-oxa-9-azaspiro[5.5]undecane-9-sulfonamide —— C17H26N2O4S
(5R)-N-benzyl-5-hydroxy-N-methyl-1-oxa-9-azaspiro[5.5]undecane-9-sulfonamide
—— 5-[(1S)-1-(2-methylimidazol-1-yl)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C12H12N6O
5-[(1S)-1-(2-methylimidazol-1-yl)ethyl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— (5R)-7-cyclopentyl-2-[3-(1,2,4-triazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O2
(5R)-7-cyclopentyl-2-[3-(1,2,4-triazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H24F4N2O
(5S)-7-(cyclopropylmethyl)-2-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(4-chloro-2-pyrrolidin-1-yl-1,3-thiazol-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C17H25ClN4OS
(5R)-2-[(4-chloro-2-pyrrolidin-1-yl-1,3-thiazol-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[(5-cyclohexylsulfanylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H28N2O2S
(5S)-2-[(5-cyclohexylsulfanylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-(2-methylthieno[3,2-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H22N4O2S
(5S)-7-(2-hydroxyethyl)-2-(2-methylthieno[3,2-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H24N4O
(5R)-2-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-propyl-1H-pyrazol-3-yl)-[(2R)-2-(trifluoromethyl)pyrrolidin-1-yl]methanone —— C12H16F3N3O
(5-propyl-1H-pyrazol-3-yl)-[(2R)-2-(trifluoromethyl)pyrrolidin-1-yl]methanone
—— (5S)-7-methyl-2-[2-[(2-methylphenyl)methylsulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H26N2O2S
(5S)-7-methyl-2-[2-[(2-methylphenyl)methylsulfanyl]acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide —— C18H16ClN5O2
5-chloro-N-[(1S)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide
—— 5-chloro-N-[(1R)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide —— C18H16ClN5O2
5-chloro-N-[(1R)-1-(4-methyl-2-pyridin-4-ylpyrimidin-5-yl)ethyl]-6-oxo-1H-pyridine-3-carboxamide