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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(2-ethylimidazol-1-yl)ethyl]-5-methylpiperidin-2-one —— C21H27N3O3
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(2-ethylimidazol-1-yl)ethyl]-5-methylpiperidin-2-one
—— 5-fluoro-N-methyl-2-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidin-4-amine —— C17H22FN9
5-fluoro-N-methyl-2-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidin-4-amine
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(3S)-3-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C19H23N5O3
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(3S)-3-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (5R)-2-(4-aminopyrimidin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H25N5O2
(5R)-2-(4-aminopyrimidin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one —— C20H22N2O5
5-[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(2-ethylimidazol-1-yl)ethyl]-5-methylpiperidin-2-one —— C21H27N3O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(2-ethylimidazol-1-yl)ethyl]-5-methylpiperidin-2-one
—— 5-[(2R)-oxolan-2-yl]-N-[(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)methyl]thiophene-2-carboxamide —— C16H15N5O3S
5-[(2R)-oxolan-2-yl]-N-[(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)methyl]thiophene-2-carboxamide
—— (5R)-7-(cyclobutylmethyl)-2-(5-methoxy-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O5
(5R)-7-(cyclobutylmethyl)-2-(5-methoxy-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(5-methylthiophen-2-yl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]-1H-pyrazole-3-carboxamide —— C16H17N5OS
5-(5-methylthiophen-2-yl)-N-[(2S)-1-pyrazin-2-ylpropan-2-yl]-1H-pyrazole-3-carboxamide
—— 5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]pyrazin-2-amine —— C14H15N3O
5-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]pyrazin-2-amine
—— (5R)-2-ethylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C15H26N2O4S
(5R)-2-ethylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R,10bS)-5-(4-ethoxy-3-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H22N2O3S
(5R,10bS)-5-(4-ethoxy-3-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-7-(oxan-4-yl)-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2
(5S)-7-(oxan-4-yl)-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(4-hydroxyphenyl)ethyl]-5-methylpiperidin-2-one —— C22H25NO4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(4-hydroxyphenyl)ethyl]-5-methylpiperidin-2-one
—— (5S)-7-(cyclobutylmethyl)-2-(5-methoxy-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O5
(5S)-7-(cyclobutylmethyl)-2-(5-methoxy-4-oxopyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one —— C20H22N2O5
5-[(3R)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-4-hydroxy-1H-pyridin-2-one
—— (5S,10bS)-5-(2-butoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H24N2O2S
(5S,10bS)-5-(2-butoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-2-ethylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C15H26N2O4S
(5S)-2-ethylsulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(7-chloro-1-methylindole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H20ClN3O2
(5R)-2-(7-chloro-1-methylindole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(7-chloro-1-methylindole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H20ClN3O2
(5S)-2-(7-chloro-1-methylindole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R,10bS)-5-(3-ethoxy-4-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H22N2O3S
(5R,10bS)-5-(3-ethoxy-4-methoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-(4-ethylphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H20N2OS
(5S,10bS)-5-(4-ethylphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-(5-methylthiophen-2-yl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]-1H-pyrazole-3-carboxamide —— C16H17N5OS
5-(5-methylthiophen-2-yl)-N-[(2R)-1-pyrazin-2-ylpropan-2-yl]-1H-pyrazole-3-carboxamide
—— (5S)-7-(2-methoxyethyl)-2-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O3
(5S)-7-(2-methoxyethyl)-2-(1-methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methanone —— C15H20ClN3O2
(5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methanone
—— (5R)-5-methyl-5-(4-methylpent-3-enyl)-1-(2-pyridin-4-ylethyl)piperidin-2-one —— C19H28N2O
(5R)-5-methyl-5-(4-methylpent-3-enyl)-1-(2-pyridin-4-ylethyl)piperidin-2-one
—— 5-[(5R)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile —— C19H24N4O2
5-[(5R)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile
—— (5R)-9-[(3-pyridin-3-yl-1,2-oxazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H19N3O3
(5R)-9-[(3-pyridin-3-yl-1,2-oxazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one —— C20H26N4O3
(5R)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one
—— (5S)-1-[(4-chlorophenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C19H23ClN4O3
(5S)-1-[(4-chlorophenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— (5S)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H26N4O3
(5S)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5R)-7-cyclohexyl-2-(1-methyl-6-oxopyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O3
(5R)-7-cyclohexyl-2-(1-methyl-6-oxopyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-methyl-5-(4-methylpent-3-enyl)-1-(2-pyridin-4-ylethyl)piperidin-2-one —— C19H28N2O
(5S)-5-methyl-5-(4-methylpent-3-enyl)-1-(2-pyridin-4-ylethyl)piperidin-2-one
—— (5R)-2-[2-(4-fluorophenyl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN2O3
(5R)-2-[2-(4-fluorophenyl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(5S)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile —— C19H24N4O2
5-[(5S)-7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methylpyrrole-3-carbonitrile
—— (5R,10bS)-5-(4-methoxy-3-methylphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H20N2O2S
(5R,10bS)-5-(4-methoxy-3-methylphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5-chloropyridin-3-yl)-[(3S)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methanone —— C15H19ClN2O2
(5-chloropyridin-3-yl)-[(3S)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methanone
—— (5S)-7-(cyclopropylmethyl)-2-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O3
(5S)-7-(cyclopropylmethyl)-2-[2-(2,4-dimethyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloropyridin-3-yl)-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methanone —— C15H19ClN2O2
(5-chloropyridin-3-yl)-[(3R)-3-(hydroxymethyl)-3-prop-2-enylpiperidin-1-yl]methanone
—— 5-[2-[4-[(3S)-oxolan-3-yl]triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C10H14N6OS
5-[2-[4-[(3S)-oxolan-3-yl]triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine
—— (5R,10bS)-5-(2-propoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H22N2O2S
(5R,10bS)-5-(2-propoxyphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-chloro-N-(4,6-difluoro-1,3-benzothiazol-2-yl)-N-[2-(dimethylamino)ethyl]thiophene-2-carboxamide —— C16H14ClF2N3OS2
5-chloro-N-(4,6-difluoro-1,3-benzothiazol-2-yl)-N-[2-(dimethylamino)ethyl]thiophene-2-carboxamide
—— (5R)-3-(3-nitrophenyl)-5-(4-nitrophenyl)-4,5-dihydro-1H-pyrazole —— C15H12N4O4
(5R)-3-(3-nitrophenyl)-5-(4-nitrophenyl)-4,5-dihydro-1H-pyrazole
—— 5-chloro-N-[3-(dimethylamino)propyl]-N-(4-methyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide —— C18H20ClN3OS2
5-chloro-N-[3-(dimethylamino)propyl]-N-(4-methyl-1,3-benzothiazol-2-yl)thiophene-2-carboxamide
—— 5-(2-methoxyphenyl)-N-(6-(methylthio)benzo[d]thiazol-2-yl)-1,3,4-oxadiazol-2-amine —— C17H14N4O2S2
5-(2-methoxyphenyl)-N-(6-(methylthio)benzo[d]thiazol-2-yl)-1,3,4-oxadiazol-2-amine
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)methanone —— C16H19N3OS
[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)methanone
—— (5R)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H26N4O3
(5R)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— [(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)methanone —— C16H19N3OS
[(5R)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-5-yl)methanone
—— (5S)-7-cyclohexyl-2-(2-ethyl-5-methylpyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H32N4O2
(5S)-7-cyclohexyl-2-(2-ethyl-5-methylpyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[2-[4-[(3R)-oxolan-3-yl]triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C10H14N6OS
5-[2-[4-[(3R)-oxolan-3-yl]triazol-1-yl]ethyl]-1,3,4-thiadiazol-2-amine