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—— (5S)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H19FN4O3
(5S)-N-[(1R)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R)-9-[(3-methyl-1-prop-2-enylpyrazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H27N3O2
(5R)-9-[(3-methyl-1-prop-2-enylpyrazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5S)-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2-oxa-9-azaspiro[4.5]decane —— C16H21N3OS
(5S)-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2-oxa-9-azaspiro[4.5]decane
—— (5S)-9-[(3-methyl-1-prop-2-enylpyrazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H27N3O2
(5S)-9-[(3-methyl-1-prop-2-enylpyrazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-(furan-2-yl)-N-[(1S)-1-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)ethyl]-1,2-oxazole-3-carboxamide —— C19H17N3O4
5-(furan-2-yl)-N-[(1S)-1-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)ethyl]-1,2-oxazole-3-carboxamide
—— (5R)-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2-oxa-9-azaspiro[4.5]decane —— C16H21N3OS
(5R)-9-[[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl]-2-oxa-9-azaspiro[4.5]decane
—— (5-methyl-1H-pyrazol-3-yl)-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C17H20N6OS
(5-methyl-1H-pyrazol-3-yl)-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— 5-ethyl-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]-1,3,4-oxadiazol-2-amine —— C13H18N6O
5-ethyl-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]-1,3,4-oxadiazol-2-amine
—— 5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[(2R)-4-phenylbutan-2-yl]furan-2-carboxamide —— C26H31FN2O2
5-[[(3-fluorophenyl)methyl-propan-2-ylamino]methyl]-N-[(2R)-4-phenylbutan-2-yl]furan-2-carboxamide
—— 5-[3-(3-fluorophenyl)pyrazol-4-ylidene]-3-(methylsulfanylmethyl)-2H-1,2,4-oxadiazole —— C13H11FN4OS
5-[3-(3-fluorophenyl)pyrazol-4-ylidene]-3-(methylsulfanylmethyl)-2H-1,2,4-oxadiazole
—— (5-methyl-1H-pyrazol-3-yl)-[(3S)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C17H20N6OS
(5-methyl-1H-pyrazol-3-yl)-[(3S)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— 5-ethyl-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]-1,3,4-oxadiazol-2-amine —— C13H18N6O
5-ethyl-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]-1,3,4-oxadiazol-2-amine
—— (5-methyl-1,2-oxazol-3-yl)-[(3S)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C17H19N5O2S
(5-methyl-1,2-oxazol-3-yl)-[(3S)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— 5-methyl-N-[3-[3-[(2S)-2-methylpiperidin-1-yl]propylamino]-3-oxopropyl]-N-propylpyrazine-2-carboxamide —— C21H35N5O2
5-methyl-N-[3-[3-[(2S)-2-methylpiperidin-1-yl]propylamino]-3-oxopropyl]-N-propylpyrazine-2-carboxamide
—— (5R)-N-[(1S)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H19FN4O3
(5R)-N-[(1S)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-[4-(aminomethyl)piperidin-1-yl]-2-[2-[(2S)-1-methylpiperidin-2-yl]ethyl]pyridazin-3-one —— C18H31N5O
5-[4-(aminomethyl)piperidin-1-yl]-2-[2-[(2S)-1-methylpiperidin-2-yl]ethyl]pyridazin-3-one
—— (5-methyl-1,2-oxazol-3-yl)-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C17H19N5O2S
(5-methyl-1,2-oxazol-3-yl)-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5S)-N-[(1S)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H19FN4O3
(5S)-N-[(1S)-1-[4-(carbamoylamino)phenyl]ethyl]-3-(3-fluorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— (5R,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H22N2O3
(5R,10bS)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(3-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-methyl-N-[3-[3-[(2R)-2-methylpiperidin-1-yl]propylamino]-3-oxopropyl]-N-propylpyrazine-2-carboxamide —— C21H35N5O2
5-methyl-N-[3-[3-[(2R)-2-methylpiperidin-1-yl]propylamino]-3-oxopropyl]-N-propylpyrazine-2-carboxamide
—— 5-chloro-6-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]pyridine-3-carboxylic acid —— C17H24ClN3O3
5-chloro-6-[4-[(1S)-1-morpholin-4-ylethyl]piperidin-1-yl]pyridine-3-carboxylic acid
—— 5-[4-(aminomethyl)piperidin-1-yl]-2-[2-[(2R)-1-methylpiperidin-2-yl]ethyl]pyridazin-3-one —— C18H31N5O
5-[4-(aminomethyl)piperidin-1-yl]-2-[2-[(2R)-1-methylpiperidin-2-yl]ethyl]pyridazin-3-one
—— 5-[1-(3,5-Dimethoxybenzoyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C21H21N3O4
5-[1-(3,5-Dimethoxybenzoyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-ethyl-4-[(3R)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-6-methylpyrimidin-2-amine —— C17H26N6O2
5-ethyl-4-[(3R)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-6-methylpyrimidin-2-amine
—— 5-chloro-6-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]pyridine-3-carboxylic acid —— C17H24ClN3O3
5-chloro-6-[4-[(1R)-1-morpholin-4-ylethyl]piperidin-1-yl]pyridine-3-carboxylic acid
—— 5-methyl-N-[3-(3-methylbutylamino)-3-oxopropyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrazine-2-carboxamide —— C19H30N4O3
5-methyl-N-[3-(3-methylbutylamino)-3-oxopropyl]-N-[[(2R)-oxolan-2-yl]methyl]pyrazine-2-carboxamide
—— (5S,7R)-3-[5-chloro-4-(furan-2-ylmethylamino)-6-oxopyridazin-1-yl]adamantane-1-carboxylate —— C20H21ClN3O4-
(5S,7R)-3-[5-chloro-4-(furan-2-ylmethylamino)-6-oxopyridazin-1-yl]adamantane-1-carboxylate
—— (5R)-7-(3-methoxypropyl)-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C22H29N3O2
(5R)-7-(3-methoxypropyl)-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-4-[(3S)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-6-methylpyrimidin-2-amine —— C17H26N6O2
5-ethyl-4-[(3S)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-6-methylpyrimidin-2-amine
—— (5S)-2-(2H-benzotriazole-5-carbonyl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5S)-2-(2H-benzotriazole-5-carbonyl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C17H18N6O2S
5-[(3R)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-Benzyl-2-{[(4-bromophenyl)methyl]sulfanyl}-3,6-dimethyl-3,4-dihydropyrimidin-4-one —— C20H19BrN2OS
5-Benzyl-2-{[(4-bromophenyl)methyl]sulfanyl}-3,6-dimethyl-3,4-dihydropyrimidin-4-one
—— [5-[[[(2R)-butan-2-yl]-[(2R)-2-ethylhexanoyl]amino]methyl]-2-methoxyphenyl] methanesulfonate —— C21H35NO5S
[5-[[[(2R)-butan-2-yl]-[(2R)-2-ethylhexanoyl]amino]methyl]-2-methoxyphenyl] methanesulfonate
—— (5S,7R)-3-[5-chloro-4-(cycloheptylamino)-6-oxopyridazin-1-yl]adamantane-1-carboxylate —— C22H29ClN3O3-
(5S,7R)-3-[5-chloro-4-(cycloheptylamino)-6-oxopyridazin-1-yl]adamantane-1-carboxylate
—— 5-[[benzyl-[(4-methoxyphenyl)methyl]amino]methyl]-N-[(2S)-3-methylbutan-2-yl]furan-2-carboxamide —— C26H32N2O3
5-[[benzyl-[(4-methoxyphenyl)methyl]amino]methyl]-N-[(2S)-3-methylbutan-2-yl]furan-2-carboxamide
—— (5S,7R)-3-[5-chloro-4-(4-fluoroanilino)-6-oxopyridazin-1-yl]adamantane-1-carboxylic acid —— C21H21ClFN3O3
(5S,7R)-3-[5-chloro-4-(4-fluoroanilino)-6-oxopyridazin-1-yl]adamantane-1-carboxylic acid
—— (5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(1,3-benzothiazol-2-yl)benzoate —— C23H15N3O3S
(5-Phenyl-1,3,4-oxadiazol-2-yl)methyl 2-(1,3-benzothiazol-2-yl)benzoate
—— (5R)-2-(2H-benzotriazole-5-carbonyl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5R)-2-(2H-benzotriazole-5-carbonyl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-(4-methylpiperazine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H32N4O2
(5R)-7-(cyclobutylmethyl)-2-(4-methylpiperazine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(3-methoxypropyl)-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C22H29N3O2
(5S)-7-(3-methoxypropyl)-2-(2-methylquinolin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-ethyl-1,2-oxazol-3-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H23N7O2
(5-ethyl-1,2-oxazol-3-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— 5-[(2Z)-2-[1-(4-bromophenyl)ethylidene]hydrazinyl]-2-chlorobenzoate —— C15H11BrClN2O2-
5-[(2Z)-2-[1-(4-bromophenyl)ethylidene]hydrazinyl]-2-chlorobenzoate
—— 5-[(3S)-3-(1-butylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyridin-2-one —— C18H24N4O2
5-[(3S)-3-(1-butylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5-[(2Z)-2-[1-(1,3-benzodioxol-5-yl)ethylidene]hydrazinyl]-2-chlorobenzoate —— C16H12ClN2O4-
5-[(2Z)-2-[1-(1,3-benzodioxol-5-yl)ethylidene]hydrazinyl]-2-chlorobenzoate
—— 5-[(3R)-3-(1-butylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyridin-2-one —— C18H24N4O2
5-[(3R)-3-(1-butylimidazol-2-yl)piperidine-1-carbonyl]-1H-pyridin-2-one
—— 5,7-dimethyl-N-[(3R)-1-propylpyrrolidin-3-yl]pyrido[2,3-d]pyrimidin-4-amine —— C16H23N5
5,7-dimethyl-N-[(3R)-1-propylpyrrolidin-3-yl]pyrido[2,3-d]pyrimidin-4-amine
—— (5R)-2-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C22H29N3O3
(5R)-2-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-pyrrolidin-1-yl-2-[[(3R)-pyrrolidin-3-yl]methyl]pyridazin-3-one —— C13H20N4O
5-pyrrolidin-1-yl-2-[[(3R)-pyrrolidin-3-yl]methyl]pyridazin-3-one
—— 5-[(3S)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C17H18N6O2S
5-[(3S)-3-[1-(1,3-thiazol-4-ylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-pyrrolidin-1-yl-2-[[(3S)-pyrrolidin-3-yl]methyl]pyridazin-3-one —— C13H20N4O
5-pyrrolidin-1-yl-2-[[(3S)-pyrrolidin-3-yl]methyl]pyridazin-3-one