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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-7-(2-hydroxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H26N4O3
(5R)-7-(2-hydroxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R,7S)-5-(2-chlorophenyl)-7-(4-phenylmethoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C24H21ClN4O
(5R,7S)-5-(2-chlorophenyl)-7-(4-phenylmethoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-[[(2R)-2-cyclopropyl-2-(dimethylamino)ethyl]amino]pyridine-2-carbonitrile —— C13H18N4
5-[[(2R)-2-cyclopropyl-2-(dimethylamino)ethyl]amino]pyridine-2-carbonitrile
—— (5R)-2-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H26N4O2
(5R)-2-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[5-[(2S)-oxolan-2-yl]thiophen-2-yl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C14H12N4O2S
5-[5-[(2S)-oxolan-2-yl]thiophen-2-yl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— (5S)-5-(2,4-dimethylanilino)-3-phenyl-1,3-thiazolidine-2,4-dione —— C17H16N2O2S
(5S)-5-(2,4-dimethylanilino)-3-phenyl-1,3-thiazolidine-2,4-dione
—— (5S)-1-(4-chlorophenyl)-4-(3,5-difluoropyridine-2-carbonyl)-5-methylpiperazin-2-one —— C17H14ClF2N3O2
(5S)-1-(4-chlorophenyl)-4-(3,5-difluoropyridine-2-carbonyl)-5-methylpiperazin-2-one
—— (5S)-7-(oxan-4-yl)-2-(6-oxo-1H-pyrazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O4
(5S)-7-(oxan-4-yl)-2-(6-oxo-1H-pyrazine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(3,5-dimethyl-1-propylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H27N3O2
(5R)-9-[(3,5-dimethyl-1-propylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-1-[[1-(hydroxymethyl)cyclobutyl]methyl]-5-methyl-5-phenylpiperidin-2-one —— C18H25NO2
(5R)-1-[[1-(hydroxymethyl)cyclobutyl]methyl]-5-methyl-5-phenylpiperidin-2-one
—— 5-[5-[(2R)-oxolan-2-yl]thiophen-2-yl]-3-pyridazin-3-yl-1,2,4-oxadiazole —— C14H12N4O2S
5-[5-[(2R)-oxolan-2-yl]thiophen-2-yl]-3-pyridazin-3-yl-1,2,4-oxadiazole
—— 5-[methyl-[(1R)-1-pyridin-2-ylethyl]amino]pyridine-2-carbonitrile —— C14H14N4
5-[methyl-[(1R)-1-pyridin-2-ylethyl]amino]pyridine-2-carbonitrile
—— (5R)-7-propan-2-yl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H29N3O2
(5R)-7-propan-2-yl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2-oxo-6-phenyl-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H21N3O3
(5S)-2-(2-oxo-6-phenyl-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-(3-phenylpropyl)-5-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl)piperidin-2-one —— C21H26N4O2
(5S)-1-(3-phenylpropyl)-5-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl)piperidin-2-one
—— 5-[methyl-[(1S)-1-pyridin-2-ylethyl]amino]pyridine-2-carbonitrile —— C14H14N4
5-[methyl-[(1S)-1-pyridin-2-ylethyl]amino]pyridine-2-carbonitrile
—— (5S)-6-oxo-N-(2-thiophen-2-ylethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide —— C15H21N3O2S
(5S)-6-oxo-N-(2-thiophen-2-ylethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-2-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H26N4O2
(5S)-2-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclopropylmethyl)-2-[2-(1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O2
(5R)-7-(cyclopropylmethyl)-2-[2-(1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2,4-Dichlorophenyl)-7-(4-methoxyphenyl)-4H,5H,6H,7H-[1,2,4]triazolo[1,5-A]pyrimidin-2-amine —— C18H17Cl2N5O
5-(2,4-Dichlorophenyl)-7-(4-methoxyphenyl)-4H,5H,6H,7H-[1,2,4]triazolo[1,5-A]pyrimidin-2-amine
—— (5S)-7-(2-hydroxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H26N4O3
(5S)-7-(2-hydroxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-chlorophenyl)-N-[(2R)-1-pyridin-2-ylpropan-2-yl]furan-2-carboxamide —— C19H17ClN2O2
5-(2-chlorophenyl)-N-[(2R)-1-pyridin-2-ylpropan-2-yl]furan-2-carboxamide
—— (5R)-6-oxo-N-(2-thiophen-2-ylethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide —— C15H21N3O2S
(5R)-6-oxo-N-(2-thiophen-2-ylethyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-7-(cyclobutylmethyl)-2-(3-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O
(5S)-7-(cyclobutylmethyl)-2-(3-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(6-morpholin-4-ylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23N5O2
(5R)-2-(6-morpholin-4-ylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(3-pyridin-3-yl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H21N5O2
(5S)-9-[2-(3-pyridin-3-yl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-1-(3-phenylpropyl)-5-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl)piperidin-2-one —— C21H26N4O2
(5R)-1-(3-phenylpropyl)-5-(1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-5-carbonyl)piperidin-2-one
—— 5-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile —— C18H19N3OS
5-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]pyridine-2-carbonitrile
—— (5S,7S)-7-(3-chlorophenyl)-5-(4-methoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine —— C18H18ClN5O
(5S,7S)-7-(3-chlorophenyl)-5-(4-methoxyphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine
—— (5S)-1-[[1-(hydroxymethyl)cyclobutyl]methyl]-5-methyl-5-phenylpiperidin-2-one —— C18H25NO2
(5S)-1-[[1-(hydroxymethyl)cyclobutyl]methyl]-5-methyl-5-phenylpiperidin-2-one
—— (5S)-9-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H22N2O2S
(5S)-9-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-9-[2-(3-pyridin-3-yl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H21N5O2
(5R)-9-[2-(3-pyridin-3-yl-1H-1,2,4-triazol-5-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-(2-chlorophenyl)-N-[(2S)-1-pyridin-2-ylpropan-2-yl]furan-2-carboxamide —— C19H17ClN2O2
5-(2-chlorophenyl)-N-[(2S)-1-pyridin-2-ylpropan-2-yl]furan-2-carboxamide
—— (5S)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one —— C21H26N4O3
(5S)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
—— (5R)-7-(cyclobutylmethyl)-2-(3-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O
(5R)-7-(cyclobutylmethyl)-2-(3-methylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3R)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methyl]-2-methoxybenzoic acid —— C21H25NO4
5-[[(3R)-3-[[4-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methyl]-2-methoxybenzoic acid
—— 5-(2-chlorophenyl)-N-[(2R)-2-hydroxy-2-pyridin-2-ylethyl]furan-2-carboxamide —— C18H15ClN2O3
5-(2-chlorophenyl)-N-[(2R)-2-hydroxy-2-pyridin-2-ylethyl]furan-2-carboxamide
—— (5R)-2-(2-oxo-6-phenyl-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H21N3O3
(5R)-2-(2-oxo-6-phenyl-1H-pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5Z)-5-(2,3-dimethoxybenzylidene)-3-phenyl-2-thioxoimidazolidin-4-one —— C18H16N2O3S
(5Z)-5-(2,3-dimethoxybenzylidene)-3-phenyl-2-thioxoimidazolidin-4-one
—— (5S)-7-(cyclopropylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2
(5S)-7-(cyclopropylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one —— C21H26N4O3
(5R)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
—— (5R)-7-(cyclopropylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2
(5R)-7-(cyclopropylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,7S)-5-(4-bromophenyl)-7-(3-methylphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine —— C18H18BrN5
(5S,7S)-5-(4-bromophenyl)-7-(3-methylphenyl)-4,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine
—— 5-(2-chlorophenyl)-N-[(2S)-2-hydroxy-2-pyridin-2-ylethyl]furan-2-carboxamide —— C18H15ClN2O3
5-(2-chlorophenyl)-N-[(2S)-2-hydroxy-2-pyridin-2-ylethyl]furan-2-carboxamide
—— (5S)-2-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3
(5S)-2-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H22N2O2S
(5R)-9-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-[2-[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione —— C20H23N3O5
5-[2-[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl]-1H-pyrimidine-2,4-dione
—— (5R)-1-cyclopentyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C19H21N5O2
(5R)-1-cyclopentyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-7-(oxan-4-yl)-2-(2H-triazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H25N5O2
(5S)-7-(oxan-4-yl)-2-(2H-triazol-4-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-cyclopentyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C19H21N5O2
(5S)-1-cyclopentyl-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one