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—— (5S)-5-(2-chlorophenyl)-3-(3,5-dichloro-2-ethoxyphenyl)-4,5-dihydro-1H-pyrazole —— C17H15Cl3N2O
(5S)-5-(2-chlorophenyl)-3-(3,5-dichloro-2-ethoxyphenyl)-4,5-dihydro-1H-pyrazole
—— 5-fluoro-4-N,4-N-dimethyl-2-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine —— C9H13FN8
5-fluoro-4-N,4-N-dimethyl-2-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine
—— 5-[[[(2S)-2-(2-ethylbenzimidazol-1-yl)butanoyl]amino]methyl]-N-methylfuran-2-carboxamide —— C20H24N4O3
5-[[[(2S)-2-(2-ethylbenzimidazol-1-yl)butanoyl]amino]methyl]-N-methylfuran-2-carboxamide
—— 5-[(3S)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoate —— C21H21N2O4-
5-[(3S)-3-(2-hydroxyphenyl)-5-(4-methylphenyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoate
—— (5S)-9-(5-fluoro-4-pyrrolidin-1-ylpyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H25FN4O2
(5S)-9-(5-fluoro-4-pyrrolidin-1-ylpyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5Z)-5-[(3,4-dichlorophenyl)methylidene]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one —— C16H16Cl2N2O2S
(5Z)-5-[(3,4-dichlorophenyl)methylidene]-2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-1,3-thiazol-4-one
—— 5-[(3R)-1-ethyl-5-oxopyrrolidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C16H21N3O3S
5-[(3R)-1-ethyl-5-oxopyrrolidine-3-carbonyl]-N-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— 5-[(3S)-3-(2-hydroxy-3-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid —— C19H20N2O5S
5-[(3S)-3-(2-hydroxy-3-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid
—— 5-Amino-N-(3,5-dimethylphenyl)-1-{[(3,4-dimethylphenyl)carbamoyl]methyl}-1H-1,2,3-triazole-4-carboxamide —— C21H24N6O2
5-Amino-N-(3,5-dimethylphenyl)-1-{[(3,4-dimethylphenyl)carbamoyl]methyl}-1H-1,2,3-triazole-4-carboxamide
—— (5R)-9-(5-fluoro-4-pyrrolidin-1-ylpyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H25FN4O2
(5R)-9-(5-fluoro-4-pyrrolidin-1-ylpyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-9-[[2-(2-imidazol-1-ylethoxy)-3-methoxyphenyl]methyl]-2-oxa-9-azaspiro[4.5]decane —— C21H29N3O3
(5R)-9-[[2-(2-imidazol-1-ylethoxy)-3-methoxyphenyl]methyl]-2-oxa-9-azaspiro[4.5]decane
—— 5-fluoro-4-N,4-N-dimethyl-2-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine —— C9H13FN8
5-fluoro-4-N,4-N-dimethyl-2-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine
—— (5R)-2-(1-benzoxepine-4-carbonyl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one —— C24H28N2O3
(5R)-2-(1-benzoxepine-4-carbonyl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[[2-(2-imidazol-1-ylethoxy)-3-methoxyphenyl]methyl]-2-oxa-9-azaspiro[4.5]decane —— C21H29N3O3
(5S)-9-[[2-(2-imidazol-1-ylethoxy)-3-methoxyphenyl]methyl]-2-oxa-9-azaspiro[4.5]decane
—— [5-(methylsulfanylmethyl)furan-2-yl]-[(3S)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone —— C18H25N3O2S
[5-(methylsulfanylmethyl)furan-2-yl]-[(3S)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone
—— (5S)-2-(5-chloropyridin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C16H22ClN3O
(5S)-2-(5-chloropyridin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-1-[2-[3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C16H24N4O3
5-methyl-1-[2-[3-[(2R)-2-methylpiperidin-1-yl]azetidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— (5R)-2-(5-chloropyridin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C16H22ClN3O
(5R)-2-(5-chloropyridin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C19H24N4O3
(5R)-7-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-ethyl-N-[(2R)-2-morpholin-4-ylbutyl]pyrimidin-2-amine —— C14H24N4O
5-ethyl-N-[(2R)-2-morpholin-4-ylbutyl]pyrimidin-2-amine
—— 5-[benzyl(methyl)amino]-2-[[(3R)-1-propan-2-ylpyrrolidin-3-yl]methyl]pyridazin-3-one —— C20H28N4O
5-[benzyl(methyl)amino]-2-[[(3R)-1-propan-2-ylpyrrolidin-3-yl]methyl]pyridazin-3-one
—— [5-(methylsulfanylmethyl)furan-2-yl]-[(3R)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone —— C18H25N3O2S
[5-(methylsulfanylmethyl)furan-2-yl]-[(3R)-3-(1-propan-2-ylimidazol-2-yl)piperidin-1-yl]methanone
—— 5-methyl-1-[2-[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C16H24N4O3
5-methyl-1-[2-[3-[(2S)-2-methylpiperidin-1-yl]azetidin-1-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— 5-ethyl-N-[(2S)-2-morpholin-4-ylbutyl]pyrimidin-2-amine —— C14H24N4O
5-ethyl-N-[(2S)-2-morpholin-4-ylbutyl]pyrimidin-2-amine
—— 5-tert-butyl-N-[(1S)-1-imidazo[2,1-b][1,3]thiazol-6-ylethyl]-1,3,4-oxadiazol-2-amine —— C13H17N5OS
5-tert-butyl-N-[(1S)-1-imidazo[2,1-b][1,3]thiazol-6-ylethyl]-1,3,4-oxadiazol-2-amine
—— (5S)-7-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C19H24N4O3
(5S)-7-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5R,7S)-N-[(2R)-butan-2-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C16H19F3N4O2
(5R,7S)-N-[(2R)-butan-2-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-tert-butyl-N-[(1R)-1-imidazo[2,1-b][1,3]thiazol-6-ylethyl]-1,3,4-oxadiazol-2-amine —— C13H17N5OS
5-tert-butyl-N-[(1R)-1-imidazo[2,1-b][1,3]thiazol-6-ylethyl]-1,3,4-oxadiazol-2-amine
—— 5-[benzyl(methyl)amino]-2-[[(3S)-1-propan-2-ylpyrrolidin-3-yl]methyl]pyridazin-3-one —— C20H28N4O
5-[benzyl(methyl)amino]-2-[[(3S)-1-propan-2-ylpyrrolidin-3-yl]methyl]pyridazin-3-one
—— 5-[(3R)-3-(2-hydroxy-3-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-5-oxopentanoate —— C19H19N2O5S-
5-[(3R)-3-(2-hydroxy-3-methoxyphenyl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-5-oxopentanoate
—— (5R,7S)-N-butyl-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C16H19F3N4O2
(5R,7S)-N-butyl-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— 5-amino-1-{2-[(3,5-dimethylphenyl)amino]-2-oxoethyl}-N-(4-fluorophenyl)-1H-1,2,3-triazole-4-carboxamide —— C19H19FN6O2
5-amino-1-{2-[(3,5-dimethylphenyl)amino]-2-oxoethyl}-N-(4-fluorophenyl)-1H-1,2,3-triazole-4-carboxamide
—— 5-amino-N-(3-chloro-2-methylphenyl)-1-{2-[(3,5-dimethylphenyl)amino]-2-oxoethyl}-1H-1,2,3-triazole-4-carboxamide —— C20H21ClN6O2
5-amino-N-(3-chloro-2-methylphenyl)-1-{2-[(3,5-dimethylphenyl)amino]-2-oxoethyl}-1H-1,2,3-triazole-4-carboxamide
—— (5R)-5-(4-propan-2-ylphenyl)-2-propan-2-ylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione —— C23H27N3O2S
(5R)-5-(4-propan-2-ylphenyl)-2-propan-2-ylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione
—— (5S)-5-(4-propan-2-ylphenyl)-2-propan-2-ylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione —— C23H27N3O2S
(5S)-5-(4-propan-2-ylphenyl)-2-propan-2-ylsulfanyl-3,5,7,8,9,10-hexahydropyrimido[4,5-b]quinoline-4,6-dione
—— (5R)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-pyridin-3-ylpyrrolidine-2,3-dione —— C21H15N3O6
(5R)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-pyridin-3-ylpyrrolidine-2,3-dione
—— (5S)-3-methyl-7-(4-methylpyrimidin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H16N4O2
(5S)-3-methyl-7-(4-methylpyrimidin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-[3-(3-fluorophenyl)pyrazol-4-ylidene]-3-[(1-methylpiperidin-4-yl)methyl]-2H-1,2,4-oxadiazole —— C18H20FN5O
5-[3-(3-fluorophenyl)pyrazol-4-ylidene]-3-[(1-methylpiperidin-4-yl)methyl]-2H-1,2,4-oxadiazole
—— (5R)-3-methyl-7-(4-methylpyrimidin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C12H16N4O2
(5R)-3-methyl-7-(4-methylpyrimidin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 5-cyclopropyl-N-[(1R)-1-(2-propoxyphenyl)ethyl]-1,3,4-oxadiazol-2-amine —— C16H21N3O2
5-cyclopropyl-N-[(1R)-1-(2-propoxyphenyl)ethyl]-1,3,4-oxadiazol-2-amine
—— (5R)-7-(2-methoxyethyl)-2-(6-methylthieno[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2S
(5R)-7-(2-methoxyethyl)-2-(6-methylthieno[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[4-[(4S)-2,2-dimethyloxan-4-yl]triazol-1-yl]methyl]thiophene-2-carboxylic acid —— C15H19N3O3S
5-[[4-[(4S)-2,2-dimethyloxan-4-yl]triazol-1-yl]methyl]thiophene-2-carboxylic acid
—— 5-ethyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine —— C15H20N4
5-ethyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
—— 5-cyclopropyl-N-[(1S)-1-(2-propoxyphenyl)ethyl]-1,3,4-oxadiazol-2-amine —— C16H21N3O2
5-cyclopropyl-N-[(1S)-1-(2-propoxyphenyl)ethyl]-1,3,4-oxadiazol-2-amine
—— 5,7-dimethyl-4-[(5R)-7-methyl-2,7-diazaspiro[4.4]nonan-2-yl]pyrido[2,3-d]pyrimidine —— C17H23N5
5,7-dimethyl-4-[(5R)-7-methyl-2,7-diazaspiro[4.4]nonan-2-yl]pyrido[2,3-d]pyrimidine
—— (5S)-7-(2-methoxyethyl)-2-(6-methylthieno[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2S
(5S)-7-(2-methoxyethyl)-2-(6-methylthieno[2,3-d]pyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5-Acetyl-2-methoxyphenyl)methyl 5-(phenoxymethyl)furan-2-carboxylate —— C22H20O6
(5-Acetyl-2-methoxyphenyl)methyl 5-(phenoxymethyl)furan-2-carboxylate
—— 5,7-dimethyl-4-[(5S)-7-methyl-2,7-diazaspiro[4.4]nonan-2-yl]pyrido[2,3-d]pyrimidine —— C17H23N5
5,7-dimethyl-4-[(5S)-7-methyl-2,7-diazaspiro[4.4]nonan-2-yl]pyrido[2,3-d]pyrimidine
—— (5R)-2-(3,5-dichloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H21Cl2N3O2
(5R)-2-(3,5-dichloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(3,5-dichloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H21Cl2N3O2
(5S)-2-(3,5-dichloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one