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—— (5S,10bS)-2-(4-chlorophenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H21ClN2O
(5S,10bS)-2-(4-chlorophenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(3S,8aS)-1-oxo-3,5,6,7,8,8a-hexahydro-2H-imidazo[1,5-a]pyridin-3-yl]furan-2-carbonitrile —— C12H13N3O2
5-[(3S,8aS)-1-oxo-3,5,6,7,8,8a-hexahydro-2H-imidazo[1,5-a]pyridin-3-yl]furan-2-carbonitrile
—— 5-[(3R,8aS)-1-oxo-3,5,6,7,8,8a-hexahydro-2H-imidazo[1,5-a]pyridin-3-yl]furan-2-carbonitrile —— C12H13N3O2
5-[(3R,8aS)-1-oxo-3,5,6,7,8,8a-hexahydro-2H-imidazo[1,5-a]pyridin-3-yl]furan-2-carbonitrile
—— 5-methyl-2-[(3S)-oxan-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one —— C12H14N2O2S
5-methyl-2-[(3S)-oxan-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one
—— 5-(3-morpholin-4-ium-4-ylpropyliminomethyl)-6-oxo-2-sulfanylidene-5H-pyrimidin-4-olate —— C12H18N4O3S
5-(3-morpholin-4-ium-4-ylpropyliminomethyl)-6-oxo-2-sulfanylidene-5H-pyrimidin-4-olate
—— (5S)-4-amino-3-(2-morpholin-4-ium-4-ylethyl)-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol —— C23H26N4O3+2
(5S)-4-amino-3-(2-morpholin-4-ium-4-ylethyl)-5-phenyl-5H-chromeno[2,3-d]pyrimidin-3-ium-8-ol
—— 5-chloro-N-[2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl]thiophene-2-sulfonamide —— C15H12ClFN2O2S3
5-chloro-N-[2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]ethyl]thiophene-2-sulfonamide
—— (5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H18N2O3
(5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(3R,8aR)-1-oxo-3,5,6,7,8,8a-hexahydro-2H-imidazo[1,5-a]pyridin-3-yl]furan-2-carbonitrile —— C12H13N3O2
5-[(3R,8aR)-1-oxo-3,5,6,7,8,8a-hexahydro-2H-imidazo[1,5-a]pyridin-3-yl]furan-2-carbonitrile
—— (5R)-5-(cyclopropyliminomethyl)-1-[(4-fluorophenyl)methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C15H14FN3O2S
(5R)-5-(cyclopropyliminomethyl)-1-[(4-fluorophenyl)methyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-bromo-N-[[(3R)-oxolan-3-yl]methyl]pyridin-3-amine —— C10H13BrN2O
5-bromo-N-[[(3R)-oxolan-3-yl]methyl]pyridin-3-amine
—— (5S,10bR)-2-(3-bromophenyl)-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C21H16BrN3O
(5S,10bR)-2-(3-bromophenyl)-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-nitro-4-N-[[(2R)-oxolan-2-yl]methyl]-2-N-prop-2-enylpyrimidine-2,4,6-triamine —— C12H18N6O3
5-nitro-4-N-[[(2R)-oxolan-2-yl]methyl]-2-N-prop-2-enylpyrimidine-2,4,6-triamine
—— 5-[2-[(1R,4S)-2-azabicyclo[2.2.1]heptan-2-yl]pyridin-4-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C16H20N4O
5-[2-[(1R,4S)-2-azabicyclo[2.2.1]heptan-2-yl]pyridin-4-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(1R,5S)-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-3-yl]-3-methyl-1,2,4-thiadiazole —— C10H15N3S
5-[(1R,5S)-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-3-yl]-3-methyl-1,2,4-thiadiazole
—— 5-[2-[(3R)-3-(1,3-dioxolan-2-yl)piperidin-1-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole —— C16H20N4O3
5-[2-[(3R)-3-(1,3-dioxolan-2-yl)piperidin-1-yl]pyridin-3-yl]-3-methyl-1,2,4-oxadiazole
—— 5-bromo-N-[[(3S)-oxolan-3-yl]methyl]pyridin-3-amine —— C10H13BrN2O
5-bromo-N-[[(3S)-oxolan-3-yl]methyl]pyridin-3-amine
—— (5S,10bS)-2-(4-methylphenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H22N2OS
(5S,10bS)-2-(4-methylphenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-bromo-N-[[(3S)-1-methylpiperidin-3-yl]methyl]pyridine-2-sulfonamide —— C12H18BrN3O2S
5-bromo-N-[[(3S)-1-methylpiperidin-3-yl]methyl]pyridine-2-sulfonamide
—— [5-(methoxymethyl)-1,2-oxazol-3-yl]-[(3S)-3-[(2-methoxyphenyl)methyl]piperidin-1-yl]methanone —— C19H24N2O4
[5-(methoxymethyl)-1,2-oxazol-3-yl]-[(3S)-3-[(2-methoxyphenyl)methyl]piperidin-1-yl]methanone
—— 5-methyl-2-[(3R)-oxan-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one —— C12H14N2O2S
5-methyl-2-[(3R)-oxan-3-yl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (5S,10bS)-2-(4-methoxyphenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H22N2O2S
(5S,10bS)-2-(4-methoxyphenyl)-5-(2-methylsulfanylethyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-5-(2-methylsulfanylethyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C17H18N2OS2
(5R,10bS)-5-(2-methylsulfanylethyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(3S)-1-[(2S)-1-oxo-1-[[(2S)-oxolan-2-yl]methylamino]propan-2-yl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H27N5O3
5-[(3S)-1-[(2S)-1-oxo-1-[[(2S)-oxolan-2-yl]methylamino]propan-2-yl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-chloro-4-[(1R,5S)-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-3-yl]-1H-pyridazin-6-one —— C11H14ClN3O
5-chloro-4-[(1R,5S)-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-3-yl]-1H-pyridazin-6-one
—— (5S)-3-ethyl-5-methyl-5-[(3S)-1-(2-pyridin-4-ylethyl)piperidin-3-yl]imidazolidine-2,4-dione —— C18H26N4O2
(5S)-3-ethyl-5-methyl-5-[(3S)-1-(2-pyridin-4-ylethyl)piperidin-3-yl]imidazolidine-2,4-dione
—— 5-[(3S)-1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C15H18N4O2S
5-[(3S)-1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-(4-methyl-3-methylsulfonylbenzoyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C18H22N4O4S
5-[(3R)-1-(4-methyl-3-methylsulfonylbenzoyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-[(5-methylpyrazin-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C15H20N6O
5-[(3R)-1-[(5-methylpyrazin-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-[(2R)-2-[(4-methoxybenzoyl)amino]-3-methylbutanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C22H29N5O4
5-[(3R)-1-[(2R)-2-[(4-methoxybenzoyl)amino]-3-methylbutanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-chloro-2-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]sulfonylbenzonitrile —— C19H22ClN5O2S
5-chloro-2-[(3S)-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)piperidin-1-yl]sulfonylbenzonitrile
—— 5-[(3S)-1-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C14H20N6O2S
5-[(3S)-1-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-(2-methylsulfonylethyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C12H20N4O3S
5-[(3R)-1-(2-methylsulfonylethyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-[(2S)-1-oxo-1-[[(2R)-oxolan-2-yl]methylamino]propan-2-yl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H27N5O3
5-[(3S)-1-[(2S)-1-oxo-1-[[(2R)-oxolan-2-yl]methylamino]propan-2-yl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-[4-(1,3-dioxoisoindol-2-yl)butanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C21H23N5O4
5-[(3R)-1-[4-(1,3-dioxoisoindol-2-yl)butanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-[(2S)-2-(2-chlorophenyl)sulfanylpropanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C18H21ClN4O2S
5-[(3S)-1-[(2S)-2-(2-chlorophenyl)sulfanylpropanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5R,10bS)-7-ethoxy-2-(4-methylphenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H28N2O2
(5R,10bS)-7-ethoxy-2-(4-methylphenyl)-5-(2-methylpropyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-bromo-N-[[(3R)-1-methylpiperidin-3-yl]methyl]pyridine-2-sulfonamide —— C12H18BrN3O2S
5-bromo-N-[[(3R)-1-methylpiperidin-3-yl]methyl]pyridine-2-sulfonamide
—— 5-[(3R)-1-[3-[(3-chlorophenyl)sulfonylamino]propanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C18H22ClN5O4S
5-[(3R)-1-[3-[(3-chlorophenyl)sulfonylamino]propanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C15H21N5OS
5-[(3S)-1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-[(2R)-2-(2-chlorophenyl)sulfanylpropanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C18H21ClN4O2S
5-[(3R)-1-[(2R)-2-(2-chlorophenyl)sulfanylpropanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-[2-oxo-2-(pyridin-3-ylmethylamino)ethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C17H22N6O2
5-[(3S)-1-[2-oxo-2-(pyridin-3-ylmethylamino)ethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3R)-1-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C14H20N6O2S
5-[(3R)-1-[(5-ethoxy-1,3,4-thiadiazol-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-[(1R)-1-pyridin-3-ylethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C16H21N5O
5-[(3S)-1-[(1R)-1-pyridin-3-ylethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H20N2O4
(5S,10bS)-2-(1,3-benzodioxol-5-yl)-5-(3-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-[(3S)-1-[(5-methylpyrazin-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C15H20N6O
5-[(3S)-1-[(5-methylpyrazin-2-yl)methyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C13H18N6O
5-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— 5-[(3S)-1-[(2S)-2-[(4-methoxybenzoyl)amino]-3-methylbutanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C22H29N5O4
5-[(3S)-1-[(2S)-2-[(4-methoxybenzoyl)amino]-3-methylbutanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5R)-5-(4-hydroxyphenyl)-4-[hydroxy-(4-prop-2-enoxyphenyl)methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione —— C23H23NO6
(5R)-5-(4-hydroxyphenyl)-4-[hydroxy-(4-prop-2-enoxyphenyl)methylidene]-1-(2-methoxyethyl)pyrrolidine-2,3-dione
—— 5-[(3R)-1-[(2S)-2-[(4-methoxybenzoyl)amino]-3-methylbutanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C22H29N5O4
5-[(3R)-1-[(2S)-2-[(4-methoxybenzoyl)amino]-3-methylbutanoyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide