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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5S)-9-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H18N2O4
(5S)-9-[[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4OS
(5S)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R,7R)-5-(4-bromophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H20BrF3N4O2
(5R,7R)-5-(4-bromophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-3-bromo-N-[(6S)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C25H25BrF3N5O3S
(5R,7R)-3-bromo-N-[(6S)-3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-5-(4-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,10bR)-9-bromo-2-phenyl-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C21H16BrN3O
(5S,10bR)-9-bromo-2-phenyl-5-pyridin-4-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-pyridin-2-yl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C19H15N3OS
(5S,10bS)-5-pyridin-2-yl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,7S)-5-(4-bromophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H20BrF3N4O2
(5R,7S)-5-(4-bromophenyl)-N-[[(2S)-oxolan-2-yl]methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S)-2-[(5-acetylthiophen-3-yl)methyl]-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2S
(5S)-2-[(5-acetylthiophen-3-yl)methyl]-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-3-oxo-N,5-diphenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C20H17N3O2S
(5R)-7-methyl-3-oxo-N,5-diphenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-7-propyl-2-[6-(1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H24N6O2
(5R)-7-propyl-2-[6-(1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-methyl-2-phenylfuran-3-yl)-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C21H23N3O3
(5-methyl-2-phenylfuran-3-yl)-[(2R)-2-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (5S)-1-[(2,4-dimethoxyphenyl)methyl]-5-methyl-5-phenylpiperidin-2-one —— C21H25NO3
(5S)-1-[(2,4-dimethoxyphenyl)methyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-7-methyl-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C14H22N4O2S
(5R)-7-methyl-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(4-methoxy-3-prop-2-enylbenzoyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H26N2O3
(5R)-2-(4-methoxy-3-prop-2-enylbenzoyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-propan-2-yl-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H24N4O
(5R)-7-propan-2-yl-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C16H21F3N2O2
(5S)-9-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-9-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C16H21F3N2O2
(5R)-9-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-N-(5,6-dimethylpyrimidin-4-yl)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-amine —— C20H28N6O
(5R)-N-(5,6-dimethylpyrimidin-4-yl)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-amine
—— (5R)-2-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H28N2O2
(5R)-2-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2-ethyl-6-oxo-1H-pyridine-4-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O4
(5S)-2-(2-ethyl-6-oxo-1H-pyridine-4-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-[(2,4-dimethoxyphenyl)methyl]-5-methyl-5-phenylpiperidin-2-one —— C21H25NO3
(5R)-1-[(2,4-dimethoxyphenyl)methyl]-5-methyl-5-phenylpiperidin-2-one
—— (5S)-5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-cyclopentylpiperidin-2-one —— C20H25ClN2O3
(5S)-5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-cyclopentylpiperidin-2-one
—— (5S)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O
(5S)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— [(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(3-pyridin-3-ylazetidin-1-yl)methanone —— C18H20N2OS
[(5S)-5-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-(3-pyridin-3-ylazetidin-1-yl)methanone
—— (5R)-2-[(5-acetylthiophen-3-yl)methyl]-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O2S
(5R)-2-[(5-acetylthiophen-3-yl)methyl]-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propan-2-yl-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H24N4O
(5S)-7-propan-2-yl-2-quinoxalin-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-(2,2,2-trifluoroethyl)-1,2-dihydropyrazole-3-carboxamide —— C12H10F3N3O2
5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-(2,2,2-trifluoroethyl)-1,2-dihydropyrazole-3-carboxamide
—— (5S)-N-(5,6-dimethylpyrimidin-4-yl)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-amine —— C20H28N6O
(5S)-N-(5,6-dimethylpyrimidin-4-yl)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-amine
—— (5R)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O
(5R)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one —— C19H25N3O3
(5S)-1-[[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one
—— (5S)-9-[2-[[5-[(dimethylamino)methyl]furan-2-yl]methylsulfanyl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H28N2O3S
(5S)-9-[2-[[5-[(dimethylamino)methyl]furan-2-yl]methylsulfanyl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H24N4O2
(5R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-N-[(2R)-2-methoxy-2-thiophen-2-ylethyl]-1,3,4-oxadiazol-2-amine —— C11H15N3O2S
5-ethyl-N-[(2R)-2-methoxy-2-thiophen-2-ylethyl]-1,3,4-oxadiazol-2-amine
—— (5S)-2-(4-methyl-3-oxo-1,2-dihydropyrazolo[3,4-b]pyridine-6-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H25N5O3
(5S)-2-(4-methyl-3-oxo-1,2-dihydropyrazolo[3,4-b]pyridine-6-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-N-[(2S)-2-methoxy-2-thiophen-2-ylethyl]-1,3,4-oxadiazol-2-amine —— C11H15N3O2S
5-ethyl-N-[(2S)-2-methoxy-2-thiophen-2-ylethyl]-1,3,4-oxadiazol-2-amine
—— (5R)-7-(cyclobutylmethyl)-2-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C23H29N3O2
(5R)-7-(cyclobutylmethyl)-2-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-methyl-5-phenyl-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl)piperidin-2-one —— C19H24N4O
(5R)-5-methyl-5-phenyl-1-(5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl)piperidin-2-one
—— (5S)-7-methyl-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C14H22N4O2S
(5S)-7-methyl-2-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-3-ylmethyl)-1,2-dihydropyrazole-3-carboxamide —— C20H21N3O3S
5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[[(2R)-oxolan-2-yl]methyl]-N-(thiophen-3-ylmethyl)-1,2-dihydropyrazole-3-carboxamide
—— (5R)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O3
(5R)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-1-[[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one —— C19H25N3O3
(5R)-1-[[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one
—— (5R)-2-(4-methyl-3-oxo-1,2-dihydropyrazolo[3,4-b]pyridine-6-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H25N5O3
(5R)-2-(4-methyl-3-oxo-1,2-dihydropyrazolo[3,4-b]pyridine-6-carbonyl)-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(cyclobutylmethyl)-2-(2-thiophen-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N2O2S
(5S)-7-(cyclobutylmethyl)-2-(2-thiophen-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-(2-hydroxyethyl)-2-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H24N4O4
(5S)-7-(2-hydroxyethyl)-2-[5-(imidazol-1-ylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-methoxyfuran-2-yl)-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C20H22N4O3
(5-methoxyfuran-2-yl)-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5R)-N,5-dimethyl-N-[2-(1-methylpyrazol-4-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C17H23N3OS
(5R)-N,5-dimethyl-N-[2-(1-methylpyrazol-4-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5S)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C19H28N4O3
(5S)-2-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5-methoxy-1-methylindol-2-yl)-[(2R)-2-pyridin-3-ylpiperidin-1-yl]methanone —— C21H23N3O2
(5-methoxy-1-methylindol-2-yl)-[(2R)-2-pyridin-3-ylpiperidin-1-yl]methanone
—— 5-[(3S)-1-methylpiperidin-3-yl]-3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazole —— C13H17N5O
5-[(3S)-1-methylpiperidin-3-yl]-3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazole
—— (5R)-2-[(2-butyl-4-chloro-1H-imidazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H25ClN4O
(5R)-2-[(2-butyl-4-chloro-1H-imidazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one