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—— (5R)-1-cyclohexyl-5-(3-morpholin-4-ium-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H29N4O3S+
(5R)-1-cyclohexyl-5-(3-morpholin-4-ium-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-1-cyclopropyl-5-(3-morpholin-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C15H22N4O3S
(5R)-1-cyclopropyl-5-(3-morpholin-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[C-ethyl-N-(3-imidazol-1-ylpropyl)carbonimidoyl]-1-phenyl-1,3-diazinane-2,4,6-trione —— C19H21N5O3
5-[C-ethyl-N-(3-imidazol-1-ylpropyl)carbonimidoyl]-1-phenyl-1,3-diazinane-2,4,6-trione
—— (5R)-7-(cyclobutylmethyl)-2-[(2-methyl-7-oxo-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H28N6O2
(5R)-7-(cyclobutylmethyl)-2-[(2-methyl-7-oxo-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[(2S)-butan-2-yl]-5-[2-(diethylamino)ethyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C15H26N4O2S
(5S)-1-[(2S)-butan-2-yl]-5-[2-(diethylamino)ethyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5,6-dimethyl-N-[(1S)-1-(5-methylpyridin-2-yl)propyl]pyrimidin-4-amine —— C15H20N4
5,6-dimethyl-N-[(1S)-1-(5-methylpyridin-2-yl)propyl]pyrimidin-4-amine
—— 5-[N-(3-hydroxypropyl)-C-methylcarbonimidoyl]-1,3-diazinane-2,4,6-trione —— C9H13N3O4
5-[N-(3-hydroxypropyl)-C-methylcarbonimidoyl]-1,3-diazinane-2,4,6-trione
—— (5R)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione —— C20H14N2O6S
(5R)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-thiophen-2-ylpyrrolidine-2,3-dione
—— (5S)-5-(1H-imidazol-5-ylmethyl)-7-(5-methylpyrimidin-2-yl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H24N8O
(5S)-5-(1H-imidazol-5-ylmethyl)-7-(5-methylpyrimidin-2-yl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 5-[(2S)-1-methylazepan-2-yl]-3-[2-(4-methylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole —— C16H29N5O
5-[(2S)-1-methylazepan-2-yl]-3-[2-(4-methylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole
—— (5S)-1-[2-(2-hydroxyethoxy)ethyl]-4-[hydroxy-(3-nitrophenyl)methylidene]-5-pyridin-3-ylpyrrolidine-2,3-dione —— C20H19N3O7
(5S)-1-[2-(2-hydroxyethoxy)ethyl]-4-[hydroxy-(3-nitrophenyl)methylidene]-5-pyridin-3-ylpyrrolidine-2,3-dione
—— (5R)-5-[[(1S,2R)-2-aminocyclohexyl]iminomethyl]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H22N4O2S
(5R)-5-[[(1S,2R)-2-aminocyclohexyl]iminomethyl]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-3-(2,4-dichlorophenyl)-7-(4-methylphenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione —— C19H14Cl2N2O3
(5S)-3-(2,4-dichlorophenyl)-7-(4-methylphenyl)-1-oxa-2,7-diazaspiro[4.4]non-2-ene-6,8-dione
—— (5R)-1-(4-fluorophenyl)-5-(3-morpholin-4-ium-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H22FN4O3S+
(5R)-1-(4-fluorophenyl)-5-(3-morpholin-4-ium-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-2-[(Z)-N-ethoxy-C-propylcarbonimidoyl]-5-[(2S)-2-ethylsulfanylpropyl]-3-hexyliminocyclohexan-1-one —— C23H42N2O2S
(5S)-2-[(Z)-N-ethoxy-C-propylcarbonimidoyl]-5-[(2S)-2-ethylsulfanylpropyl]-3-hexyliminocyclohexan-1-one
—— (5R)-1-butyl-5-(3-morpholin-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C16H26N4O3S
(5R)-1-butyl-5-(3-morpholin-4-ylpropyliminomethyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(3-methoxypropyl)-5-(4-methylphenyl)pyrrolidine-2,3-dione —— C23H25NO4
(5R)-4-[hydroxy-(4-methylphenyl)methylidene]-1-(3-methoxypropyl)-5-(4-methylphenyl)pyrrolidine-2,3-dione
—— 5-cyclohexyl-1-[(1R)-1-phenylethyl]-1,3,5-triazinan-5-ium-2-thione —— C17H26N3S+
5-cyclohexyl-1-[(1R)-1-phenylethyl]-1,3,5-triazinan-5-ium-2-thione
—— 5-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C17H20N8O2
5-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-[[[(2S)-2-(dimethylamino)-2-(3-fluorophenyl)acetyl]amino]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C15H18FN5O3
5-[[[(2S)-2-(dimethylamino)-2-(3-fluorophenyl)acetyl]amino]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— (5R)-1-(4-ethoxyphenyl)-5-(2-fluorophenyl)-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione —— C25H20FNO4
(5R)-1-(4-ethoxyphenyl)-5-(2-fluorophenyl)-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione
—— 5-[(2R)-1-methylazepan-2-yl]-3-[2-(4-methylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole —— C16H29N5O
5-[(2R)-1-methylazepan-2-yl]-3-[2-(4-methylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole
—— (5R)-5-(1H-imidazol-5-ylmethyl)-7-(5-methylpyrimidin-2-yl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C19H24N8O
(5R)-5-(1H-imidazol-5-ylmethyl)-7-(5-methylpyrimidin-2-yl)-3-(oxan-4-yl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— (5R,10bS)-9-chloro-2-(furan-2-yl)-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H15ClN2O2
(5R,10bS)-9-chloro-2-(furan-2-yl)-5-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-5-(1,3-benzodioxol-5-ylmethyliminomethyl)-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H17N3O5S
(5S)-5-(1,3-benzodioxol-5-ylmethyliminomethyl)-1-(2-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-phenylpyrrolidine-2,3-dione —— C22H16N2O6
(5S)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-phenylpyrrolidine-2,3-dione
—— (5R)-2-[(Z)-N-ethoxy-C-propylcarbonimidoyl]-5-[(2R)-2-ethylsulfanylpropyl]-3-hexyliminocyclohexan-1-one —— C23H42N2O2S
(5R)-2-[(Z)-N-ethoxy-C-propylcarbonimidoyl]-5-[(2R)-2-ethylsulfanylpropyl]-3-hexyliminocyclohexan-1-one
—— 5-fluoro-2-N-[(1R)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]-4-N,4-N-dimethylpyrimidine-2,4-diamine —— C13H20FN7O
5-fluoro-2-N-[(1R)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]-4-N,4-N-dimethylpyrimidine-2,4-diamine
—— 5-[[[(2R)-2-(dimethylamino)-2-(3-fluorophenyl)acetyl]amino]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide —— C15H18FN5O3
5-[[[(2R)-2-(dimethylamino)-2-(3-fluorophenyl)acetyl]amino]methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
—— 5-fluoro-2-N-[(1S)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]-4-N,4-N-dimethylpyrimidine-2,4-diamine —— C13H20FN7O
5-fluoro-2-N-[(1S)-1-[4-(2-methoxyethyl)-1,2,4-triazol-3-yl]ethyl]-4-N,4-N-dimethylpyrimidine-2,4-diamine
—— 5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,2-dihydropyrazole-3-carboxamide —— C14H14N6O2S
5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,2-dihydropyrazole-3-carboxamide
—— 5-[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C17H20N8O2
5-[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-phenylpyrrolidine-2,3-dione —— C22H16ClNO4
(5S)-4-[(4-chlorophenyl)-hydroxymethylidene]-1-(furan-2-ylmethyl)-5-phenylpyrrolidine-2,3-dione
—— (5S)-N-[(3-fluorophenyl)methyl]-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide —— C19H26FN3O3
(5S)-N-[(3-fluorophenyl)methyl]-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5R)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H25N3O4
(5R)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-phenylpyrrolidine-2,3-dione —— C22H16N2O6
(5R)-1-(furan-2-ylmethyl)-4-[hydroxy-(3-nitrophenyl)methylidene]-5-phenylpyrrolidine-2,3-dione
—— (5Z)-3-cyclohexyl-5-[(2,4-dimethylanilino)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H22N2OS2
(5Z)-3-cyclohexyl-5-[(2,4-dimethylanilino)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H25N3O4
(5S)-9-[[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-N-[(3-fluorophenyl)methyl]-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide —— C19H26FN3O3
(5R)-N-[(3-fluorophenyl)methyl]-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5E)-5-[(4-ethylanilino)methylidene]-3-(3-methoxypropyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C16H20N2O2S2
(5E)-5-[(4-ethylanilino)methylidene]-3-(3-methoxypropyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-ethyl-4-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2,6-dimethylpyrimidine —— C20H28N8
5-ethyl-4-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2,6-dimethylpyrimidine
—— (5R)-N-(1,3-benzodioxol-5-yl)-2-oxa-9-azaspiro[4.5]decane-9-carboxamide —— C16H20N2O4
(5R)-N-(1,3-benzodioxol-5-yl)-2-oxa-9-azaspiro[4.5]decane-9-carboxamide
—— (5S)-1-[(2R)-butan-2-yl]-5-[[(2R)-oxolan-2-yl]methyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C14H21N3O3S
(5S)-1-[(2R)-butan-2-yl]-5-[[(2R)-oxolan-2-yl]methyliminomethyl]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[(3R)-3-(2-chlorophenyl)-5-(4-ethylphenyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid —— C22H23ClN2O3
5-[(3R)-3-(2-chlorophenyl)-5-(4-ethylphenyl)-3,4-dihydropyrazol-2-yl]-5-oxopentanoic acid
—— 5-cyclobutyl-N-[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]-1,3,4-oxadiazol-2-amine —— C18H25N5O
5-cyclobutyl-N-[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]-1,3,4-oxadiazol-2-amine
—— (5S,10bR)-2-phenyl-5-[4-(trifluoromethyl)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17F3N2O
(5S,10bR)-2-phenyl-5-[4-(trifluoromethyl)phenyl]-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-N-(1,3-benzodioxol-5-yl)-2-oxa-9-azaspiro[4.5]decane-9-carboxamide —— C16H20N2O4
(5S)-N-(1,3-benzodioxol-5-yl)-2-oxa-9-azaspiro[4.5]decane-9-carboxamide
—— (5R)-7-(6-amino-2-butylsulfanylpyrimidin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C15H23N5O2S
(5R)-7-(6-amino-2-butylsulfanylpyrimidin-4-yl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (5E)-5-[(3,5-dimethylanilino)methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one —— C15H18N2OS2
(5E)-5-[(3,5-dimethylanilino)methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-ethyl-4-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2,6-dimethylpyrimidine —— C20H28N8
5-ethyl-4-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]-2,6-dimethylpyrimidine