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—— 5-[2-(4-Carboxylato-3,3-dimethylbutanoyl)hydrazinyl]-1-methylpyrazole-4-carboxylate —— C12H16N4O5-2
5-[2-(4-Carboxylato-3,3-dimethylbutanoyl)hydrazinyl]-1-methylpyrazole-4-carboxylate
—— (5S)-1-[2-[4-(hydroxymethyl)piperidin-1-yl]ethyl]-5-methyl-5-phenylpiperidin-2-one —— C20H30N2O2
(5S)-1-[2-[4-(hydroxymethyl)piperidin-1-yl]ethyl]-5-methyl-5-phenylpiperidin-2-one
—— 5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylamino)-3,3-dimethyl-5-oxopentanoate —— C16H20NO5-
5-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylamino)-3,3-dimethyl-5-oxopentanoate
—— (5S)-2,2-dimethyl-5-[2-(trifluoromethyl)phenyl]-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one —— C26H22F3NO
(5S)-2,2-dimethyl-5-[2-(trifluoromethyl)phenyl]-1,3,5,6-tetrahydrobenzo[a]phenanthridin-4-one
—— 5-[(3R)-3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C21H20N4O3
5-[(3R)-3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— (5S)-2-[2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3
(5S)-2-[2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5-acetyl-2-methoxyphenyl)methyl (E)-3-(4-methylphenyl)prop-2-enoate —— C20H20O4
(5-acetyl-2-methoxyphenyl)methyl (E)-3-(4-methylphenyl)prop-2-enoate
—— 5-cyclohexyl-N-methyl-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide —— C16H22N4O2
5-cyclohexyl-N-methyl-N-[(1S)-1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[3-(2-ethylimidazol-1-yl)propyl]-5-methylpiperidin-2-one —— C22H29N3O3
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[3-(2-ethylimidazol-1-yl)propyl]-5-methylpiperidin-2-one
—— (5R)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methyl-5-phenylpiperidin-2-one —— C19H23N3O
(5R)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-7-cyclopentyl-2-[2-(1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H25N5O2
(5R)-7-cyclopentyl-2-[2-(1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(5-methoxy-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N3O3
(5S)-2-(5-methoxy-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one —— C21H20N4O3
5-[(3S)-3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-pyridin-3-yl-1H-pyrimidin-6-one
—— (5S)-2-[2-(2-chloro-4-fluorophenyl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H22ClFN2O3
(5S)-2-[2-(2-chloro-4-fluorophenyl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H24N2O3
(5S)-9-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-propyl-2-(1,2,5-trimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O2
(5R)-7-propyl-2-(1,2,5-trimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H26N2O3
(5R)-2-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H24N2O3
(5R)-9-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-cyclohexyl-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide —— C16H22N4O2
5-cyclohexyl-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[3-(2-ethylimidazol-1-yl)propyl]-5-methylpiperidin-2-one —— C22H29N3O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[3-(2-ethylimidazol-1-yl)propyl]-5-methylpiperidin-2-one
—— (5R)-9-[2-(5-methylthiophen-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H21NO2S
(5R)-9-[2-(5-methylthiophen-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(2-methoxyethyl)-2-(4-propylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H30N2O3
(5R)-7-(2-methoxyethyl)-2-(4-propylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(5-methoxy-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N3O3
(5R)-2-(5-methoxy-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propyl-2-(1,2,5-trimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O2
(5S)-7-propyl-2-(1,2,5-trimethylpyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-fluoro-N-[(5R)-4,5,6,7-tetrahydro-1H-indazol-5-yl]quinazolin-4-amine —— C15H14FN5
5-fluoro-N-[(5R)-4,5,6,7-tetrahydro-1H-indazol-5-yl]quinazolin-4-amine
—— (5S)-9-[2-(5-methylthiophen-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C15H21NO2S
(5S)-9-[2-(5-methylthiophen-2-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(2-hydroxyethyl)-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H22N6O2
(5R)-7-(2-hydroxyethyl)-2-(1-phenyltetrazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(2-methoxyethyl)piperidin-2-one —— C17H19N5O3
(5R)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(2-methoxyethyl)piperidin-2-one
—— 5-[(3R)-3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1,7-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C19H26N4O4
5-[(3R)-3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1,7-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— (5R)-1-[2-[4-(hydroxymethyl)piperidin-1-yl]ethyl]-5-methyl-5-phenylpiperidin-2-one —— C20H30N2O2
(5R)-1-[2-[4-(hydroxymethyl)piperidin-1-yl]ethyl]-5-methyl-5-phenylpiperidin-2-one
—— (5R)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H23N3O3
(5R)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-7-cyclopentyl-2-[2-(1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H25N5O2
(5S)-7-cyclopentyl-2-[2-(1,2,4-triazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methylpiperidin-2-one —— C21H27N3O4
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methylpiperidin-2-one
—— (5S)-2-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C21H26N2O3
(5S)-2-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(1-ethyl-2,5-dimethylpyrrole-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H29N3O3
(5R)-2-(1-ethyl-2,5-dimethylpyrrole-3-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H23N3O3
(5S)-9-[2-(4,6-dimethyl-2-oxopyrimidin-1-yl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-7-(cyclopropylmethyl)-2-(3-ethoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H28N2O3
(5R)-7-(cyclopropylmethyl)-2-(3-ethoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)-1-(2-morpholin-4-ylethyl)piperidin-2-one —— C20H24N6O3
(5R)-5-(3-imidazo[1,2-a]pyridin-2-yl-1,2,4-oxadiazol-5-yl)-1-(2-morpholin-4-ylethyl)piperidin-2-one
—— (5R)-2-[2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3
(5R)-2-[2-(2-ethyl-4-methyl-6-oxo-1H-pyrimidin-5-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-fluoro-N-[(5S)-4,5,6,7-tetrahydro-1H-indazol-5-yl]quinazolin-4-amine —— C15H14FN5
5-fluoro-N-[(5S)-4,5,6,7-tetrahydro-1H-indazol-5-yl]quinazolin-4-amine
—— (5R)-7-methyl-2-(5-methyl-4-phenylthiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H24N2O2S
(5R)-7-methyl-2-(5-methyl-4-phenylthiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(2-methoxyethyl)piperidin-2-one —— C17H19N5O3
(5S)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(2-methoxyethyl)piperidin-2-one
—— (5S)-2-[3-(5-methyltetrazol-1-yl)benzoyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H26N6O2
(5S)-2-[3-(5-methyltetrazol-1-yl)benzoyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C16H21N5O3
5-[(3R)-3-[1-(2-methoxyethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5R)-7-(2-methoxyethyl)-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one —— C14H26N2O4S
(5R)-7-(2-methoxyethyl)-2-(2-methylsulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methylpiperidin-2-one —— C21H27N3O4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methylpiperidin-2-one
—— 5-tert-butyl-4-[[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]methyl]furan-2-carboxamide —— C19H30N2O4
5-tert-butyl-4-[[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]methyl]furan-2-carboxamide
—— 5-[(6S)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carbonyl]-1H-pyrimidine-2,4-dione —— C15H21N5O4
5-[(6S)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecane-4-carbonyl]-1H-pyrimidine-2,4-dione
—— (5R)-2-[3-(5-methyltetrazol-1-yl)benzoyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H26N6O2
(5R)-2-[3-(5-methyltetrazol-1-yl)benzoyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-1'-[[5-[(2S)-oxan-2-yl]furan-2-yl]methyl]spiro[6,7-dihydro-1H-imidazo[4,5-c]pyridine-4,4'-piperidine] —— C21H30N4O2
5-methyl-1'-[[5-[(2S)-oxan-2-yl]furan-2-yl]methyl]spiro[6,7-dihydro-1H-imidazo[4,5-c]pyridine-4,4'-piperidine]