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—— 5-ethyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine —— C15H20N4
5-ethyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
—— 5-[[4-[(4R)-2,2-dimethyloxan-4-yl]triazol-1-yl]methyl]thiophene-2-carboxylic acid —— C15H19N3O3S
5-[[4-[(4R)-2,2-dimethyloxan-4-yl]triazol-1-yl]methyl]thiophene-2-carboxylic acid
—— 5-chloro-6-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]pyridine-3-carboxylic acid —— C16H22ClN3O3
5-chloro-6-[4-[(3S)-3-hydroxypiperidin-1-yl]piperidin-1-yl]pyridine-3-carboxylic acid
—— 5-[benzyl(methyl)amino]-2-[[(2R)-oxan-2-yl]methyl]pyridazin-3-one —— C18H23N3O2
5-[benzyl(methyl)amino]-2-[[(2R)-oxan-2-yl]methyl]pyridazin-3-one
—— 5-[1-[(2S)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]pyrimidine —— C13H13N5OS
5-[1-[(2S)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]pyrimidine
—— 5-ethyl-2-[(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]pyrimidine —— C15H21N5
5-ethyl-2-[(3S)-3-(imidazol-1-ylmethyl)piperidin-1-yl]pyrimidine
—— 5-[benzyl(methyl)amino]-2-[[(2S)-oxan-2-yl]methyl]pyridazin-3-one —— C18H23N3O2
5-[benzyl(methyl)amino]-2-[[(2S)-oxan-2-yl]methyl]pyridazin-3-one
—— 5-ethyl-2-[(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]pyrimidine —— C15H21N5
5-ethyl-2-[(3R)-3-(imidazol-1-ylmethyl)piperidin-1-yl]pyrimidine
—— 5-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-methyl-2-(1,2,4-triazol-4-yl)pyridine —— C19H20N4O2
5-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-methyl-2-(1,2,4-triazol-4-yl)pyridine
—— 5-chloro-6-[4-[(3R)-3-hydroxypiperidin-1-yl]piperidin-1-yl]pyridine-3-carboxylic acid —— C16H22ClN3O3
5-chloro-6-[4-[(3R)-3-hydroxypiperidin-1-yl]piperidin-1-yl]pyridine-3-carboxylic acid
—— 5-[1-[(2R)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]pyrimidine —— C13H13N5OS
5-[1-[(2R)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]pyrimidine
—— (5R)-5-methoxy-9-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecane —— C16H25N3O4S
(5R)-5-methoxy-9-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecane
—— 5-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-methyl-2-(1,2,4-triazol-4-yl)pyridine —— C19H20N4O2
5-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-methyl-2-(1,2,4-triazol-4-yl)pyridine
—— 5-fluoro-4-N-methyl-2-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrimidine-2,4-diamine —— C16H19FN4O
5-fluoro-4-N-methyl-2-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrimidine-2,4-diamine
—— (5R)-9-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C21H27N3O2
(5R)-9-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5S)-5-methoxy-9-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecane —— C16H25N3O4S
(5S)-5-methoxy-9-(2-methyl-5-methylsulfonylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecane
—— (5S)-9-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C21H27N3O2
(5S)-9-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-fluoro-4-N-methyl-2-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrimidine-2,4-diamine —— C16H19FN4O
5-fluoro-4-N-methyl-2-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]pyrimidine-2,4-diamine
—— 5-oxo-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C18H17N3O3S
5-oxo-N-[[(4S)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— (5R)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O2S
(5R)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(5-ethylthiophene-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H28N2O3S
(5R)-2-(5-ethylthiophene-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(morpholin-4-ylmethyl)-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]furan-3-carboxamide —— C19H25N5O3
5-(morpholin-4-ylmethyl)-N-[(3S)-1-pyrimidin-2-ylpiperidin-3-yl]furan-3-carboxamide
—— (5S)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H24N4O2S
(5S)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(1R)-1-(4-chloropyrazol-1-yl)ethyl]-1-(2-phenylethyl)-1,2,4-triazole —— C15H16ClN5
5-[(1R)-1-(4-chloropyrazol-1-yl)ethyl]-1-(2-phenylethyl)-1,2,4-triazole
—— 5,6-dimethyl-2-[2-oxo-2-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl]pyridazin-3-one —— C19H24N4O3
5,6-dimethyl-2-[2-oxo-2-[(3R)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl]pyridazin-3-one
—— 5-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C15H17N3O2
5-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— (5S)-2-(5-ethylthiophene-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H28N2O3S
(5S)-2-(5-ethylthiophene-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-4-N-[(2R)-2-phenyl-2-piperidin-1-ylethyl]pyrimidine-2,4-diamine —— C19H27N5
5-ethyl-4-N-[(2R)-2-phenyl-2-piperidin-1-ylethyl]pyrimidine-2,4-diamine
—— 5-(morpholin-4-ylmethyl)-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]furan-3-carboxamide —— C19H25N5O3
5-(morpholin-4-ylmethyl)-N-[(3R)-1-pyrimidin-2-ylpiperidin-3-yl]furan-3-carboxamide
—— 5-ethyl-4-N-[(2S)-2-phenyl-2-piperidin-1-ylethyl]pyrimidine-2,4-diamine —— C19H27N5
5-ethyl-4-N-[(2S)-2-phenyl-2-piperidin-1-ylethyl]pyrimidine-2,4-diamine
—— 5-[(1S)-1-(4-chloropyrazol-1-yl)ethyl]-1-(2-phenylethyl)-1,2,4-triazole —— C15H16ClN5
5-[(1S)-1-(4-chloropyrazol-1-yl)ethyl]-1-(2-phenylethyl)-1,2,4-triazole
—— 5-oxo-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide —— C18H17N3O3S
5-oxo-N-[[(4R)-2,3,4,5-tetrahydro-1-benzoxepin-4-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
—— 5-ethyl-4-N-[[(3S)-1-(3-methoxypropyl)pyrrolidin-3-yl]methyl]-6-methylpyrimidine-2,4-diamine —— C16H29N5O
5-ethyl-4-N-[[(3S)-1-(3-methoxypropyl)pyrrolidin-3-yl]methyl]-6-methylpyrimidine-2,4-diamine
—— 5-ethyl-4-N-[[(3R)-1-(3-methoxypropyl)pyrrolidin-3-yl]methyl]-6-methylpyrimidine-2,4-diamine —— C16H29N5O
5-ethyl-4-N-[[(3R)-1-(3-methoxypropyl)pyrrolidin-3-yl]methyl]-6-methylpyrimidine-2,4-diamine
—— (5R)-7-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide —— C20H29N3O4
(5R)-7-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
—— 5-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine —— C15H17N3O2
5-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine
—— 5,6-dimethyl-2-[2-oxo-2-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl]pyridazin-3-one —— C19H24N4O3
5,6-dimethyl-2-[2-oxo-2-[(3S)-3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl]pyridazin-3-one
—— (5S)-7-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide —— C20H29N3O4
(5S)-7-(2-methoxyethyl)-N-[(4-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5R)-2-(7-chloroquinolin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H24ClN3O2
(5R)-2-(7-chloroquinolin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H23N5O3S2
(5R)-2-[2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-fluoro-N-methyl-2-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine —— C19H22FN7
5-fluoro-N-methyl-2-[(3S)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine
—— 5-fluoro-N-methyl-2-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine —— C19H22FN7
5-fluoro-N-methyl-2-[(3R)-3-[1-(pyridin-2-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyrimidin-4-amine
—— (5S)-7-(cyclobutylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2
(5S)-7-(cyclobutylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[6-(4-fluorophenyl)pyridazin-3-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H25FN4O2
(5S)-2-[6-(4-fluorophenyl)pyridazin-3-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(4-Methylphenyl)-2-[[2-(trifluoromethyl)phenyl]methyl]tetrazole —— C16H13F3N4
5-(4-Methylphenyl)-2-[[2-(trifluoromethyl)phenyl]methyl]tetrazole
—— 5-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C18H23N5O2
5-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— (5R)-7-(cyclobutylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H26N4O2
(5R)-7-(cyclobutylmethyl)-2-(2-pyrazin-2-ylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one —— C18H23N5O2
5-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]-1H-pyrazin-2-one
—— 5-(4-Methylphenyl)-2-[(4-propan-2-ylphenyl)methyl]tetrazole —— C18H20N4
5-(4-Methylphenyl)-2-[(4-propan-2-ylphenyl)methyl]tetrazole
—— (5S)-2-(7-chloroquinolin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H24ClN3O2
(5S)-2-(7-chloroquinolin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one