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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(2R)-2-(cyclohexylmethyl)pyrrolidine-1-carbonyl]furan-2-sulfonamide —— C16H24N2O4S
5-[(2R)-2-(cyclohexylmethyl)pyrrolidine-1-carbonyl]furan-2-sulfonamide
—— (5-ethyl-1H-pyrazol-4-yl)-[(4S)-4-propylazepan-1-yl]methanone —— C15H25N3O
(5-ethyl-1H-pyrazol-4-yl)-[(4S)-4-propylazepan-1-yl]methanone
—— (5S)-9-[(2-morpholin-4-yl-1,3-thiazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decane —— C16H25N3O2S
(5S)-9-[(2-morpholin-4-yl-1,3-thiazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decane
—— 5-[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C15H18N2O3
5-[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-ethyl-4-N-[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidine-2,4-diamine —— C18H26N6
5-ethyl-4-N-[(2R)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidine-2,4-diamine
—— (5-chlorothiophen-2-yl)-[(3S)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone —— C17H18ClNO2S
(5-chlorothiophen-2-yl)-[(3S)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone
—— (5R)-1-(2-methoxyethyl)-5-[2-[(3-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]piperidin-2-one —— C18H24N4O3
(5R)-1-(2-methoxyethyl)-5-[2-[(3-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]piperidin-2-one
—— 5-[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]-3-propan-2-yl-1,2,4-oxadiazole —— C15H18N2O3
5-[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5-propan-2-yl-1,2-oxazol-3-yl)-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C21H25N5O2
(5-propan-2-yl-1,2-oxazol-3-yl)-[(3S)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5-propan-2-yl-1,2-oxazol-3-yl)-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C21H25N5O2
(5-propan-2-yl-1,2-oxazol-3-yl)-[(3R)-3-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5R)-9-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H23N5O2
(5R)-9-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-methoxy-N-methyl-4-oxo-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]pyran-2-carboxamide —— C19H22N2O4
5-methoxy-N-methyl-4-oxo-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]pyran-2-carboxamide
—— 5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ylethyl]-2-methoxybenzamide —— C22H28ClN3O2
5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ylethyl]-2-methoxybenzamide
—— 5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ylethyl]-2-methoxybenzamide —— C22H28ClN3O2
5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ylethyl]-2-methoxybenzamide
—— 5-fluoro-4-N,4-N-dimethyl-2-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine —— C11H14FN5S
5-fluoro-4-N,4-N-dimethyl-2-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine
—— (5S)-9-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one —— C16H23N5O2
(5S)-9-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-3-methyl-1-oxa-3,9-diazaspiro[4.5]decan-2-one
—— 5-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]pyridine-2-carbonitrile —— C20H23N5O
5-[(3R)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]pyridine-2-carbonitrile
—— 5-chloro-N-[(2R)-2-(dimethylamino)-2-[4-(dimethylamino)phenyl]ethyl]-2-nitrobenzamide —— C19H23ClN4O3
5-chloro-N-[(2R)-2-(dimethylamino)-2-[4-(dimethylamino)phenyl]ethyl]-2-nitrobenzamide
—— 5-(5-methylfuran-2-yl)-2-(3-nitrophenyl)-N-[(1S)-1-phenylethyl]pyrazole-3-carboxamide —— C23H20N4O4
5-(5-methylfuran-2-yl)-2-(3-nitrophenyl)-N-[(1S)-1-phenylethyl]pyrazole-3-carboxamide
—— 5-[[2-[[(2-methoxyacetyl)-propylamino]methyl]pyrrol-1-yl]methyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide —— C23H34N4O4
5-[[2-[[(2-methoxyacetyl)-propylamino]methyl]pyrrol-1-yl]methyl]-N-(2-pyrrolidin-1-ylethyl)furan-2-carboxamide
—— 5-methyl-1-[2-[(6S)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecan-4-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C17H25N5O4
5-methyl-1-[2-[(6S)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecan-4-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— 5-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]pyridine-2-carbonitrile —— C20H23N5O
5-[(3S)-3-[1-(cyclobutylmethyl)imidazol-2-yl]piperidine-1-carbonyl]pyridine-2-carbonitrile
—— 5-fluoro-4-N,4-N-dimethyl-2-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine —— C11H14FN5S
5-fluoro-4-N,4-N-dimethyl-2-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine
—— 5-methoxy-N-methyl-4-oxo-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]pyran-2-carboxamide —— C19H22N2O4
5-methoxy-N-methyl-4-oxo-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]pyran-2-carboxamide
—— [5-[[[(2R)-butan-2-yl]-(4-methylbenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate —— C21H27NO5S
[5-[[[(2R)-butan-2-yl]-(4-methylbenzoyl)amino]methyl]-2-methoxyphenyl] methanesulfonate
—— (5S,6S,7R)-6,8-dimethyl-7-phenyl-1,3,8-triazaspiro[4.5]decane-2,4-dithione —— C15H19N3S2
(5S,6S,7R)-6,8-dimethyl-7-phenyl-1,3,8-triazaspiro[4.5]decane-2,4-dithione
—— 5-[(3-Chloro-4-nitrobenzoyl)amino]benzene-1,3-dicarboxylate —— C15H7ClN2O7-2
5-[(3-Chloro-4-nitrobenzoyl)amino]benzene-1,3-dicarboxylate
—— (5S,6R,7R)-6,8-dimethyl-7-phenyl-1,3,8-triazaspiro[4.5]decane-2,4-dithione —— C15H19N3S2
(5S,6R,7R)-6,8-dimethyl-7-phenyl-1,3,8-triazaspiro[4.5]decane-2,4-dithione
—— 5-methyl-1-[2-[(6R)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecan-4-yl]-2-oxoethyl]pyrimidine-2,4-dione —— C17H25N5O4
5-methyl-1-[2-[(6R)-1-methyl-9-oxo-1,4,10-triazaspiro[5.6]dodecan-4-yl]-2-oxoethyl]pyrimidine-2,4-dione
—— (5R,10bR)-1'-methyl-2-(4-methylphenyl)spiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one —— C25H21N3O2
(5R,10bR)-1'-methyl-2-(4-methylphenyl)spiro[3,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-indole]-2'-one
—— (5S,6S,7S)-6,8-dimethyl-7-phenyl-1,3,8-triazaspiro[4.5]decane-2,4-dithione —— C15H19N3S2
(5S,6S,7S)-6,8-dimethyl-7-phenyl-1,3,8-triazaspiro[4.5]decane-2,4-dithione
—— 5-fluoro-2-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]pyridine —— C16H24FN3
5-fluoro-2-[4-[(1R)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]pyridine
—— (5S,10bS)-2-(4-fluorophenyl)-5-(3-nitrophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H16FN3O3
(5S,10bS)-2-(4-fluorophenyl)-5-(3-nitrophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-9-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H25N3O3
(5R)-9-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-[(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N-[(2R)-butan-2-yl]furan-2-carboxamide —— C20H22N2O5
5-[(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N-[(2R)-butan-2-yl]furan-2-carboxamide
—— 5-[(3S)-1-acetylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide —— C18H25N3O3S
5-[(3S)-1-acetylpiperidine-3-carbonyl]-N,N-dimethyl-6,7-dihydro-4H-thieno[3,2-c]pyridine-2-carboxamide
—— (5R)-1-(2-methoxyethyl)-5-(7-methoxy-1,2,4,5-tetrahydro-3-benzazepine-3-carbonyl)piperidin-2-one —— C20H28N2O4
(5R)-1-(2-methoxyethyl)-5-(7-methoxy-1,2,4,5-tetrahydro-3-benzazepine-3-carbonyl)piperidin-2-one
—— (5S)-9-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H25N3O3
(5S)-9-[(5-propan-2-yl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-5-methoxy-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecane —— C15H20F3N3O2
(5R)-5-methoxy-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecane
—— (5S)-5-methoxy-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecane —— C15H20F3N3O2
(5S)-5-methoxy-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecane
—— 5-ethyl-4-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidine-2,4-diamine —— C14H23N7
5-ethyl-4-N-[(1R)-3-methyl-1-(2-methyl-1,2,4-triazol-3-yl)butyl]pyrimidine-2,4-diamine
—— 5,7-dimethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine —— C20H24N6O
5,7-dimethyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine
—— 5-[(2S)-2-(furan-2-yl)azepane-1-carbonyl]-1H-pyrazin-2-one —— C15H17N3O3
5-[(2S)-2-(furan-2-yl)azepane-1-carbonyl]-1H-pyrazin-2-one
—— 5,7-dimethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine —— C20H24N6O
5,7-dimethyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-4-ylethyl]pyrido[2,3-d]pyrimidin-4-amine
—— 5-fluoro-2-[4-[(1S)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]pyridine —— C16H24FN3
5-fluoro-2-[4-[(1S)-1-pyrrolidin-1-ylethyl]piperidin-1-yl]pyridine
—— (5R)-7-(2-methoxyethyl)-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one —— C23H35N3O2
(5R)-7-(2-methoxyethyl)-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(5,6,7,8-tetrahydroquinolin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C18H26N2O2
(5S)-9-(5,6,7,8-tetrahydroquinolin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5-cyclobutyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-1,3,4-oxadiazol-2-amine —— C14H16FN3O
5-cyclobutyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-1,3,4-oxadiazol-2-amine
—— 5-cyclobutyl-N-[(1S)-1-(4-fluorophenyl)ethyl]-1,3,4-oxadiazol-2-amine —— C14H16FN3O
5-cyclobutyl-N-[(1S)-1-(4-fluorophenyl)ethyl]-1,3,4-oxadiazol-2-amine
—— (5S)-9-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]-2-oxa-9-azaspiro[4.5]decane —— C16H21N3O4S
(5S)-9-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]-2-oxa-9-azaspiro[4.5]decane