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—— 5,6-dimethyl-2-oxo-N-[(1S,2S)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide —— C19H20F3N3O2
5,6-dimethyl-2-oxo-N-[(1S,2S)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide
—— 5,8-dimethyl-2-[[2-[(2S)-oxan-2-yl]ethylamino]methyl]-1H-quinolin-4-one —— C19H26N2O2
5,8-dimethyl-2-[[2-[(2S)-oxan-2-yl]ethylamino]methyl]-1H-quinolin-4-one
—— (5R)-7-(cyclopropylmethyl)-2-[2-(2-methylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O2
(5R)-7-(cyclopropylmethyl)-2-[2-(2-methylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[(2-pyrrolidin-1-yl-1,3-thiazol-4-yl)methyl]piperidin-2-one —— C20H31N3OS
(5S)-5-methyl-5-(4-methylpent-3-enyl)-1-[(2-pyrrolidin-1-yl-1,3-thiazol-4-yl)methyl]piperidin-2-one
—— (5S)-3-[2-(1H-imidazol-5-yl)ethylimino]-5-thiophen-2-ylcyclohexan-1-one —— C15H17N3OS
(5S)-3-[2-(1H-imidazol-5-yl)ethylimino]-5-thiophen-2-ylcyclohexan-1-one
—— (5R)-7-cyclopentyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O2
(5R)-7-cyclopentyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-propan-2-yl-2-[2-(tetrazol-1-yl)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H23N7O2
(5R)-7-propan-2-yl-2-[2-(tetrazol-1-yl)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[(1-ethylindazol-3-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H23N3O2
(5R)-9-[(1-ethylindazol-3-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C12H18N4O2
(5S)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5,6-dimethyl-2-oxo-N-[(1R,2S)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide —— C19H20F3N3O2
5,6-dimethyl-2-oxo-N-[(1R,2S)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide
—— (5S)-7-cyclohexyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O3S
(5S)-7-cyclohexyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-propan-2-yl-2-[2-(tetrazol-1-yl)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H23N7O2
(5S)-7-propan-2-yl-2-[2-(tetrazol-1-yl)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(2-hydroxyethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25N3O2
(5R)-7-(2-hydroxyethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C19H31N3O2
(5S)-9-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— 5,6-dimethyl-2-oxo-N-[(1R,2R)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide —— C19H20F3N3O2
5,6-dimethyl-2-oxo-N-[(1R,2R)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide
—— (5R)-5-(3,3-diphenylpiperidine-1-carbonyl)-1-methylpiperidin-2-one —— C24H28N2O2
(5R)-5-(3,3-diphenylpiperidine-1-carbonyl)-1-methylpiperidin-2-one
—— 5,6-dimethyl-2-oxo-N-[(1S,2R)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide —— C19H20F3N3O2
5,6-dimethyl-2-oxo-N-[(1S,2R)-2-[2-(trifluoromethyl)phenyl]cyclopentyl]-1H-pyrazine-3-carboxamide
—— [5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3S)-3-phenylpiperazin-1-yl]methanone —— C20H19FN4O
[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3S)-3-phenylpiperazin-1-yl]methanone
—— (5S)-9-[(1-ethylindazol-3-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H23N3O2
(5S)-9-[(1-ethylindazol-3-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-chloro-2-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine —— C19H20ClN5
5-chloro-2-[(3S)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine
—— (5R)-7-cyclopentyl-2-(4-fluoro-2-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN2O2
(5R)-7-cyclopentyl-2-(4-fluoro-2-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-2-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine —— C19H20ClN5
5-chloro-2-[(3R)-3-[1-(pyridin-4-ylmethyl)imidazol-2-yl]piperidin-1-yl]pyridine
—— 5-(4-chlorophenyl)-1-(2-fluorophenyl)-2-methyl-N-(2-methylpropyl)pyrrole-3-carboxamide —— C22H22ClFN2O
5-(4-chlorophenyl)-1-(2-fluorophenyl)-2-methyl-N-(2-methylpropyl)pyrrole-3-carboxamide
—— (5S)-7-(2-hydroxyethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H25N3O2
(5S)-7-(2-hydroxyethyl)-2-(4-methylquinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methanone —— C20H22N4O3
[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methanone
—— (5S)-5-(4-fluoroanilino)-3-methyl-1,3-thiazolidine-2,4-dione —— C10H9FN2O2S
(5S)-5-(4-fluoroanilino)-3-methyl-1,3-thiazolidine-2,4-dione
—— [5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methanone —— C20H22N4O3
[5-(3-methoxyphenyl)-1H-pyrazol-4-yl]-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methanone
—— (5S)-7-cyclopentyl-2-(4-fluoro-2-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN2O2
(5S)-7-cyclopentyl-2-(4-fluoro-2-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O3S
(5S)-2-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone —— C20H19FN4O
[5-(3-fluorophenyl)-1H-pyrazol-4-yl]-[(3R)-3-phenylpiperazin-1-yl]methanone
—— (5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[(2-pyrrolidin-1-yl-1,3-thiazol-4-yl)methyl]piperidin-2-one —— C20H31N3OS
(5R)-5-methyl-5-(4-methylpent-3-enyl)-1-[(2-pyrrolidin-1-yl-1,3-thiazol-4-yl)methyl]piperidin-2-one
—— 5-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-thiophen-2-yl-1H-pyrimidin-6-one —— C17H16N4O3S
5-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-2-thiophen-2-yl-1H-pyrimidin-6-one
—— (5S)-7-(cyclopropylmethyl)-2-[2-(2-methylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O2
(5S)-7-(cyclopropylmethyl)-2-[2-(2-methylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3-chlorobenzoyl)amino]-2-(dimethylamino)-N-[(1S)-1-phenylethyl]benzamide —— C24H24ClN3O2
5-[(3-chlorobenzoyl)amino]-2-(dimethylamino)-N-[(1S)-1-phenylethyl]benzamide
—— (5R)-7-cyclohexyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O3S
(5R)-7-cyclohexyl-2-pyridin-3-ylsulfonyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-[2-(3-methoxyphenyl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C17H23NO3
(5R)-9-[2-(3-methoxyphenyl)ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R)-9-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C19H31N3O2
(5R)-9-[[2-(cyclopentylmethyl)-1H-imidazol-5-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-methylpiperidin-2-one —— C19H23N3O4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-methylpiperidin-2-one
—— (5S)-7-cyclopentyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H27N3O2
(5S)-7-cyclopentyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C21H25N3O3
(5R)-2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-(3-methoxyphenyl)-N-methyl-N-[3-[(2S)-oxolan-2-yl]propyl]-1H-pyrazole-4-carboxamide —— C19H25N3O3
5-(3-methoxyphenyl)-N-methyl-N-[3-[(2S)-oxolan-2-yl]propyl]-1H-pyrazole-4-carboxamide
—— (5S)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3
(5S)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-one —— C20H25N3O4
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-one —— C20H25N3O4
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-one
—— (5R)-1-[(2-methoxyphenyl)methyl]-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C18H23N3O3
(5R)-1-[(2-methoxyphenyl)methyl]-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5R)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H28N4O3
(5R)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-[(3-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H29FN2O
(5R)-7-cyclohexyl-2-[(3-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H26N4O3
(5S)-2-[[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H27N3O3
(5R)-2-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H27N3O3
(5S)-2-(2-oxo-1,5,6,7-tetrahydrocyclopenta[b]pyridine-3-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one