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中文名称 英文名称 CAS号 化学式 结构式图片
—— (5R)-5-(1,3-benzodioxol-5-yl)-1-hexyl-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione —— C24H25NO5
(5R)-5-(1,3-benzodioxol-5-yl)-1-hexyl-4-[hydroxy(phenyl)methylidene]pyrrolidine-2,3-dione
—— (5S)-1-hexyl-4-[hydroxy(phenyl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C24H27NO4
(5S)-1-hexyl-4-[hydroxy(phenyl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— (5R)-7-(2-methoxyethyl)-2-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H23N3O5S
(5R)-7-(2-methoxyethyl)-2-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H27N5O
(5R)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-methyl-2-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrimidine —— C16H27N5
5-methyl-2-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrimidine
—— (5S)-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one —— C18H24N2O3S
(5S)-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
—— (5S)-1-hexyl-4-[hydroxy(phenyl)methylidene]-5-(4-methylphenyl)pyrrolidine-2,3-dione —— C24H27NO3
(5S)-1-hexyl-4-[hydroxy(phenyl)methylidene]-5-(4-methylphenyl)pyrrolidine-2,3-dione
—— (5S)-1-hexyl-4-[hydroxy-(4-methylphenyl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione —— C25H29NO4
(5S)-1-hexyl-4-[hydroxy-(4-methylphenyl)methylidene]-5-(4-methoxyphenyl)pyrrolidine-2,3-dione
—— (5S)-7-(2-methoxyethyl)-2-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one —— C15H23N3O5S
(5S)-7-(2-methoxyethyl)-2-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3S)-3-(1-butylimidazol-2-yl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide —— C16H24N6O2
5-[[(3S)-3-(1-butylimidazol-2-yl)piperidin-1-yl]methyl]-1,2,4-oxadiazole-3-carboxamide
—— 5-[[[(1R)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-fluorophenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C23H21FN4OS
5-[[[(1R)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-fluorophenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— (5S,10bR)-9-chloro-5-(4-fluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14ClFN2OS
(5S,10bR)-9-chloro-5-(4-fluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O3
(5R)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— [(5S,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-chlorophenyl)methanone —— C21H15ClN2O2S
[(5S,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-chlorophenyl)methanone
—— (5R)-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one —— C18H24N2O3S
(5R)-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
—— [(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(3-pyrazol-1-ylphenyl)methanone —— C19H23N3O3
[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(3-pyrazol-1-ylphenyl)methanone
—— 5-methyl-2-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrimidine —— C16H27N5
5-methyl-2-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]pyrimidine
—— (5S)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H27N5O
(5S)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-butyl-4-[hydroxy(phenyl)methylidene]-5-(2-methoxyphenyl)pyrrolidine-2,3-dione —— C22H23NO4
(5S)-1-butyl-4-[hydroxy(phenyl)methylidene]-5-(2-methoxyphenyl)pyrrolidine-2,3-dione
—— (5S,10bS)-2-(4-methylphenyl)-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H22N2O
(5S,10bS)-2-(4-methylphenyl)-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O3
(5S)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— [(5S,10bS)-9-chloro-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-fluorophenyl)methanone —— C21H14ClFN2O2S
[(5S,10bS)-9-chloro-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-fluorophenyl)methanone
—— 5-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-fluorophenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C23H21FN4OS
5-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-fluorophenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(3-pyrazol-1-ylphenyl)methanone —— C19H23N3O3
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(3-pyrazol-1-ylphenyl)methanone
—— (5S,10bS)-9-chloro-2-(4-methoxyphenyl)-5-methyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C18H17ClN2O2
(5S,10bS)-9-chloro-2-(4-methoxyphenyl)-5-methyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-9-chloro-2-(4-chlorophenyl)-5-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14Cl2N2OS
(5R,10bS)-9-chloro-2-(4-chlorophenyl)-5-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-propyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C17H18N2OS
(5S,10bS)-5-propyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-9-chloro-5-propyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C17H17ClN2OS
(5S,10bS)-9-chloro-5-propyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-9-bromo-5-methyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C15H13BrN2OS
(5S,10bS)-9-bromo-5-methyl-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-9-[(3-methylthiophen-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H23NO2S
(5S)-9-[(3-methylthiophen-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-9-[(3-methylthiophen-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C15H23NO2S
(5R)-9-[(3-methylthiophen-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-2-(6-aminopyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H23N5O2
(5R)-2-(6-aminopyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R,10bS)-9-bromo-2-phenyl-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C19H19BrN2O
(5R,10bS)-9-bromo-2-phenyl-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-2-(6-aminopyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C15H23N5O2
(5S)-2-(6-aminopyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bR)-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H15ClN2OS
(5S,10bR)-5-(4-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-(4-chlorophenyl)-5-methyl-2-thiophen-2-yl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C21H17ClN2OS
(5S,10bS)-5-(4-chlorophenyl)-5-methyl-2-thiophen-2-yl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-2-(4-methoxyphenyl)-5-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H22N2O2
(5S,10bS)-2-(4-methoxyphenyl)-5-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-9-bromo-2,5-diphenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H17BrN2O
(5R,10bS)-9-bromo-2,5-diphenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-9-chloro-5-(4-methylphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H19ClN2O
(5S,10bS)-9-chloro-5-(4-methylphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-cyclohexyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H24N2O
(5S,10bS)-5-cyclohexyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-2-phenyl-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C19H20N2O
(5S,10bS)-2-phenyl-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-9-bromo-5-methyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C17H15BrN2O
(5S,10bS)-9-bromo-5-methyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-cyclohexyl-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H26N2O
(5S,10bS)-5-cyclohexyl-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-2,5-bis(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H22N2O
(5R,10bS)-2,5-bis(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-phenyl-N-[[(3S)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide —— C21H23N5O
5-phenyl-N-[[(3S)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide
—— (5S,10bR)-5-cyclohexyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H24N2O
(5S,10bR)-5-cyclohexyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-phenyl-N-[[(3R)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide —— C21H23N5O
5-phenyl-N-[[(3R)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide
—— (5S)-9-(5-phenyl-1,3,4-thiadiazol-2-yl)-2-oxa-9-azaspiro[4.5]decane —— C16H19N3OS
(5S)-9-(5-phenyl-1,3,4-thiadiazol-2-yl)-2-oxa-9-azaspiro[4.5]decane
—— (5R)-9-(5-phenyl-1,3,4-thiadiazol-2-yl)-2-oxa-9-azaspiro[4.5]decane —— C16H19N3OS
(5R)-9-(5-phenyl-1,3,4-thiadiazol-2-yl)-2-oxa-9-azaspiro[4.5]decane
—— 5-[[(3R)-3-(1-butylimidazol-2-yl)piperidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H28N6O
5-[[(3R)-3-(1-butylimidazol-2-yl)piperidin-1-yl]methyl]-2-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one