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—— 5-[(1S,2S)-2-(5-methylthiophen-2-yl)cyclopropyl]-3-(propan-2-yloxymethyl)-1,2,4-oxadiazole —— C14H18N2O2S
5-[(1S,2S)-2-(5-methylthiophen-2-yl)cyclopropyl]-3-(propan-2-yloxymethyl)-1,2,4-oxadiazole
—— 5,7-dimethyl-6-[3-oxo-3-[(4R)-4-propylazepan-1-yl]propyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one —— C20H30N4O2
5,7-dimethyl-6-[3-oxo-3-[(4R)-4-propylazepan-1-yl]propyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one
—— 5-[(2S)-1-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidin-2-yl]-3-pyrimidin-2-yl-1,2,4-oxadiazole —— C16H18N6O2
5-[(2S)-1-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidin-2-yl]-3-pyrimidin-2-yl-1,2,4-oxadiazole
—— 5-ethyl-3-[[(2R)-2-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1,2,4-oxadiazole —— C16H19N7O2
5-ethyl-3-[[(2R)-2-(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1,2,4-oxadiazole
—— 5-bromo-2-[(3S)-3-imidazol-1-ylpiperidin-1-yl]pyrimidine —— C12H14BrN5
5-bromo-2-[(3S)-3-imidazol-1-ylpiperidin-1-yl]pyrimidine
—— 5-cyano-N-[(2S)-2-hydroxy-3-[(1R)-1-phenylethoxy]propyl]pyridine-2-carboxamide —— C18H19N3O3
5-cyano-N-[(2S)-2-hydroxy-3-[(1R)-1-phenylethoxy]propyl]pyridine-2-carboxamide
—— 5,7-dimethyl-6-[3-oxo-3-[(4S)-4-propylazepan-1-yl]propyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one —— C20H30N4O2
5,7-dimethyl-6-[3-oxo-3-[(4S)-4-propylazepan-1-yl]propyl]-1H-pyrazolo[1,5-a]pyrimidin-2-one
—— 5-bromo-N-[(2S)-2-hydroxypropyl]-2-methoxy-N-phenylbenzenesulfonamide —— C16H18BrNO4S
5-bromo-N-[(2S)-2-hydroxypropyl]-2-methoxy-N-phenylbenzenesulfonamide
—— 5-cyano-N-[(2R)-2-hydroxy-3-[(1R)-1-phenylethoxy]propyl]pyridine-2-carboxamide —— C18H19N3O3
5-cyano-N-[(2R)-2-hydroxy-3-[(1R)-1-phenylethoxy]propyl]pyridine-2-carboxamide
—— 5-cyano-N-[(2R)-2-hydroxy-3-[(1S)-1-phenylethoxy]propyl]pyridine-2-carboxamide —— C18H19N3O3
5-cyano-N-[(2R)-2-hydroxy-3-[(1S)-1-phenylethoxy]propyl]pyridine-2-carboxamide
—— 5-bromo-N-[(2R)-2-hydroxypropyl]-2-methoxy-N-phenylbenzenesulfonamide —— C16H18BrNO4S
5-bromo-N-[(2R)-2-hydroxypropyl]-2-methoxy-N-phenylbenzenesulfonamide
—— 5-cyano-N-[(2S)-2-hydroxy-3-[(1S)-1-phenylethoxy]propyl]pyridine-2-carboxamide —— C18H19N3O3
5-cyano-N-[(2S)-2-hydroxy-3-[(1S)-1-phenylethoxy]propyl]pyridine-2-carboxamide
—— [5-[(3,5-Dimethylpyrazol-1-yl)methyl]furan-2-yl]-piperidin-1-ylmethanone —— C16H21N3O2
[5-[(3,5-Dimethylpyrazol-1-yl)methyl]furan-2-yl]-piperidin-1-ylmethanone
—— [5-[(3,5-Dimethylpyrazol-1-yl)methyl]furan-2-yl]-pyrrolidin-1-ylmethanone —— C15H19N3O2
[5-[(3,5-Dimethylpyrazol-1-yl)methyl]furan-2-yl]-pyrrolidin-1-ylmethanone
—— 5-methyl-N-[3-(2-methylpropylamino)-3-oxopropyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrazine-2-carboxamide —— C18H28N4O3
5-methyl-N-[3-(2-methylpropylamino)-3-oxopropyl]-N-[[(2S)-oxolan-2-yl]methyl]pyrazine-2-carboxamide
—— 5-(2-chlorophenyl)-2-(4-methoxyphenyl)-N-[(2R)-3-methylbutan-2-yl]pyrazole-3-carboxamide —— C22H24ClN3O2
5-(2-chlorophenyl)-2-(4-methoxyphenyl)-N-[(2R)-3-methylbutan-2-yl]pyrazole-3-carboxamide
—— (5S)-4-anilino-7,7-dimethyl-1-(4-methylphenyl)-8-oxa-1,3-diazaspiro[4.5]dec-3-ene-2-thione —— C22H25N3OS
(5S)-4-anilino-7,7-dimethyl-1-(4-methylphenyl)-8-oxa-1,3-diazaspiro[4.5]dec-3-ene-2-thione
—— 5-fluoro-2-methoxy-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-6-yl)benzenesulfonamide —— C17H19FN2O5S2
5-fluoro-2-methoxy-N-(1-methylsulfonyl-3,4-dihydro-2H-quinolin-6-yl)benzenesulfonamide
—— 5-ethyl-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-sulfonamide —— C19H24N2O3S2
5-ethyl-N-(1-isobutyryl-1,2,3,4-tetrahydroquinolin-6-yl)thiophene-2-sulfonamide
—— 5,6-dimethyl-4-[(2S)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine —— C17H20N4S2
5,6-dimethyl-4-[(2S)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine
—— (5-methyl-4-nitro-1H-pyrazol-3-yl)-[(2R)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone —— C16H18N4O3
(5-methyl-4-nitro-1H-pyrazol-3-yl)-[(2R)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone
—— (5R)-N-[1-(2-methoxyethyl)indol-5-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H21N3O3
(5R)-N-[1-(2-methoxyethyl)indol-5-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-nitro-4-N-[[(2R)-oxolan-2-yl]methyl]-2-pyrrolidin-1-ylpyrimidine-4,6-diamine —— C13H20N6O3
5-nitro-4-N-[[(2R)-oxolan-2-yl]methyl]-2-pyrrolidin-1-ylpyrimidine-4,6-diamine
—— (5-methyl-4-nitro-1H-pyrazol-3-yl)-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone —— C16H18N4O3
(5-methyl-4-nitro-1H-pyrazol-3-yl)-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]methanone
—— 5-methoxy-3-methyl-N-[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1-benzofuran-2-carboxamide —— C18H20N4O3
5-methoxy-3-methyl-N-[(6S)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1-benzofuran-2-carboxamide
—— 5-methoxy-3-methyl-N-[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1-benzofuran-2-carboxamide —— C18H20N4O3
5-methoxy-3-methyl-N-[(6R)-3-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]-1-benzofuran-2-carboxamide
—— 5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ium-1-ylethyl]thiophene-2-sulfonamide —— C18H25ClN3O2S2+
5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ium-1-ylethyl]thiophene-2-sulfonamide
—— 5-chloro-N-[(2S)-2-(dimethylamino)-2-[4-(dimethylamino)phenyl]ethyl]thiophene-2-sulfonamide —— C16H22ClN3O2S2
5-chloro-N-[(2S)-2-(dimethylamino)-2-[4-(dimethylamino)phenyl]ethyl]thiophene-2-sulfonamide
—— (5S)-N-[1-(2-methoxyethyl)indol-5-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide —— C21H21N3O3
(5S)-N-[1-(2-methoxyethyl)indol-5-yl]-3-phenyl-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5,6-dimethyl-4-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine —— C17H20N4S2
5,6-dimethyl-4-[(2R)-2-(4-methyl-1,3-thiazol-2-yl)piperidin-1-yl]thieno[2,3-d]pyrimidine
—— (5-chlorothiophen-2-yl)-[(3R)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone —— C17H18ClNO2S
(5-chlorothiophen-2-yl)-[(3R)-3-[[3-(hydroxymethyl)phenyl]methyl]pyrrolidin-1-yl]methanone
—— (5-ethyl-1,3-oxazol-4-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H23N7O2
(5-ethyl-1,3-oxazol-4-yl)-[(3R)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— 5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-(4-methylpiperazin-1-yl)ethyl]-2-methoxybenzamide —— C23H31ClN4O2
5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-(4-methylpiperazin-1-yl)ethyl]-2-methoxybenzamide
—— 5-cyano-N-[2-[(2R)-4-methyl-2-phenylpiperazin-1-yl]ethyl]pyridine-2-carboxamide —— C20H23N5O
5-cyano-N-[2-[(2R)-4-methyl-2-phenylpiperazin-1-yl]ethyl]pyridine-2-carboxamide
—— 5-[2-oxo-2-[3-oxo-2-[[(2S)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]ethyl]-1H-pyrimidine-2,4-dione —— C20H28N4O5
5-[2-oxo-2-[3-oxo-2-[[(2S)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]ethyl]-1H-pyrimidine-2,4-dione
—— 5-[2-oxo-2-[3-oxo-2-[[(2R)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]ethyl]-1H-pyrimidine-2,4-dione —— C20H28N4O5
5-[2-oxo-2-[3-oxo-2-[[(2R)-oxolan-2-yl]methyl]-2,9-diazaspiro[5.5]undecan-9-yl]ethyl]-1H-pyrimidine-2,4-dione
—— (5S)-9-(1-methylimidazol-4-yl)sulfonyl-2-oxa-9-azaspiro[4.5]decane —— C12H19N3O3S
(5S)-9-(1-methylimidazol-4-yl)sulfonyl-2-oxa-9-azaspiro[4.5]decane
—— 5-bromo-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-morpholin-4-ylethyl]furan-2-carboxamide —— C19H24BrN3O3
5-bromo-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-morpholin-4-ylethyl]furan-2-carboxamide
—— 5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-(4-methylpiperazine-1,4-diium-1-yl)ethyl]-2-methoxybenzamide —— C23H33ClN4O2+2
5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-(4-methylpiperazine-1,4-diium-1-yl)ethyl]-2-methoxybenzamide
—— (5-ethyl-1,3-oxazol-4-yl)-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H23N7O2
(5-ethyl-1,3-oxazol-4-yl)-[(3S)-3-[5-(imidazol-1-ylmethyl)-4-methyl-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— 5-ethyl-3-[(3S)-3-methyl-3-phenylpiperidin-1-yl]-1,2,4-oxadiazole —— C16H21N3O
5-ethyl-3-[(3S)-3-methyl-3-phenylpiperidin-1-yl]-1,2,4-oxadiazole
—— (5R)-9-(1-methylimidazol-4-yl)sulfonyl-2-oxa-9-azaspiro[4.5]decane —— C12H19N3O3S
(5R)-9-(1-methylimidazol-4-yl)sulfonyl-2-oxa-9-azaspiro[4.5]decane
—— 5-ethyl-4-N-[(2S)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidine-2,4-diamine —— C18H26N6
5-ethyl-4-N-[(2S)-2-piperidin-1-yl-2-pyridin-3-ylethyl]pyrimidine-2,4-diamine
—— 5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ium-1-ylethyl]-2-nitrobenzamide —— C21H26ClN4O3+
5-chloro-N-[(2S)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ium-1-ylethyl]-2-nitrobenzamide
—— 5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-morpholin-4-ium-4-ylethyl]-2-methoxybenzamide —— C22H29ClN3O3+
5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-morpholin-4-ium-4-ylethyl]-2-methoxybenzamide
—— 5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ium-1-ylethyl]-2-methoxybenzamide —— C22H29ClN3O2+
5-chloro-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-pyrrolidin-1-ium-1-ylethyl]-2-methoxybenzamide
—— 5-ethyl-3-[(3R)-3-methyl-3-phenylpiperidin-1-yl]-1,2,4-oxadiazole —— C16H21N3O
5-ethyl-3-[(3R)-3-methyl-3-phenylpiperidin-1-yl]-1,2,4-oxadiazole
—— 5-bromo-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-morpholin-4-ylethyl]furan-2-carboxamide —— C19H24BrN3O3
5-bromo-N-[(2R)-2-[4-(dimethylamino)phenyl]-2-morpholin-4-ylethyl]furan-2-carboxamide
—— (5S)-1-(2-methoxyethyl)-5-[2-[(3-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]piperidin-2-one —— C18H24N4O3
(5S)-1-(2-methoxyethyl)-5-[2-[(3-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]piperidin-2-one
—— (5R)-9-[(2-morpholin-4-yl-1,3-thiazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decane —— C16H25N3O2S
(5R)-9-[(2-morpholin-4-yl-1,3-thiazol-5-yl)methyl]-2-oxa-9-azaspiro[4.5]decane