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—— (5R)-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one —— C18H23N3O2
(5R)-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one
—— (5-chloro-2-fluorophenyl)-[(3R)-3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methanone —— C16H21ClFNO3
(5-chloro-2-fluorophenyl)-[(3R)-3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methanone
—— (5R)-7-(cyclopropylmethyl)-2-(2,3-dimethoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O4
(5R)-7-(cyclopropylmethyl)-2-(2,3-dimethoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bR)-9-bromo-5-cyclohexyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H23BrN2O
(5S,10bR)-9-bromo-5-cyclohexyl-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5,6-dimethyl-2-[2-[(3R)-3-methyl-3-phenylpiperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C20H25N3O2
5,6-dimethyl-2-[2-[(3R)-3-methyl-3-phenylpiperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— (5R)-1-cycloheptyl-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H27N3O2
(5R)-1-cycloheptyl-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S)-2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O3
(5S)-2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [(5S,10bR)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-methylphenyl)methanone —— C25H22N2O2
[(5S,10bR)-2-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-(4-methylphenyl)methanone
—— (5S,10bR)-9-bromo-2-(4-methylphenyl)-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H21BrN2O
(5S,10bR)-9-bromo-2-(4-methylphenyl)-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(cyclohexylmethyl)piperidin-2-one —— C21H25N5O2
(5R)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(cyclohexylmethyl)piperidin-2-one
—— (5R)-7-methyl-6-oxo-N-(2-phenylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide —— C22H25N3O2
(5R)-7-methyl-6-oxo-N-(2-phenylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-5-phenyl-3,4,5,6-tetrahydro-2H-benzo[a]phenanthridin-1-one —— C23H19NO
(5S)-5-phenyl-3,4,5,6-tetrahydro-2H-benzo[a]phenanthridin-1-one
—— (5R,10bS)-9-bromo-2-(4-chlorophenyl)-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C19H18BrClN2O
(5R,10bS)-9-bromo-2-(4-chlorophenyl)-5-propyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-tert-butyl-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine —— C11H18N6O
5-tert-butyl-N-[(1S)-1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
—— (5R)-9-[(1-benzylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C19H23N3O2
(5R)-9-[(1-benzylpyrazol-4-yl)methyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— [(5R)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C19H23N5O2
[(5R)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]-[4-[1-(pyridin-3-ylmethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (5S)-7-(cyclopropylmethyl)-2-(2,3-dimethoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one —— C21H28N2O4
(5S)-7-(cyclopropylmethyl)-2-(2,3-dimethoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(2-chlorophenyl)furan-2-yl]-[(2R)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone —— C16H14ClNO3
[5-(2-chlorophenyl)furan-2-yl]-[(2R)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]methanone
—— (5R)-1-cyclopentyl-5-(2-methyl-1,2,4-triazol-3-yl)piperidin-2-one —— C13H20N4O
(5R)-1-cyclopentyl-5-(2-methyl-1,2,4-triazol-3-yl)piperidin-2-one
—— 5-[(3R)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1H-pyridin-2-one —— C20H22N2O4
5-[(3R)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1H-pyridin-2-one
—— [(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone —— C16H24N2O3S
[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(2-propan-2-yl-1,3-thiazol-4-yl)methanone
—— (5S)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H25N5O2
(5S)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C18H25N5O2
(5S)-2-(2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H23FN4O3
(5S)-2-(3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]-6-methylpyridin-2-amine —— C16H18N2O
5-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]-6-methylpyridin-2-amine
—— (5R)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H25N5O2
(5R)-7-(cyclobutylmethyl)-2-[2-(1,2,4-triazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H29N3O3
(5R)-2-[3-(2-methyl-6-oxopyridin-1-yl)propanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R,6R)-6-methyl-3-(2-oxo-2-thiophen-2-ylethyl)-1,3-diazaspiro[4.5]decane-2,4-dione —— C15H18N2O3S
(5R,6R)-6-methyl-3-(2-oxo-2-thiophen-2-ylethyl)-1,3-diazaspiro[4.5]decane-2,4-dione
—— (5S)-1-cycloheptyl-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C17H27N3O2
(5S)-1-cycloheptyl-5-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— 5-[(3S)-3-ethyl-4-propan-2-ylpiperazine-1-carbonyl]-2-(4-methylphenyl)-1H-pyrimidin-6-one —— C21H28N4O2
5-[(3S)-3-ethyl-4-propan-2-ylpiperazine-1-carbonyl]-2-(4-methylphenyl)-1H-pyrimidin-6-one
—— (5S)-7-methyl-6-oxo-N-(2-phenylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide —— C22H25N3O2
(5S)-7-methyl-6-oxo-N-(2-phenylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
—— (5S)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3S
(5S)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C16H24N4O3S
(5R)-2-[2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1H-pyridin-2-one —— C20H22N2O4
5-[(3S)-3-(1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1H-pyridin-2-one
—— (5R)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H27N3O3
(5R)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-chloro-2-fluorophenyl)-[(3S)-3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methanone —— C16H21ClFNO3
(5-chloro-2-fluorophenyl)-[(3S)-3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methanone
—— (5R)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one —— C19H31N3O2
(5R)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one
—— (5R)-5-(2-bromophenyl)-3,4,5,6-tetrahydro-2H-benzo[a]phenanthridin-1-one —— C23H18BrNO
(5R)-5-(2-bromophenyl)-3,4,5,6-tetrahydro-2H-benzo[a]phenanthridin-1-one
—— (5S)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C22H27N3O3
(5S)-7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(3R)-3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)-1H-pyrimidin-6-one —— C22H20FN3O2
5-[(3R)-3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)-1H-pyrimidin-6-one
—— (5R)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one —— C17H26N4O4
(5R)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
—— (5S)-7-(cyclopropylmethyl)-2-(4,4,4-trifluorobutanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H23F3N2O2
(5S)-7-(cyclopropylmethyl)-2-(4,4,4-trifluorobutanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(2,5-dimethylpyrazol-3-yl)methyl]-5-methylpiperidin-2-one —— C20H25N3O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-1-[(2,5-dimethylpyrazol-3-yl)methyl]-5-methylpiperidin-2-one
—— (5S)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one —— C17H26N4O4
(5S)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
—— (5S)-1-[3-(1H-imidazol-2-yl)propyl]-5-methyl-5-phenylpiperidin-2-one —— C18H23N3O
(5S)-1-[3-(1H-imidazol-2-yl)propyl]-5-methyl-5-phenylpiperidin-2-one
—— (5-methylpyrazin-2-yl)-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H22N8O
(5-methylpyrazin-2-yl)-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (5R)-2-[2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C16H25N5O3S
(5R)-2-[2-[(5-ethyl-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H23FN4O3
(5R)-2-(3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H24N2O3
(5S)-2-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one —— C19H31N3O2
(5S)-1-[[3-(2-methoxyethyl)imidazol-4-yl]methyl]-5-methyl-5-(4-methylpent-3-enyl)piperidin-2-one