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—— 5-(2-Acetyl-phenyl)-thiophene-2-carbaldehyde —— C13H10O2S
5-(2-Acetyl-phenyl)-thiophene-2-carbaldehyde
—— (5-methoxyfuran-2-yl)-[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H22N6O3
(5-methoxyfuran-2-yl)-[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (5S)-2-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C17H26N4O2S
(5S)-2-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-9-(2-methoxyphenyl)sulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C16H23NO5S
(5R)-9-(2-methoxyphenyl)sulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5S)-9-(2-methoxyphenyl)sulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C16H23NO5S
(5S)-9-(2-methoxyphenyl)sulfonyl-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-1-cyclopentyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C15H23N3O2
(5R)-1-cyclopentyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5S,10bS)-9-chloro-2,5-bis(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H21ClN2O3
(5S,10bS)-9-chloro-2,5-bis(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5,8-dimethyl-2-[[[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]amino]methyl]-1H-quinolin-4-one —— C23H29N3O3
5,8-dimethyl-2-[[[(2S)-2-(5-methylfuran-2-yl)-2-morpholin-4-ylethyl]amino]methyl]-1H-quinolin-4-one
—— (5S)-1-cyclopentyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one —— C15H23N3O2
(5S)-1-cyclopentyl-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
—— (5R)-4-(5,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one —— C23H21N3O3
(5R)-4-(5,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)-5-phenyl-3,5-dihydro-1H-1,4-benzodiazepin-2-one
—— (5R,10bS)-9-chloro-2-phenyl-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C19H19ClN2O
(5R,10bS)-9-chloro-2-phenyl-5-propan-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5-methoxyfuran-2-yl)-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone —— C18H22N6O3
(5-methoxyfuran-2-yl)-[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methanone
—— (5S)-7-cyclohexyl-2-(cyclopentanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H32N2O2
(5S)-7-cyclohexyl-2-(cyclopentanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C16H25N5O2S
(5S)-2-[2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-propyl-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24N4O2S
(5R)-7-propyl-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-9-(3-indazol-1-ylpropyl)-2-oxa-9-azaspiro[4.5]decan-8-one —— C18H23N3O2
(5S)-9-(3-indazol-1-ylpropyl)-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5R,10bS)-2-(4-fluorophenyl)-5-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H19FN2O
(5R,10bS)-2-(4-fluorophenyl)-5-(4-methylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C14H19F3N4O3
(5S)-7-(2-hydroxyethyl)-2-[[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(2-morpholin-4-yl-2-oxoethyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C17H29N3O3
(5S)-2-(2-morpholin-4-yl-2-oxoethyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bS)-5-(4-bromophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H15BrN2OS
(5S,10bS)-5-(4-bromophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 5-cyclopropyl-N-[(5R)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1H-pyrazole-3-carboxamide —— C21H28N6O2
5-cyclopropyl-N-[(5R)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1H-pyrazole-3-carboxamide
—— (5R)-7-(2-methoxyethyl)-2-(3-pyrazin-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O3
(5R)-7-(2-methoxyethyl)-2-(3-pyrazin-2-ylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-cyclohexyl-2-(cyclopentanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C20H32N2O2
(5R)-7-cyclohexyl-2-(cyclopentanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one —— C19H24N4O2S
(5S)-5-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one
—— (5S)-4-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one —— C19H23N3O3
(5S)-4-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
—— (5S)-7-(cyclobutylmethyl)-2-[2-(1-methylpyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H30N4O
(5S)-7-(cyclobutylmethyl)-2-[2-(1-methylpyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one —— C19H24N4O2S
(5R)-5-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-one —— C19H23N3O4S
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[[3-(methylsulfanylmethyl)-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-one
—— (5R)-7-(cyclopropylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H24N4O2S
(5R)-7-(cyclopropylmethyl)-2-(2-pyrimidin-2-ylsulfanylacetyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-1-ethyl-5-(3-phenylmethoxyazetidine-1-carbonyl)piperidin-2-one —— C18H24N2O3
(5S)-1-ethyl-5-(3-phenylmethoxyazetidine-1-carbonyl)piperidin-2-one
—— (5S)-7-(2-methoxyethyl)-2-(1-methyl-2-oxopyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O4
(5S)-7-(2-methoxyethyl)-2-(1-methyl-2-oxopyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-4-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one —— C19H23N3O3
(5R)-4-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
—— (5R)-2-[2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C16H25N5O2S
(5R)-2-[2-[(4-methyl-1,2,4-triazol-3-yl)sulfanyl]acetyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-ethyl-2-[[(2S)-piperidin-2-yl]methyl]pyridine —— C13H20N2
5-ethyl-2-[[(2S)-piperidin-2-yl]methyl]pyridine
—— (5R)-7-(cyclobutylmethyl)-2-[2-(1-methylpyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one —— C19H30N4O
(5R)-7-(cyclobutylmethyl)-2-[2-(1-methylpyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-chloro-3-[(3R)-3-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-4,6-dimethyl-1H-pyridin-2-one —— C18H23ClN4O2
5-chloro-3-[(3R)-3-(1-ethylimidazol-2-yl)piperidine-1-carbonyl]-4,6-dimethyl-1H-pyridin-2-one
—— (5R)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O2
(5R)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O2
(5S)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5-fluoro-1,3-dimethylindol-2-yl)-[(3R)-3-(piperidin-1-ylmethyl)piperidin-1-yl]methanone —— C22H30FN3O
(5-fluoro-1,3-dimethylindol-2-yl)-[(3R)-3-(piperidin-1-ylmethyl)piperidin-1-yl]methanone
—— 5-[(2R)-oxolan-2-yl]-N-[[3-(pyrrolidin-1-ylmethyl)phenyl]methyl]thiophene-2-carboxamide —— C21H26N2O2S
5-[(2R)-oxolan-2-yl]-N-[[3-(pyrrolidin-1-ylmethyl)phenyl]methyl]thiophene-2-carboxamide
—— (5R)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one —— C16H22N2O2
(5R)-2-[(E)-3-(furan-2-yl)-2-methylprop-2-enyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(cyclohexylmethyl)piperidin-2-one —— C21H25N5O2
(5S)-5-[3-(3H-benzimidazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(cyclohexylmethyl)piperidin-2-one
—— 5-[(3S)-3-(hydroxymethyl)-3-prop-2-enylpiperidine-1-carbonyl]-1-methylpyrimidine-2,4-dione —— C15H21N3O4
5-[(3S)-3-(hydroxymethyl)-3-prop-2-enylpiperidine-1-carbonyl]-1-methylpyrimidine-2,4-dione
—— (5S)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C12H13N5O2
(5S)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-ethyl-4-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidine-2,4-diamine —— C14H19N5O
5-ethyl-4-N-[(2S)-2-pyridin-3-yloxypropyl]pyrimidine-2,4-diamine
—— (5S)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C14H22N4O2S
(5S)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-cyclopropyl-N-[(5S)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1H-pyrazole-3-carboxamide —— C21H28N6O2
5-cyclopropyl-N-[(5S)-7,7-dimethyl-2-morpholin-4-yl-6,8-dihydro-5H-quinazolin-5-yl]-1H-pyrazole-3-carboxamide
—— (5-fluoro-1,3-dimethylindol-2-yl)-[(3S)-3-(piperidin-1-ylmethyl)piperidin-1-yl]methanone —— C22H30FN3O
(5-fluoro-1,3-dimethylindol-2-yl)-[(3S)-3-(piperidin-1-ylmethyl)piperidin-1-yl]methanone
—— (5R)-2-[1-(2-fluorophenyl)cyclopropanecarbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C21H27FN2O2
(5R)-2-[1-(2-fluorophenyl)cyclopropanecarbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one —— C14H22N4O2S
(5R)-2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one