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—— (5R)-7-(2-methoxyethyl)-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O4
(5R)-7-(2-methoxyethyl)-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[(2-aminopyrimidin-5-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C18H27N5O2
(5S)-2-[(2-aminopyrimidin-5-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(5-methylfuran-2-yl)-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide —— C21H24N4O2
5-(5-methylfuran-2-yl)-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide
—— 5-[[(2R)-2-ethylhexanoyl]amino]-2-(4-methylpiperidin-1-yl)-N-propan-2-ylbenzamide —— C24H39N3O2
5-[[(2R)-2-ethylhexanoyl]amino]-2-(4-methylpiperidin-1-yl)-N-propan-2-ylbenzamide
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 4-(2,5-dimethylphenyl)-4-oxobutanoate —— C19H18N2O4S
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 4-(2,5-dimethylphenyl)-4-oxobutanoate
—— (5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1-methylpiperidin-4-yl)piperidin-2-one —— C20H28N2O3
(5R)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1-methylpiperidin-4-yl)piperidin-2-one
—— 5-[(S)-[4-(5-ethylfuran-2-yl)triazol-1-yl]-phenylmethyl]-1,3,4-thiadiazol-2-amine —— C17H16N6OS
5-[(S)-[4-(5-ethylfuran-2-yl)triazol-1-yl]-phenylmethyl]-1,3,4-thiadiazol-2-amine
—— (5R)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O
(5R)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2R)-oxolan-2-yl]-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)thiophene-2-carboxamide —— C16H16N4O2S
5-[(2R)-oxolan-2-yl]-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)thiophene-2-carboxamide
—— (5S)-2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24ClN5O2
(5S)-2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(4-Methoxyphenyl)-1,3-oxazol-4-yl]-[4-(pyridin-3-ylmethyl)piperazin-4-ium-1-yl]methanone —— C21H23N4O3+
[5-(4-Methoxyphenyl)-1,3-oxazol-4-yl]-[4-(pyridin-3-ylmethyl)piperazin-4-ium-1-yl]methanone
—— (5S)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one —— C20H28N4O
(5S)-2-[(7-methylimidazo[1,2-a]pyridin-2-yl)methyl]-7-propan-2-yl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1-methylpiperidin-4-yl)piperidin-2-one —— C20H28N2O3
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1-methylpiperidin-4-yl)piperidin-2-one
—— (5R)-2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C17H24ClN5O2
(5R)-2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-methyl-2-(1,4,6-trimethyl-2-oxopyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O3
(5R)-7-methyl-2-(1,4,6-trimethyl-2-oxopyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— 5-(5-methylfuran-2-yl)-N-[(1R)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide —— C21H24N4O2
5-(5-methylfuran-2-yl)-N-[(1R)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-pyrazole-3-carboxamide
—— (5S)-7-(2-methoxyethyl)-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O4
(5S)-7-(2-methoxyethyl)-2-[2-(2-oxopyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-(2-chlorophenyl)-N-[(1R)-1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]furan-2-carboxamide —— C17H16ClN3O3
5-(2-chlorophenyl)-N-[(1R)-1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]furan-2-carboxamide
—— 5-[(2S)-oxolan-2-yl]-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)thiophene-2-carboxamide —— C16H16N4O2S
5-[(2S)-oxolan-2-yl]-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)thiophene-2-carboxamide
—— (5S)-2-amino-5-[[4-(trifluoromethoxy)phenyl]methyl]-1,3-thiazol-4-one —— C11H9F3N2O2S
(5S)-2-amino-5-[[4-(trifluoromethoxy)phenyl]methyl]-1,3-thiazol-4-one
—— (5S)-9-[(5-ethylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H26N2O2
(5S)-9-[(5-ethylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (5R)-2-(1,3-benzothiazol-2-yl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one —— C19H25N3O2S
(5R)-2-(1,3-benzothiazol-2-yl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(oxan-4-yl)-2-[2-(triazol-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C17H25N5O3
(5R)-7-(oxan-4-yl)-2-[2-(triazol-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(R)-[4-(5-ethylfuran-2-yl)triazol-1-yl]-phenylmethyl]-1,3,4-thiadiazol-2-amine —— C17H16N6OS
5-[(R)-[4-(5-ethylfuran-2-yl)triazol-1-yl]-phenylmethyl]-1,3,4-thiadiazol-2-amine
—— (5R)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one —— C20H27N5O2
(5R)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one
—— (5R)-7-(cyclobutylmethyl)-2-[2-(4,5-dimethylimidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5R)-7-(cyclobutylmethyl)-2-[2-(4,5-dimethylimidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-[(4,6-dimethylpyrimidin-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5S)-2-[(4,6-dimethylpyrimidin-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one —— C20H27N5O2
(5S)-5-[3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)piperidin-2-one
—— (5R)-9-[2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H20F3N3O2
(5R)-9-[2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— 5-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]pyrazin-2-amine —— C14H15N3O
5-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]pyrazin-2-amine
—— (5R)-2-(4-chloro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H22ClN3O2
(5R)-2-(4-chloro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-2-[(4,6-dimethylpyrimidin-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C20H30N4O2
(5R)-2-[(4,6-dimethylpyrimidin-2-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(2-amino-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl)-1-cyclopentylpiperidin-2-one —— C17H24N4O2S
(5S)-5-(2-amino-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl)-1-cyclopentylpiperidin-2-one
—— 5-fluoro-N-methyl-2-[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidin-4-amine —— C17H22FN9
5-fluoro-N-methyl-2-[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyrimidin-4-amine
—— (5R)-2-[3-(4-hydroxyphenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H24N2O3
(5R)-2-[3-(4-hydroxyphenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-5-(2-amino-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl)-1-cyclopentylpiperidin-2-one —— C17H24N4O2S
(5R)-5-(2-amino-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl)-1-cyclopentylpiperidin-2-one
—— (5S)-2-(4-ethoxyphenyl)sulfonyl-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O4S
(5S)-2-(4-ethoxyphenyl)sulfonyl-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-7-methyl-2-(1,4,6-trimethyl-2-oxopyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H25N3O3
(5S)-7-methyl-2-(1,4,6-trimethyl-2-oxopyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
—— (5R)-7-(oxan-4-yl)-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one —— C18H26N4O2
(5R)-7-(oxan-4-yl)-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
—— [5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(3R)-3-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C19H23N5O3
[5-(5-methylfuran-2-yl)-1H-pyrazol-3-yl]-[(3R)-3-(3-propan-2-yl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (5S)-2-(4-aminopyrimidin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one —— C17H25N5O2
(5S)-2-(4-aminopyrimidin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
—— (5S,10bS)-5-(4-propan-2-ylphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H22N2OS
(5S,10bS)-5-(4-propan-2-ylphenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S)-9-[2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one —— C16H20F3N3O2
(5S)-9-[2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl]-2-oxa-9-azaspiro[4.5]decan-8-one
—— (5S)-2-[3-(4-hydroxyphenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C22H24N2O3
(5S)-2-[3-(4-hydroxyphenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— 5-[(2S)-oxolan-2-yl]-N-[(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)methyl]thiophene-2-carboxamide —— C16H15N5O3S
5-[(2S)-oxolan-2-yl]-N-[(3-pyrimidin-2-yl-1,2,4-oxadiazol-5-yl)methyl]thiophene-2-carboxamide
—— (5R)-2-(4-ethoxyphenyl)sulfonyl-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C17H24N2O4S
(5R)-2-(4-ethoxyphenyl)sulfonyl-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-2-(4-chloro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one —— C19H22ClN3O2
(5S)-2-(4-chloro-1-methylindole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
—— (5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(4-hydroxyphenyl)ethyl]-5-methylpiperidin-2-one —— C22H25NO4
(5S)-5-(1,3-benzodioxol-5-ylmethyl)-1-[2-(4-hydroxyphenyl)ethyl]-5-methylpiperidin-2-one
—— (5S)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one —— C20H26N4O3
(5S)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-(2-morpholin-4-ylethyl)piperidin-2-one
—— 5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[3-(pyridin-3-ylamino)propyl]-1,2-dihydropyrazole-3-carboxamide —— C18H19N5O2
5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[3-(pyridin-3-ylamino)propyl]-1,2-dihydropyrazole-3-carboxamide